Results 121 to 130 of about 9,297,922 (227)

Enhanced antipyretic activity of new 2, 5-substituted 1, 3, 4-oxadiazoles encapsulated in alginate/gelatin particulated systems [PDF]

, 2012
cited By 4International audienceNew 1,3,4-oxadiazoles with pharmacological potential, derived from 5-nitroindazole, have been synthesized. Their chemical structure has been established by elemental and spectral analyses (FT-IR and 1H-NMR).
Holban, M., Cheptea, C., Desbrieres, Jacques, Lionte, C., Şunel, V., Popa, M.   +5 more
core  

Tandem diazotization/cyclization approach for the synthesis of a fused 1,2,3-triazinone-furazan/furoxan heterocyclic system

Beilstein Journal of Organic Chemistry
A straightforward protocol for the synthesis of a previously unknown [1,2,5]oxadiazolo[3,4-d][1,2,3]triazin-7(6H)-one heterocyclic system was developed. The described approach is based on tandem diazotization/azo coupling reactions of (1,2,5-oxadiazolyl ...
Yuri A. Sidunets, Valeriya G. Melekhina, Leonid L. Fershtat   +2 more
doaj   +1 more source

Synthesis and Antimicrobial Activities of Some New Pyrazoles, Oxadiazoles and Isoxazole Bearing Benzofuran Moiety [PDF]

, 2015
The synthesis of novel derivatives of pyrazole-3-carboxylate (3–5) from methyl 4-(benzofuran-2-yl)-2,4-dioxobutanoate (1) is reported. Synthesis of substituted 1,3,4-oxadiazoles (7–11) and 5-amino pyrazole-4-carboxylate (12) derivatives starting fromthe ...
Idrees, M, Siddiqui, NJ, Khati, NT, Dhonde, MG   +3 more
core   +1 more source

Design, synthesis, and enzyme kinetic evaluation of oxadiazole derivatives as nucleoside triphosphate diphosphohydrolase (NTPDase) inhibitors: an integrated <i>in vitro</i> and <i>in silico</i> approach. [PDF]

RSC Adv
Abbas SZ, Ashraf Z, Roshan S, Sughra K, Rahat MA, Shakir I, Latif M.   +6 more
europepmc   +1 more source

Assessment of 1, 3, 4- Oxadiazole Derivatives for Memory Enhancing Activity

International Journal of Pharma Research and Health Sciences, 2019
Veneetha FT, Krishna KL, Monisha Harini S, Vishwanathan B   +3 more
openaire   +1 more source

Activity Profiling of Nitro-Substituted Di(Hetero)Aryl 1,3,4- and 1,2,4-Oxadiazoles: Antimicrobial, Cholinesterase Inhibition and Antioxidant Potential. [PDF]

Arch Pharm (Weinheim)
Šikorová E, Štěpánková Š, Frýbová E, Konečná K, Korbielová J, Švarcová M, Janďourek O, Pflégr V, Bősze S, Krátký M.   +9 more
europepmc   +1 more source

Chemo- and Regioselective Synthesis of 3,4-Dihydropyrimidin-4-ones from 4,5-Dihydro-1,2,4-oxadiazoles and Chromium Alkoxy Alkynyl Fischer Carbene Complexes. [PDF]

Org Lett
Sánchez-Alonso S, Menéndez MI, Merino I, Aguilar E.   +3 more
europepmc   +1 more source

Benzo[<i>d</i>]imidazole anchored oxadiazole derivatives: synthesis, characterization, biological evaluation, <i>in silico</i> docking and ADME-T analysis. [PDF]

RSC Adv
Salluri YR, Chepuri K, Anwar S.
europepmc   +1 more source

A novel and sustainable synthesis-functionalization strategy for the oxidative cyclization towards 2,5-disubstituted-1,3,4-oxadiazoles using bentonite-supported copper(i) iodide as a green catalyst. [PDF]

RSC Adv
Tran VQ, Tran DM, Tran MH, Tran PH, Nguyen HT.   +4 more
europepmc   +1 more source

Effect of 1,3,4-oxadiazoles on expression of biofilm-associated bap gene in clinical isolates of multidrug-resistant Acinetobacter baumannii. [PDF]

Sci Rep
Rahimbakhsh A, Seyfahmadi M, Souldozi A, Hakimelahi R, Alikhani MY, Kafilzadeh F.   +5 more
europepmc   +1 more source