Synthesis, evaluation, molecular docking, and molecular dynamics studies of novel N-(4-[pyridin-2-yloxy]benzyl)arylamine derivatives as potential antitubercular agents. [PDF]
Drug Dev Res, 2020 Verma R +6 more
europepmc +3 more sources
Development of 6-Methanesulfonyl-8-nitrobenzothiazinone Based Antitubercular Agents. [PDF]
ACS Med Chem Lett, 2022 Shi R +9 more
europepmc +3 more sources
Synthesis and structure−activity relationship of 8-substituted protoberberine derivatives as a novel class of antitubercular agents [PDF]
, 2013 Yinghong Li +8 more
core +3 more sources
Tetrahydropyrazolo[1,5-a]Pyrimidine-3-Carboxamide and N-Benzyl-6′,7′-Dihydrospiro[Piperidine-4,4′-Thieno[3,2-c]Pyran] analogues with bactericidal efficacy against Mycobacterium tuberculosis targeting MmpL3 [PDF]
, 2013 Mycobacterium tuberculosis is a major human pathogen and the causative agent for the pulmonary disease, tuberculosis (TB). Current treatment programs to combat TB are under threat due to the emergence of multi-drug and extensively-drug resistant TB.
A Hill +48 more
core +15 more sources
New Application of 1,2,4-Triazole Derivatives as Antitubercular Agents. Structure, In Vitro Screening and Docking Studies. [PDF]
Molecules, 2020 Karczmarzyk Z +6 more
europepmc +3 more sources
Discovery of (3-Benzyl-5-hydroxyphenyl)carbamates as New Antitubercular Agents with Potent In Vitro and In Vivo Efficacy. [PDF]
Molecules, 2019 Cheng YJ +6 more
europepmc +3 more sources
Causality assessment, severity and preventability of adverse drug reactions due to first-line antitubercular agents [PDF]
Pharmaciana, 2022 TB (Tuberculosis) is a common infectious disease affecting humans since very long time. Multidrug therapy with its associated adverse drug reactions is one of the major concerns for the management of TB.
Gunjan Upadhyay +2 more
doaj +1 more source
Microbial glycosylation of antitubercular agent chlorflavonin [PDF]
Journal of Bioscience and Bioengineering, 2023 Flavonoids have shown health-benefiting properties, such as antioxidative and anti-inflammatory activities, and are commonly used as nutraceuticals and pharmaceuticals. Although flavonoids are predominantly identified from plants, several filamentous fungal species have also been reported to produce bioactive flavonoids, including chlorflavonin from ...
Jie Ren, Jixun Zhan
openaire +3 more sources
Design, Synthesis and Biological Evaluation of Some Triazole Schiff's Base Derivatives as Potential Antitubercular Agents. [PDF]
Open Med Chem J, 2018 Sager AA +11 more
europepmc +3 more sources
Inhalable spray-dried chondroitin sulphate microparticles: effect of different solvents on particle properties and drug activity [PDF]
, 2020 Spray-drying stands as one of the most used techniques to produce inhalable microparticles, but several parameters from both the process and the used materials affect the properties of the resulting microparticles.
Buttini, Francesca +6 more
core +1 more source