Results 61 to 70 of about 878 (177)

Synthesis and Structural Studies of Aza Analogues of Functionalized Amino Acids:  New Anticonvulsant Agents

, 2016
We have reported that functionalized amino acids 1 display potent anticonvulsant activities in mice and rats, and that the activity resides primarily in the d-isomer.
Harold Kohn (1333722), J. P. Stables (3011676), Cécile Béguin (445447), Shridhar V. Andurkar (3011679)   +3 more
core   +1 more source

Submonomer Synthesis of A Hybrid Peptoid–Azapeptoid Library

, 2016
We recently reported efficient conditions for the synthesis of N-azapeptoid libraries via the typical submonomer strategy of peptoid synthesis but that substitutes N-acyl hydrazides for primary amines as submonomers.
Bani Kanta Sarma (2037217), Thomas Kodadek (61725)   +1 more
core   +1 more source

Estudo da síntese espectros I.V. e atividade farmacobiológica de 1-acil-4-aril-tiosemicarbazidas e triazóis 3,4,5-trissubstituídos [PDF]

, 1987
Dissertação (mestrado) - Universidade Federal de Santa Catarina, Curso de Pós-Graduação em Físico ...
Peres, Marize Terezinha Lopes Pereira
core  

Design, Synthesis and Biological Activities of (Thio)Urea Benzothiazole Derivatives. [PDF]

Int J Mol Sci, 2023
Mendieta-Wejebe JE, Rosales-Hernández MC, Padilla-Martínez II, García-Báez EV, Cruz A.   +4 more
europepmc   +1 more source

Solid-Phase Synthesis of Hybrid 2,5-Diketopiperazines Using Acylhydrazide, Carbazate, Semicarbazide, Amino Acid, and Primary Amine Submonomers

, 2020
We report the solid-phase synthesis of N,N′-di­(acylamino)-2,5-diketopiperazine, an acylhydrazide-based conformationally rigid 2,5-DKP scaffold having exocyclic N–N bonds.
Abdur Rahim (5699147), Kalpita Baruah (8435520), Bani Kanta Sarma (2037217), Jugal Kishore Rai Deka (8435523), Biswajit Sahariah, Jugal Kishore Rai Deka, Abdur Rahim, Kalpita Baruah, Biswajit Sahariah (5699150), Bani Kanta Sarma   +9 more
core   +1 more source

di‐π‐methane rearrangement of benzonorbornadiene system

, 1998
The [4 + 2] cycloadduct 17 of 2,3-dimethylidene-1,2,3,4-tetrahydro-1,3-methanonaphthalene and 4-phenyl-4H-1,2,4-triazole-3,5-dione (PTAD) was subjected to a tripler-sensitized di-pi-methane rearrangement.
Altundas, ALİYE, Aliye Altundaş, Akbulut, N, Akbulut, Nihat, BALCI, M, Balcı, Metin, Nihat Akbulut, Metin Balci, Altundas, A   +8 more
core   +1 more source

Manipulation of N,O-Nucleophilicity:  Efficient Formation of 4-N-Substituted 2,4-Dihydro-3H-1,2,4-Triazolin-3-ones

, 2016
A new efficient two-step synthesis of 2,4-dihydro-3H-1,2,4-triazolin-3-ones (triazolinones) from readily available amines is reported. Our novel conditions using hexamethyl disilazane, bromotrimethylsilane, and a catalytic amount of ammonium sulfate ...
Xianhai Huang (2026387), Dong Xiao (162830), Neng-Yang Shih (1834609), Anandan Palani (1930282), Robert Aslanian (1811806)   +4 more
core   +1 more source

Synthesis and anti-microbial activity of (Z)-4-(4-substituted-thiazol-2-yl)-1-(2-oxoindolin-3-ylidene) semicarbazide and its derivatives

, 2010
1117-11263-[(2S)-3-Acetyl-5-amino-N-(4-substituted-thiazol-2-yl)2,3-dihydro-1,3,4-oxadiazol-2-yl]-indolin-2-yl acetates, 1-{N-[(2R)-2-(-2-oxoindolin-3-ylidene)-4-oxo-1,3-thiazolidin-3-yl]-3-(4-substituted-thiazol-2yl)ureas, N-(4-substituted-thiazol-2 ...
Basavarajaiah, S M, Mruthyunjayaswamy, B H M   +1 more
core  

Synthesis of 1-benzyl-6-azauracil derivatives, chlorinated in the nucleus

, 1981
Glyoxylic acid 2-benzylsemicarbazone derivatives, chlorinated in the aromatic nucleus (Ia-Id) were prepared either by reaction of glyoxylic acid semicarbazone with the corresponding benzyl chlorides or by treatment of benzylidene semicarbazide with ...
Petr Bedrník, Jiří Gut, Venuše Sedláčková, Bohumil Ševčík, Alois Nováček, Bohumír Vondráček   +5 more
core   +1 more source

Pathway complexity in fibre assembly: from liquid crystals to hyper-helical gelmorphs. [PDF]

Chem Sci, 2023
Contreras-Montoya R, Smith JP, Boothroyd SC, Aguilar JA, Mirzamani M, Screen MA, Yufit DS, Robertson M, He L, Qian S, Kumari H, Steed JW.   +11 more
europepmc   +1 more source