Quinone-catalyzed oxidative deformylation: synthesis of imines from amino alcohols [PDF]
Beilstein Journal of Organic Chemistry, 2017 A new method for imine synthesis by way of quinone-catalyzed oxidative deformylation of 1,2-amino alcohols is reported. A wide range of readily accessible amino alcohols and primary amines can be reacted to provide N-protected imine products.
Xinyun Liu +4 more
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Diastereoselective synthesis of vicinal amino alcohols [PDF]
Organic & Biomolecular Chemistry, 2012 The vicinal amino alcohol is a common motif in natural products and pharmaceuticals. Amino acids constitute a natural, inexpensive, and enantiopure choice of starting material for the synthesis of such functionalities. However, the matters concerning diastereoselectivity are not obvious.
Koskinen, Ari, Karjalainen, Oskari
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Synthesis of Azetidine-Based Beta-Amino Alcohols
Medical Sciences Forum, 2022 Beta-amino alcohols are versatile chemicals used as scaffolds in medicinal chemistry and they are key factors for the efficacy of numerous pharmaceutical products.
Linda Supe
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Highly Enantioselective Synthesis of β-Amino Alcohols [PDF]
Organic Letters, 2006 AbstractChemInform is a weekly Abstracting Service, delivering concise information at a glance that was extracted from about 200 leading journals. To access a ChemInform Abstract, please click on HTML or PDF.
Métro, Thomas-Xavier +3 more
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PHARMACOLOGY OF TREMOR-PRODUCING AMINO ALCOHOLS
Journal of Pharmacy and Pharmacology, 1958 Abstract The pharmacological properties of a series of amino alcohols of the general formula RCH(NH2)ṁ(CH2)nṁC(OH)R2 have been studied The most striking action of these compounds is their ability to produce a sustained tremor, which is compared with those produced by other tremorogenic agents.
A, AHMED, P B, MARSHALL, D M, SHEPHERD
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Microwave-Assisted Kabachnik–Fields Reaction with Amino Alcohols as the Amine Component [PDF]
Molecules, 2019 In this paper, the microwave (MW)-assisted catalyst-free and mostly solvent-free Kabachnik−Fields reaction of amino alcohols, paraformaldehyde, and various >P(O)H reagents (dialkyl phosphites, ethyl phenyl-H-phosphinate, and secondary phosphine ...
Ádám Tajti +4 more
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Hydrogen‐Borrowing Alkylation of 1,2‐Amino Alcohols in the Synthesis of Enantioenriched γ‐Aminobutyric Acids [PDF]
Angewandte Chemie - International Edition, 2021 William R F Goundry, Timothy J Donohoe
exaly +2 more sources
Asymmetric Synthesis of γ-Amino Alcohols by Copper-Catalyzed Hydroamination. [PDF]
Org Lett, 2019 Asymmetric synthesis of γ-amino alcohols from unprotected allylic alcohols by a copper-catalyzed hydroamination strategy has been developed. Using easily accessible starting materials, a range of chiral 1,3-amino alcohols were prepared with excellent ...
Ichikawa S, Buchwald SL.
europepmc +2 more sources
In situ epoxide generation by dimethyldioxirane oxidation and the use of epichlorohydrin in the flow synthesis of a library of β-amino alcohols [PDF]
Royal Society Open Science, 2018 The flow coupling of epichlorohydrin with substituted phenols, while efficient, limits the nature of the epoxide available for the development of focused libraries of β-amino alcohols.
Peter J. Cossar +3 more
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Synthesis of Amino-Acid-Based Nitroalkenes
Organics, 2022 Fatty-acid-based nitroalkenes have recently received great attention because of their bioactivities. On the contrary, peptide- or amino-acid-based nitroalkenes have been scarcely explored so far, although they may exhibit interesting biological ...
Velisaria-Eleni Gerogianni +3 more
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