Results 161 to 170 of about 11,765 (225)

Structure-Guided Optimization and Biological Validation of 1,3,4-Thiadiazole-Based SIRT2 Inhibitors Reinforcing Channel Entrance Interactions. [PDF]

Drug Dev Res
Aksel AB, Ozgencil F, Bakar-Ates F, Gunindi HB, Massarotti A, Ozkan E, Kaya SG, Gozelle M, Ozkan Y, Eren G.   +9 more
europepmc   +1 more source

Lipophilic Ligand Efficiency-Monitored Discovery of Potent, Achiral, and Bioavailable Apo-IDO1 Inhibitors. [PDF]

ACS Med Chem Lett
Kazmierski WM, Miriyala N, De la Rosa M, Miller J, Gentry ZO, Samano V, Catalano J, Chong PY, Wang F, Price DJ, Basilla J, Mebrahtu M, Wang L, Shewchuk L, Matico R, Dunham R.   +15 more
europepmc   +1 more source

Synthesis and antifungal activity of thiadiazole-functionalized chitosan derivatives

Carbohydrate Research, 2013
A groups of novel water soluble chitosan derivatives containing 1,3,4-thiadiazole group were synthesized including 1,3,4-thiadiazole (TPCTS), 2-methyl-1,3,4-thiadiazole (MTPCTS), and 2-phenyl-1,3,4-thiadiazole (PTPCTS).
Qing Li, Zhanyong Guo, Guodong Gu
exaly   +2 more sources

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A 1,2,3-thiadiazole–1,2,3-thiadiazole rearrangement

J. Chem. Soc., Chem. Commun., 1983
During its preparation, 4-ethoxycarbonyl-5-diazomethyl-1,2,3-thiadiazole (4), undergoes a ring transformation into the isomeric structure (5), but when the ester function in (4) is replaced by a phenyl group, no isomerization is observed.
Gerrit L'abbé, Jean-Paul Dekerk, Martine Deketele   +2 more
openaire   +1 more source

The 1,2,5-Thiadiazoles

1968
Publisher Summary This chapter presents the review of organic and physical chemistry of monocyclic 1, 2, 5-thiadiazoles up to the early part of 1967. Reference is made to the 2, 1, 3-benzothiadiazoles and related compounds only as they contribute to the chemistry of the basic ring system. The 1, 2, 5-thiadiazole nucleus is numbered as in 4.
L M, Weinstock, P I, Pollak
openaire   +2 more sources

SYNTHESIS AND METHYLATION OF SOME 1,2,4-THIADIAZOLE-5-THIONES

Phosphorus, Sulfur and Silicon and the Related Elements, 1992
3,4-Disubstituted-1,2,4-thiadiazole-5(4H)-thiones (4) have been prepared by the treatment of 3,4-di-substituted-1,2,4-thiadiazole-5(4H)-ones (3) with P4S10.
Yaşar Dürüst, Hikmet Agirbas
exaly   +2 more sources

Microwave spectra of 1,3,4-thiadiazole and [34S]1,3,4-thiadiazole. Dipole moment of 1,3,4-thiadiazole

Journal of Molecular Spectroscopy, 1962
Abstract The microwave spectra of 1, 3, 4-thiadiazole (I) and [ 34 S] 1, 3, 4-thiadiazole (II) have been recorded in the 15,000–30,000 Mc/sec region. Twelve and ten transitions, respectively, were assigned. The rotational constants of (I) are, A = 8907.51 ± 0.10, B = 5569.27 ± 0.02, and C = 3424.80 ± 0.03 Mc/sec. For (II), A = 8908.15 ± 0.20,
Børge Bak, Daniel Christensen, Lise Hansen-Nygaard, Leif Lipschitz, John Rastrup-Andersen   +4 more
openaire   +1 more source

Thiadiazoles

Heterocycles containing nitrogen, oxygen and sulfur have been under investigation for a long time because of their important medicinal properties. The literature survey has described that thiadiazole moieties serve as analgesic, anti-inflammatory, anti-microbial activities, antihypertensive,anticancer, antituberculosis and vasodilator and this ...
G. Nagendra, D. N. Akshitha, H. S. Lalithamba, G. K. Prashanth   +3 more
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1,2,3‐Thiadiazoles

ChemInform, 2005
AbstractFor Abstract see ChemInform Abstract in Full Text.
D. J. Wilkins, P. A. Bradley
openaire   +1 more source