Results 111 to 120 of about 12,908,442 (282)

The Synthesis, Antimicrobial Activity, and Molecular Docking of New 1, 2, 4-Triazole, 1, 2, 4-Triazepine, Quinoline, and Pyrimidine Scaffolds Condensed to Naturally Occurring Furochromones. [PDF]

Pharmaceuticals (Basel), 2022
Abu-Hashem AA, Al-Hussain SA.
europepmc   +1 more source

Direct Functionalization of an Acid-Terminated Nanodiamond with Azide: Enabling Access to 4‑Substituted-1,2,3-Triazole-Functionalized Particles

, 2017
Azides on the periphery of nanodiamond materials (ND) are of great utility because they have been shown to undergo Cu-catalyzed and Cu-free cycloaddition reactions with structurally diverse alkynes, affording particles tailored for applications in ...
Zachary C. Kennedy (1476781), Christopher A. Barrett (1995808), Marvin G. Warner (1634740)   +2 more
core   +1 more source

Vaporisation Thermodynamics: Are Triazolium Ionic Liquids a Real Alternative to Popular Imidazolium-Based Ionic Liquids?

Liquids
New experimental vapour pressures and vaporisation enthalpies of the ionic liquids [2,4-dimethyl-1,2,4-triazolium][NTf2], [2-methyl-4-ethyl-1,2,4-triazolium][NTf2], and [2-ethyl-4-methyl-1,2,4-triazolium][NTf2] were measured using the Langmuir method in ...
Sergey P. Verevkin, Dzmitry H. Zaitsau
doaj   +1 more source

Synthesis and cytotoxic activity evaluation of some new 1, 3, 4-oxadiazole, 1, 3, 4-thiadiazole and 1, 2, 4- triazole derivatives attached to phthalimide. [PDF]

Res Pharm Sci, 2021
Hassanzadeh F, Jafari E, Shojaei F, Sadeghi-Aliabadi H.   +3 more
europepmc   +1 more source

Click‐Spaltung quartärer Anilinium‐Tetrazine ermöglicht Kaskadenaufbau multifunktioneller biomolekularer Gerüste

Angewandte Chemie, EarlyView.
Die Click‐Chemie hat sich von dem Aufbau kovalenter Bindungen hin zum Spalten von Bindungen weiterentwickelt. Hier wird über einen Kaskaden‐Aufbau berichtet, der diese Verfahren kombiniert, um multifunktionale biomolekulare Gerüste in einer modularen Ein‐Topf‐Reaktion aufzubauen.
Markus Staudt, Christian B. M. Poulie, Andreas Löffler, Peter R. Meinig, Riley J. Deutsch‐Williams, Barbara Herrmann, Ralph Weissleder, Hannes Mikula, Jonathan C. T. Carlson, Matthias M. Herth   +9 more
wiley   +1 more source

2H‑1,2,3-Triazole-Based Dipeptidyl Nitriles: Potent, Selective, and Trypanocidal Rhodesain Inhibitors by Structure-Based Design

, 2018
Macrocyclic inhibitors of rhodesain (RD), a parasitic cysteine protease and drug target for the treatment of human African trypanosomiasis, have shown low metabolic stability at the macrocyclic ether bridge.
Saint-Auret, Sarah, Wolfgang Haap (1856404), Tanja Schirmeister, Haap, Wolfgang, Bernd Kuhn, Maude Giroud, Bernd Kuhn (260084), Christoph Kuratli (2184006), Rainer E. Martin (1934101), Rainer E. Martin, Marcel Kaiser (41510), Schuler, Franz, Schirmeister, Tanja, Diederich, François, Kaiser, Marcel, Tanja Schirmeister (634370), François Diederich, Marcel Kaiser, Maude Giroud (2017114), Kuratli, Christoph, Christoph Kuratli, Franz Schuler (1416097), Franz Schuler, Sarah Saint-Auret (5071748), Brun, Reto, Sarah Saint-Auret, Giroud, Maude, Reto Brun, Reto Brun (41511), François Diederich (1336185), Martin, Rainer E., Kuhn, Bernd, Wolfgang Haap   +32 more
core   +1 more source

5-Methyl-N′-[5-methyl-1-(4-methylphenyl)-1H-1,2,3-triazole-4-carbonyl]-1-(4-methylphenyl)-1H-1,2,3-triazole-4-carbohydrazide, C22H22N8O2

Zeitschrift für Kristallographie - New Crystal Structures, 2019
C22H22N8O2, monoclinic, P21/c (no. 14), a = 15.5175(5) Å, b = 7.9715(3) Å, c = 17.3941(5) Å, β = 90.005(3)°, V = 2151.61(12) Å3, Z = 4, Rgt(F) = 0.0592, wRref(F2) = 0.1780, T = 293(2) K.
Aldosari Obaid Fahad, Abdel-Wahab Bakr F., Alotaibi Mohammad Hayal, Hegazy Amany S., Kariuki Benson M., El-Hiti Gamal A.   +5 more
doaj   +1 more source

New 1,2,3-Triazole-genipin Analogues and Their Anti-Alzheimer’s Activity

A novel series of 1,2,3-triazole-genipin analogues were designed, synthesized, and evaluated for neuroprotective activity, acetylcholinesterase (AChE), and butyrylcholinesterase (BuChE) inhibitory activity.
Jiraporn Tocharus (4672513), Apichart Suksamrarn (482768), Suwichada Jaipea (13008125), Patamawadee Silalai (13008122), Rungnapha Saeeng (2686342), Anan Athipornchai (6160775)   +5 more
core   +1 more source

Cu(OTf)₂-Catalyzed 1,2,3-triazole-ring-controlled selective phenolic O–H bond methylthiomethylation

, 2019
Copper-catalyzed selective methylthiomethylation of 1,4-disubstituted 1,2,3-triazole phenols using DMSO as a methylthiomethylation reagent was achieved.
Weigen Du (6918761), Yubo Jiang (4426555), Huiling Cheng (2898452), Xinyuan Ma (5262572), Wei Liu (20030)   +4 more
core   +1 more source

Jahn-Teller distortion in 2-pyridyl-(1,2,3)-triazole-containing copper(ii) compounds

, 2018
© The Royal Society of Chemistry and the Centre National de la Recherche Scientifique. The syntheses, characterization and experimental solid state X-ray structures of five low-spin paramagnetic 2-pyridyl-(1,2,3)-triazole-copper compounds, [Cu(Ln)2Cl2 ...
C Wilson (7748510), J Conradie (19157167), Johannes Potgieter (23880057), SJ Coles (14547215), KM Tawfiq (24002700), MM Conradie (24002697), GJ Tizzard (19694878)   +6 more
core