Results 201 to 210 of about 37,127 (212)

Dicationic liquid mediated synthesis of tetrazoloquinolinyl methoxy phenyl 4-thiazolidinones and their antibacterial and antitubercular evaluation

Synthetic Communications, 2019
In a search of new potentially active antitubercular agents here we have synthesized 3-substituted phenyl-2-(4-(tetrazolo[1,5-a]quinolin-4-ylmethoxy)phenyl)thiazolidin-4-ones (8a-l) and evaluated their antibacterial, particularly antitubercular activity.
Amarsinh R. Deshmukh, Sambhaji T. Dhumal, Laxman U. Nawale, V. Khedkar, D. Sarkar, R. Mane   +5 more
semanticscholar   +1 more source

Dry powder inhalers of antitubercular drugs.

Tuberculosis, 2022
Nidhi Nainwal, Yuwanshi Sharma, Vikas Jakhmola   +2 more
semanticscholar   +1 more source

Novel 1,3,4-oxadiazoles as antitubercular agents with limited activity against drug-resistant tuberculosis.

Future Medicinal Chemistry, 2019
AIM In recent times, heterocyclic chemotypes are being explored for the development of new antimycobacterials that target the drug-resistant tuberculosis.
Vitthal B. Makane, V. Krishna, E. V. Krishna, Manjulika Shukla, B. Mahizhaveni, S. Misra, S. Chopra, D. Sriram, V. N. Azger Dusthackeer, H. Rode   +9 more
semanticscholar   +1 more source

Antitubercular Potential of Novel Isoxazole Encompassed 1, 2, 4- Triazoles: Design, Synthesis, Molecular Docking Study and Evaluation of Antitubercular Activity

, 2020
Decaprenylphosphoryl-β-D-ribose epimerase (DprE1), a flavoprotein enzyme engaged in the biosynthesis of decaprenylphosphoryl-β-D-arabinofuranose (DPA), is the only contributor of arabinose residues which is fundamental for the mycobacterium cell wall ...
N. Ganesh, A. S, Manisha Singh, V. M. Chandrashekar, G. Pujar   +4 more
semanticscholar   +1 more source

iAtbP-Hyb-EnC: Prediction of antitubercular peptides via heterogeneous feature representation and genetic algorithm based ensemble learning model

Comput. Biol. Medicine, 2021
S. Akbar, Ashfaq Ahmad, Maqsood Hayat, A. Rehman, Salman Khan, Farman Ali   +5 more
semanticscholar   +1 more source

Mycobacterium enoyl acyl carrier protein reductase (InhA): A key target for antitubercular drug discovery.

Bioorganic chemistry (Print), 2021
M. Prasad, R. Bhole, P. Khedekar, R. Chikhale   +3 more
semanticscholar   +1 more source

Synthesis, biological evaluation and molecular docking studies of new pyrazolines as an antitubercular and cytotoxic agents.

Infectious Diseases - Drug Targets, 2019
A series of new pyrazolines containing 2,5-dichloro-3-acetylthiophene chalcone moiety (PZT1-PZT20) have been synthesized, characterized by 1HNMR and 13CNMR and evaluated for them in vitro antitubercular activity against M.
B. V. Lokesh, Y. Prasad, A. Shaik
semanticscholar   +1 more source

Synthesis, structural, biological andin silicostudies of new 5-arylidene-4-thiazolidinone derivatives as possible anticancer, antimicrobial and antitubercular agents

New Journal of Chemistry, 2019
Thiazolidinone–sulfonamide hybrids emerged as promising anticancer and antitubercular agents, and their anticancer activity was confirmed by docking studies.
A. Sunil Kumar, Jyothi Kudva, B. Bharath, K. Ananda, Rajitha Sadashiva, S. Madan Kumar, B. Revanasiddappa, Vasantha Kumar, P. Rekha, Damodara Naral   +9 more
semanticscholar   +1 more source

Antitubercular properties of thiazolidin-4-ones - A review.

European journal of medicinal chemistry, 2021
Nazar Trotsko
semanticscholar   +1 more source

Development of Antimicrobial, Antimalarial and Antitubercular Compounds Based on a Quinoline-Pyrazole Clubbed Scaffold Derived via Doebner Reaction

Chemistry Africa, 2020
K. Pandya, Arpan Patel, P. Desai
semanticscholar   +1 more source