Results 51 to 60 of about 806 (175)

Synthesis and antimicrobial properties of new 4-(alkylidene/arylidene)-amino-5-(2-furanyl)-2,4-dihydro-3H-1,2,4-triazole-3-thiones and 6-aryl-3-(2-furanyl)-7H-1,2,4-triazolo[3,4-b][1,3,4]thiadiazines

, 2021
A series of 4-(alkylidene/arylidene)amino-5-(2-furanyl)-2,4-dihydro-3H-1,2,4-triazole-3-thiones (2) and 6-aryl-3-(2-furanyl)-7H-1,2,4-triazolo[3,4-b][1,3,4] thiadiazines (3) were synthesized.
Ulusoy, Nuray, Kiraz, M, Kiraz, Muammer, Sanis, GO, Ergenc, N, Ötük-Sanış, Gülten, Çapan, Gültaze, Capan, G, Ulusoy, N, Ergenç, Nedime   +9 more
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Studies on Chemical Entities of Therapeutic Interest [PDF]

, 2011
Not ...
Dodiya, Bhavesh L.
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Synthesis of Novel Bibrachial Lariat Ethers (BiBLEs) Containing [1,2,4]Triazolo[3,4-b][1,3,4]Thiadiazines [PDF]

, 2015
A practical and regioselective method for the synthesis of cis-diastereomers of bibrachial lariat ethers (BiBLEs) bearing ester and amide groups is reported.
Ebrahimi, S
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Thiazolyl-thiadiazines as Beta Site Amyloid Precursor Protein Cleaving Enzyme‑1 (BACE-1) Inhibitors and Anti-inflammatory Agents: Multitarget-Directed Ligands for the Efficient Management of Alzheimer’s Disease

, 2018
Alzheimer’s disease (AD) is associated with multiple neuropathological events including β-site amyloid precursor protein cleaving enzyme-1 (BACE-1) inhibition and neuronal inflammation, ensuing degeneracy, and death to neuronal cells.
Kamala K. Vasu (5205158), Rajesh D. Das (5205173), Nirupa B. Panchal (5205152), Manish Nivsarkar (5205170), Sneha R. Sagar (5205155), Devendra Pratap Singh (5205167), Vasudevan Sudarsanam (5205161), Dhaivat H. Pandya (5205164)   +7 more
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The Acid and/or Thermal Mediated Ring Contraction of 4H‑1,2,6-Thiadiazines To Afford 1,2,5-Thiadiazoles

, 2016
A near-quantitative acid and/or thermal mediated ring contraction of 3′,5′-diarylspiro­(benzo­[d]­[1,3]­dioxole-2,4′-[1,2,6]­thiadiazines) affords 3-aryl-4-(2-arylbenzo­[d]­[1,3]­dioxol-2-yl)-1,2,5-thiadiazoles.
Andreas Kourtellaris (1693780), Panayiotis A. Koutentis (1278807), Andreas S. Kalogirou (1546180)   +2 more
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Molecular Iodine Promoted Divergent Synthesis of Benzimidazoles, Benzothiazoles, and 2‑Benzyl-3-phenyl-3,4-dihydro‑2H‑benzo[e][1,2,4]thiadiazines

, 2016
An unprecedented formation of a new class of 2-benzyl-3-phenyl-3,4-dihydro-2H-benzo­[e]­[1,2,4]­thiadiazines has been discovered during the course of benzimidazole and benzothiazole synthesis, through the molecular iodine-mediated oxidative cyclization ...
Gunaganti Naresh (1667257), Tadigoppula Narender (1667254), Ruchir Kant (1433839)   +2 more
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3-Substituted-6-aryl-7 -thioaryloxy-s-triazolo[ 3,4-b ][ 1 ,3,4 ]thiadiazines and their corresponding Sulphones as Potential Antimicrobial and Antiparasitic Derivatives

, 1993
Department of Chemistry, THe Institute of Science, 15 Madam Cama Road, Bombay-400 032 Manuscript received 26 August 1991, revised 14 September 1992, accepted 12 November 1992 3-Substituted-6-aryl-7 -thioaryloxy-s-triazolo[ 3,4-b ][ 1 ,3,4 ]thiadiazines
M.S. CHANDE, B. M. KARNIK
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Identifying potential candidates for donor-acceptor copolymers on a series of 4H-1,2,6-thiadiazines: An electrochemical approach

, 2013
A series of synthesized small organic molecules based on the 4H-1,2,6-thiadiazine moiety are studied using electrochemistry, to probe their potential as comonomer building blocks for solar-absorbing polymers for organic solar cells.
Choulis, Stelios A., Ioannidou, Heraklidia A., Koutentis, Panayiotis A., Economopoulos, Solon P.   +3 more
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Synthesis and antimicrobial activity of 1,3,5-thiadiazines and their isomerism into 1,3,5-triazines

, 2005
638-642A series of 2,6-diphenylimino-4-(substituted)-benzylidene amino-1,3,5-thiadiazines 4a-g have been obtained by the basification of their hydrochlorides 3a-g, which are prepared by interaction of N-phenyl isocyanodichloride and 1-(substituted ...
Pradip P. Deohate, Deohate, Pradip P, Berad, B N, B. N. Berad   +3 more
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Synthesis of 3,6-disubstituted 7H-1,2,4-triazolo[3,4-b]-1,3,4-thiadiazines as novel analgesic/anti-inflammatory compounds

, 2009
In this study, a new class of 4-amino-3-substituted-1,2,4-triazole-5-thiones (1-4) and their corresponding condensed derivatives 3,6-disubstituted 7H-1,2,4-triazolo[3,4-bi-1,3,4-thiadiazines (1a-4c) were synthesized and evaluated for their analgesic/anti-
AYTAÇ, SAİT AYKUT, Uenuevar, Songuel, Goektas, Oezguer, KAYNAK, FİLİZ BETÜL, Aktay, Goeknur, Tozkoparan, BİRSEN   +5 more
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