ANTIMICROBIAL INVESTIGATION AND BINDING MODE ANALYSIS OF SOME NEWLY SYNTHESIZED 4-AMINO-5-((ARYL SUBSTITUTED)-4H-1, 2, 4-TRIAZOLE-3-YL)-THIO LINKED HYDROXAMIC ACID DERIVATIVES [PDF]
, 2019 Objective: A series of 5-substituted-4-amino-1, 2, 4-triazole-linked hydroxamic acid derivatives have been synthesized and explored in vitro to evaluate antibacterial and antifungal activities.
BANERJEE, SUBHASIS +4 more
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Науковий вісник Львівського національного університету ветеринарної медицини та біотехнологій імені С.З. Ґжицького: Серія Ветеринарні наукиThe process of creating new medicines includes many stages that make it possible to use them in veterinary practice in the future. These tests guarantee the effectiveness and safety of newly synthesized compounds.
V. P. Martynyshyn, V. M. Semtsov
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Synthesis and Characterization of Novel Schiff Bases, N-Acyl and Diazetines Derived from 3-((5-hydrazinyl-4-phenyl-4H-1,2,4-triazol-3-yl)methyl)-1H-indole [PDF]
, 2014 This work involves synthesis of some new heterocyclic compounds including 1,3-diazetine. The new Schiff bases[VI]a-d derived from 3-((5-hydrazinyl-4-phenyl-4H-1,2,4-triazol-3-yl)methyl)-1H-indole [V] which was synthesized by refluxing 5-((1H-indol-3-yl ...
AL-Aliawi, Kadhim M. Lazim +2 more
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The synthesis of triazole derivatives on mushroom tyrosinase and their mechanisms [PDF]
, 2016 酪氨酸酶广泛的存在于各生物体内，其产物多巴醌能与氨基酸或者蛋白质聚合黑色素，该酶是合成黑色素的关键酶。然而黑色素的过量合成会引起雀斑、黄褐斑、老年斑等色素沉积性皮肤病，此外研究表明，酪氨酸酶还与帕金森综合症、昆虫蜕皮、果蔬褐变有密切关系。因此，控制酪氨酸酶活性的研究在农业、制药业及化妆品行业有重要开发价值。 4-氨基-3-肼基-5-巯基-1，2，4-三唑（AHMT）为五元氮杂环，是酰胺键的电子等排物，也具有潜在的配位键，而苯甲醛类衍生物为酪氨酸酶底物的类似物，可以竞争性抑制酶失活性 ...
喻枫
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Studies on Nitrogen Containing Heterocyclic Compounds as Bioactive Agents [PDF]
, 2011 Not ...
Vekariya, Piyush B.
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Regioselective ring opening of 2,2-dicyanooxiranes by 1,3-dinucleophiles in the presence of Lewis acids such as bismuth(III) nitrate pentahydrate [Bi(NO)·5HO] and zirconium(IV) chloride (ZrCl) [PDF]
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Corrosion Study of Mild Steel in Aqueous Sulfuric Acid Solution Using 4-Methyl-4H-1,2,4-Triazole-3-Thiol and 2-Mercaptonicotinic Acid-An Experimental and Theoretical Study. [PDF]
Front Chem, 2017 Mehmeti VV, Berisha AR.
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Rational design and synthesis of Co(ii), Ni(ii) and Cu(ii) complexes bearing 1,2,4-triazole scaffold for biological applications. [PDF]
RSC AdvHassoon AA +8 more
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Novel pyrazole-clubbed triazole scaffolds as promising inhibitors for carbon steel corrosion in sulfuric acid and as antibacterial agents: electrochemical and computational evaluation. [PDF]
BMC ChemBelal K +3 more
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