Results 51 to 60 of about 1,673 (99)
Palladium Catalyzed C–C Coupling Reactions of 3,5-Dichloro-4H-1,2,6-thiadiazin-4-one
, 2016 Palladium catalyzed Suzuki–Miyaura, Stille, and Sonogashira coupling reactions are reported for the electron-deficient heterocyclic scaffold 3,5-dichloro-4H-1,2,6-thiadiazin-4-one (1).
Heraklidia A. Ioannidou (1332144) +2 more
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3,5-Bis(4-dodecylthiophen-2-yl)-4H-1,2,6-thiadiazin-4-one
, 2012 3,5-Dichloro-4H-1,2,6-thiadiazin-4-one 1 reacts with (4-dodecylthiophen-2-yl)trimethylstannane 4 (2.2 equiv.) and Pd(Ph3P)2Cl2 (5 mol%) in acetonitrile at ca.
Heraklidia A. Ioannidou +1 more
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Synthesis of (R) and (S)-3-Chloro-5-(2,4-dimethylpiperazin-1-yl)-4H-1,2,6-thiadiazin-4-ones
, 2020 The reaction of 3,5-dichloro-4H-1,2,6-thiadiazin-4-one with (R) and (S)-1,3-dimethylpiperazines (1 equiv), in THF, at ca. 20 °C gives (R) and (S)-3-chloro-5-(2,4-dimethylpiperazin-1-yl)-4H-1,2,6-thiadiazin-4-ones in 70% and 68% yields, respectively.
Christopher Asquith +2 more
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Fungitoxicity of 6H-Pyrazolo[3,4-c] [1,2,5]thiadiazine 2,2-Dioxides
, 1990 A base‐promoted cyclisation of 4‐nitroso‐5‐benzylsulphonamidopyrazoles (VII) afforded 6H‐pyrazolo[3,4‐c][1,2,5]thiadiazine‐2,2‐dioxides (VIII). They were tested in vitro for antifungal activity against a series of phytopathogenic fungi of different ...
GIORI, Paolo +5 more
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Design and synthesis of matrix metalloproteinase inhibitors derived from a 6H-1,3,4-thiadiazine scaffold [PDF]
, 2001 Schröder J. Design and synthesis of matrix metalloproteinase inhibitors derived from a 6H-1,3,4-thiadiazine scaffold. Bielefeld (Germany): Bielefeld University; 2001.The discovery and optimization of a series of heterocyclic non-peptide matrix ...
Schröder, Jörg
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3-Chloro-5-(4-dodecylthiophen-2-yl)-4H-1,2,6-thiadiazin-4-one
, 2012 3-Chloro-5-trifluoromethanesulfonate-4H-1,2,6-thiadiazin-4-one 3 reacts with (4-dodecylthiophen-2-yl)trimethylstannane 5 (1 equiv.) in the presence of Pd(Ph3P)2Cl2 (5 mol%) in benzene at ca.
Heraklidia A. Ioannidou +1 more
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This dissertation involves the development of new synthetic methods for the preparation of various organosulfur compounds using solvent-based and solvent-free mechanochemical methods.
Passia, Marco Thomas
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Selective Stille Coupling Reactions of 3-Chloro-5-halo(pseudohalo)-4H-1,2,6-thiadiazin-4-ones
, 2016 A series of 3-chloro-5-halo(pseudohalo)-4H-1,2,6-thiadiazin-4-ones (halo/pseudohalo = Br, I, OTf) are prepared from 3,5-dichloro-4H-1,2,6-thiadiazin-4-one (3) in good yields.
Heraklidia A. Ioannidou (1332144) +2 more
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, 2013 A series of 2-substituted 2H-thieno[3,4-e][1,2,4]thiadiazin-3(4H)-one 1,1-dioxides (2), 2-substituted 2H-thieno[2,3-e][1,2,4]thiadiazin-3(4H)-one 1,1-dioxides (3), 2-substituted 4,6-dihydropyrazolo[4,3-e]-[1,2,4]thiadiazin- 3(2H)-one 1,1-dioxides (4), 2 ...
Arán, Vicente J. +2 more
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Postoperative analgesia by D-myo-inositol-1,2,6-trisphosphate in patients undergoing cholecystectomy
, 1998 D-myo-inositol-1,2,6-trisphosphate (1,2,6-IP3) possesses antiinflammatory properties, such as reduced eicosanoid synthesis and inhibition of inflammation-induced edema. These properties suggest possible analgesic effects.
Cassuto, Jean, +4 more
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