N-[4-Acetyl-5-(2-methylprop-1-enyl)-5-(2-p-tolylpropyl)-4,5-dihydro-1,3,4-thiadiazol-2-yl]acetamide
The title heterocyclic compound, C20H27N3O2S, was synthesized from 2-(4-methylcyclohex-3-enyl)-6-methylhepta-2,5-dien-4-one, which was isolated from the essential oil Cedrus atlantica.
Noureddine Mazoir +5 more
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MOLECULAR DOCKING STUDIES ON THIADIAZOLE DERIVATIVES AS PROTEIN KINASE INHIBITORS [PDF]
Objective: In the present study, a novel series of 1, 3, 4-thiadiazole derivatives were docked against the mycobacterium tuberculosis protein kinase G.
Geetha, G., Sivakumar, D.
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SELENIUM HETEROCYCLES XXXX [I] SYNTHESES OF 4- (2-PYRAZINYL) - 1, 2, 3: SELENADIAZOLE AND 4- (2-PYRAZILYL)' - l,2,3- THIADIAZOLE [PDF]
Reaction of thionyl chloride with 2-acetyl-1- benzenesulfonylpyrrole semicarbazone (6 c) gave 4 - (1- benzenesulfonyl-2 - pyrrolyl) - 1, 2, 3 -thiadiazole (lc). Selenium dioxide oxidation of 2-acetylpyrazine semicarbazone (10) in acetic acid afforded 4- (
doaj
Understanding the synergistic interaction between a 1,3,4-thiadiazole derivative and amphotericin B using spectroscopic and theoretical studies [PDF]
We present a comprehensive spectroscopic study supported by theoretical quantum chemical calculations conducted on a molecular system (4-(5-methyl-1,3,4-thiadiazol-2-yl)benzene-1,3-diol (C1) and the antibiotic Amphotericin B (AmB)) that exhibits highly ...
Ceresa, Luca +11 more
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Unexpected electron acceptor behavior of the 1,3,4-thiadiazole oligomer, a DFT study [PDF]
Electronic and structural properties of two conformations including conjugated compounds of fluorene 1,3,4 thiadiazole and the electron acceptor [6,6]-phenyl C61-butyric acid methyl ester or PCBM, (PCBM/TDA10FL) were calculated using density functional ...
NORMA ROSARIO FLORES HOLGUIN
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SYNTHESIS AND ANTIMICROBIAL ACTIVITY OF SOME (2-AMINO-5-THIOL-1, 3, 4-THIADIAZOLE DERIVATIVES [PDF]
Five derivatives of thiadiazole were prepared with aldehydes and alkyl halides, compoundA: 2-amino-5-thiol-1,3,4- thiadiazole, compound B :2-(o-hydroxybenzylidine)amino-5-thiol-1,3,4-thiadiazole, compoundC: 2(2-butan-lidine)amino-5-thiol-1,3,4 ...
AL-Joubori, Sabiha F- +2 more
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(E)-N-(4-Chlorobenzylidene)-5-(4-methylphenyl)-1,3,4-thiadiazol-2-amine
The title compound, C16H12ClN3S, was synthesized by the reaction of 5-(4-methylphenyl)-1,3,4-thiadiazol-2-amine and 4-chlorobenzaldehyde. The thiadiazole ring is essentially planar with mean deviation of 0.0042 Å.
Peng Yu +4 more
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Substituent Effect on the Absorption Spectra of Mesoionic 1, 3, 4-Thiadiazoles
Substituent Effect on the Absorption Spectra of Mesoionic 1, 3, 4 ...
P. B. Talukdar, S. K. Sengupta
openaire +1 more source
Contribution to the Structm·e of 2,5-Dimercapto-1,3,4-thiadiazole and Related Compounds [PDF]
The structure of 2,5 - dimercapto-1,3,4-thiadiazole and some derivatives was studied from the dependence of UV spectra on pH and H 0 and a monomercapto monodipolar structure is proposed.
B. Stanovnik, M. Tišler
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Background Nowadays, cancer is an important public health problem in all countries. Limitations of current chemotherapy for neoplastic diseases such as severe adverse reactions and tumor resistance to the chemotherapeutic drugs have been led to a ...
Sobhi M. Gomha +3 more
semanticscholar +1 more source

