Etude par des méthodes quantiques et empiriques des relations SAR et QSAR dans des hétérocycles à intérêt médicinale [PDF]
La tuberculose (TB) demeure la première maladie infectieuse mortelle chez les adultes des pays en développement. Plus tôt, il a été rapporté qu'un certain nombre de 2, 5-disubstitués-1, 3, 4-oxadiazoles ont été conçus, synthétisés et criblés pour leur ...
Benbrahim, Imane
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Graph theoretical analysis, pharmacoinformatics and molecular docking investigation of Chalcone-Schiff base hybrids as Cyclin-Dependent kinase inhibitors [PDF]
One of the promising classes of compounds in medicinal chemistry and drug design is those with azomethine linkages. The Chalcone-Schiff base hybrids contain this linkage and some heteroatoms, which are versatile molecules, play a vital role in drug ...
Arivanantham, Sathishkumar +5 more
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Ammonium Formate-Pd/C as a New Reducing System for 1,2,4-Oxadiazoles. Synthesis of Guanidine Derivatives and Reductive Rearrangement to Quinazolin-4-Ones with Potential Anti-Diabetic Activity [PDF]
Paola Marzullo +5 more
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EX VIVO ANTICOAGULANT ACTIVITY OF 1, 3, 4-OXADIAZOLE DERIVATIVES [PDF]
Objective: The present medication for the management of arterial thromboembolism (ATE) disorders by anticoagulant therapy highlights its lacunae due to recurrent ATE episodes and indicates the need for better anticoagulant agents with clinical advantage ...
Gurupadayya, B. M., Vishwanathan, B.
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Synthesis and Antioxidant Characteristics of Novel Heterocyclic Derivatives from 2-Thiol-5-Phenyl-1,3,4-Oxadiazole Compounds [PDF]
The 1,3,4-Oxadiazole-bearing compounds are among the most attractive classes for researchers because of their biological processes. The study used a current show of quinazoline-4-one and oxazine-4-one derivatives (8-13) were synthesized.
Mohammed R. Ahmad, Sumaya J. Jamal
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Photophysical characterizations of 2-(4-biphenylyl)-5 phenyl-1,3,4-oxadiazole in restricted geometry [PDF]
Pabitra Kumar Paul +2 more
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5-(4-pyridinyl)-1,3,4-oxadiazole-2-thiol on gold: SAM Formation and electroactivity [PDF]
Tércio de F. Paulo +9 more
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Synthesis , Characterization , Antimicrobial New 2,2'-[(1E,2E)-ethane-1,2-diylidenedi(2E)hydrazin-1-yl-2-ylidene]bis (5-methyl-1,3,4-oxadiazole) and their transition metal complexes [PDF]
Transition metal complexes of new legend 2,2'-[(1E,2E)-ethane-1,2-diylidenedi(2E) hydrazin-1-yl-2-ylidene] bis (5-methyl-1,3,4-oxadiazole) with some transition metal ion such as Cr3, Co3+, Ni2+ were synthesis ,characterization by magnetic ...
Azhar H. Katea
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Chemoinformatic design and profiling of some derivatives of 1, 2, 4-oxadiazole as potential dengue virus NS-5 inhibitors [PDF]
Samuel Ndaghiya Adawara +3 more
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