Synthesis, anti-tuberculosis activity and QSAR study of 2,4-diarylquinolines and analogous polycyclic derivatives [PDF]
The multicomponent syntheses of 2,4-di-aryl-quinolines and analogous polycyclic derivatives as anti-tuberculosis agents were described. They were prepared via Beyer and Friedländer methods under microwave irradiation in short reaction times and good ...
Asís, Silvia Elizabeth +7 more
core +1 more source
Gas Chromatography-Mass Spectrometry Study of the Essential Oils of Schinus longifolia (Lindl.) Speg., Schinus fasciculata (Griseb.) I. M. Johnst., and Schinus areira L. [PDF]
The essential oil composition from the aerial parts of three Anacardiaceae growing in Bah¨ªa Blanca, Argentina was studied by gas chromatography and gas chromatography-mass spectrometry. The essential oils of S. longifolia and S.
Frontera, Maria Eugenia +3 more
core +1 more source
Bile acids: Lipase-catalyzed synthesis of new hyodeoxycholic acid derivatives [PDF]
In this work we present an efficient, environmentally friendly approach to the synthesis of a series of hyodeoxycholic acid derivatives applying Biocatalysis.
Baldessari, Alicia +3 more
core +1 more source
Volatiles from Subtropical Convolvulaceae That Interfere with Bacterial Cell-to-Cell Communication as Potential Antipathogenic Drugs [PDF]
Increasing chronic bacterial infections create an urgent need for new antimicrobial agents or strategies for their control. Targetingvirulence is one of the alternative approaches to find new medicines to treat persistent infections due to bacteria with ...
Arena, Mario Eduardo +5 more
core +4 more sources
Derivatives of grindelic acid: from a non-active natural diterpene to synthetic antitumor derivatives [PDF]
Using several reactions that include homologations and asymmetric epoxidations as well as Ugi and Huisgen couplings, we generated a small focused library of new derivatives from the labdane-type diterpene grindelic acid. These compounds were evaluated as
Chiaramello, Alejandra Ilda +7 more
core +3 more sources
Multicomponent synthesis of 4,4-dimethyl sterol analogues and their effect on eukaryotic cells [PDF]
Most sterols, such as cholesterol and ergosterol, become functional only after the removal of the two methyl groups at C-4 from their biosynthetic precursors.
Alonso, Fernando +7 more
core +1 more source
Chemoenzymatic Synthesis of Triazololactams Structurally Related to Pancratistatin [PDF]
Four tricyclic lactams that structurally resemble alkaloids with the pancratistatin skeleton were synthetized from bromobenzene by a chemoenzymatic strategy.
Bastida +48 more
core +1 more source
Gas Phase Structure and Reactivity of Doubly Charged Microhydrated Calcium(II)-Catechol Complexes Probed by Infrared Spectroscopy [PDF]
Doubly charged microhydrated adducts formed from catechol and calcium(II) were produced in the gas phase using electrospray ionization (ESI) appearing as the most important ions in the mass spectra recorded. The gas phase structures of [Ca(catechol)2(H2O)
Arroyo Mañez, Pau +3 more
core +1 more source
Radical Fluoroalkylation Reactions [PDF]
Recent protocols and reactions for catalytic radical perfluoroalkylations will be described. The production of perfluoroalkyl radicals (RF = CnF2n+1, n ≥ 2), which effect both addition and substitution reactions on organic substrates, can be realized ...
Barata Vallejo, Sebastian +2 more
core +1 more source
Optimization of β-cyclodextrin-based extraction of antioxidant and anti-browning activities from thyme leaves by response surface methodology [PDF]
Thyme (Thymus vulgaris) has been demonstrated to extend the shelf-life of food products, being also a potential source of bioactive compounds. The aim of this research was to optimize the ultrasound assisted extraction employing β-cyclodextrin aqueous ...
Buera, Maria del Pilar +4 more
core +1 more source

