Results 41 to 50 of about 5,904 (191)

Stereoselective synthesis of fused tetrahydroquinazolines through one-pot double [3 + 2] dipolar cycloadditions followed by [5 + 1] annulation

Beilstein Journal of Organic Chemistry, 2016
The one-pot [3 + 2] cycloaddition of an azomethine ylide with a maleimide followed by another [3 + 2] cycloaddition of an azide with the second maleimide gives a 1,5-diamino intermediate which is used for a sequential aminomethylation reaction with ...
Xiaofeng Zhang, Kenny Pham, Shuai Liu, Marc Legris, Alex Muthengi, Jerry P. Jasinski, Wei Zhang   +6 more
doaj   +1 more source

Cristais líquidos termotrópicos calamíticos contendo o heterociclo [1,2,3]-triazol 1,4-dissubstituído [PDF]

, 2006
Dissertação (mestrado) - Universidade Federal de Santa Catarina, Centro de Ciências Físicas e Matemáticas. Programa de Pós-Graduação em QuímicaA síntese e as propriedades térmicas de cinco séries homólogas de compostos calamíticos lineares e não lineares,
Santos, Deise Maria Pereira de Oliveira
core  

1 : 3 Dipolar Cycloaddition of Benzonitrile Oxide on to Cinnamyl Arylamines

, 1971
1:3 Dipolar Cycloaddition of Benzonitrile Oxide on to Cinnamyl Arylamines.
Mohan, Suresh, J. S. Sandhu, Kumar, Baldev   +2 more
openaire   +2 more sources

Highly Enantio‐ and Diastereoselective Synthesis of Tetrahydrofuran Frameworks via Chiral Lewis Acid‐Catalyzed Formal [3+2] Cycloaddition of Allylsilanes

Angewandte Chemie International Edition, EarlyView.
The first catalytic asymmetric formal [3+2] cycloaddition of allylsilanes delivers cis‐2,5‐disubstituted tetrahydrofuran‐3‐ones that serve as versatile intermediates for the synthesis of diverse bioactive scaffolds. ABSTRACT A formal [3+2] cycloaddition via cyclization/1,2‐hydride shift initiated by nucleophilic attack of allylsilanes has been ...
Hosung Lee, Dong Kyu Kim, Pingshan Xin, Jin Won Lee, Terim Seo, Do Hyun Ryu   +5 more
wiley   +1 more source

Asymmetric 1,3-Dipolar Cycloadditions of Cyclic Stabilized Ylides Derived from Chiral 1,2-Amino Alcohols [PDF]

, 2006
International audienceThe use of structurally similar chiral non-racemic azomethine ylides, nitrones and azomethine imines derived from 1,2-aminol alcohols in asymmetric dipolar cycloadditions is reviewed.
Chauveau, Ariane, Bonin, Martine, Micouin, Laurent   +2 more
core   +1 more source

Synthesis of novel phosphorylated chrysin derivatives by 1, 3-dipolar cycloaddition reaction

Phosphorus, Sulfur, and Silicon and the Related Elements, 2016
Through 1,3-dipolar cycloaddition reaction, 1,4,5-trisubstituted-1,2,3-triazole and phosphate-containing chrysin derivatives were synthesized with high yields. The target compounds were characterized by 1H, 31P, 13C NMR spectroscopy and HRMS.
Shaohua Zhu, Zhang, Yan, Peipei Li, Wenzhu Bi, Xiaolan Chen, Yufen Zhao   +5 more
openaire   +1 more source

The Jekyll and Hyde Nature of Tetrazoles in Polymer Science: From Intrinsic Electronic Duality to Programmable Macromolecular Function

Angewandte Chemie International Edition, EarlyView.
Tetrazoles are reframed as substitution‐programmable heterocycles rather than static functional groups in polymer chemistry. By linking electronic identity to synthetic strategy and polymer architecture, this mini‐review establishes a design framework for translating tetrazole duality into predictable macromolecular function.
Meryem S. Akdemir, Hatice Mutlu
wiley   +1 more source

Synthesis and Biological Evaluation of Well‐Defined M6P(n)‐Modified Glycopeptides for Targeted Protein Degradation

Chemistry – A European Journal, EarlyView.
A synthetic methodology has been developed to prepare multifunctional M6P and M6Pn ligands of different valency. The glycopeptides were conjugated to cetuximab and then examined to mediate cellular uptake of fluorescently labeled EGFRvIII. Only cetuximab modified by glycopeptides having 3 or 6 M6P or M6Pn residues demonstrated greater uptake.
Patrycja Lenartowicz, Jan‐Willem H. Langenbach, Nataliia Voloshyna, David Aidukas, Arwin J. Brouwer, John A. W. Kruijtzer, Geert‐Jan Boons   +6 more
wiley   +1 more source

Novel (3+2) dipolar cycloadditions of pyridinium ylides [PDF]

, 2017
This thesis describes advances in novel (3+2) dipolar cycloadditions of pyridinium ylides, their reactions with electrophilic alkenes afford tetrahydroindolizines which can possess alkaloid-like scaffolds.
Tongue, Tom
core  

Studies in Conjugated lmines: Nucleophilic Additions and the 1 ,3-Dipolar Cycloadditions

, 1970
Studies in Conjugated lmines: Nucleophilic Additions and the 1 ,3-Dipolar ...
Singh, Nazar, P. S. Sethi
openaire   +1 more source