Results 111 to 120 of about 822 (147)

Approach to synthesis of 8-azasteroids

Bulletin of the Academy of Sciences of the USSR Division of Chemical Science, 1972
A. A. Akhrem, A. M. Moiseenkov, A. I. Poselenov   +2 more
openaire   +2 more sources

Azasteroids as inhibitors of testosterone 5α-reductase in mammalian skin

, 1993
T. Mellin, R. Busch, G. H. Rasmusson
semanticscholar   +1 more source

6-Azasteroids: structure-activity relationships for inhibition of type 1 and 2 human 5 alpha-reductase and human adrenal 3 beta-hydroxy-delta 5-steroid dehydrogenase/3-keto-delta 5-steroid isomerase.

Journal of Medicinal Chemistry, 1994
S. Frye, C. Haffner, P. Maloney, R. Mook, G. Dorsey, R. Hiner, C. Cribbs, T. Wheeler, J. A. Ray, R. Andrews   +9 more
semanticscholar   +1 more source

4,7 beta-Dimethyl-4-azacholestan-3-one (MK-386) and related 4-azasteroids as selective inhibitors of human type 1 5 alpha-reductase.

Journal of Medicinal Chemistry, 1994
R. Bakshi, G. Patel, G. H. Rasmusson, W. Baginsky, G. Cimis, K. Ellsworth, B. Chang, H. Bull, R. Tolman, G. Harris   +9 more
semanticscholar   +1 more source

6-Azasteroids: potent dual inhibitors of human type 1 and 2 steroid 5 alpha-reductase.

Journal of Medicinal Chemistry, 1993
S. Frye, C. Haffner, P. Maloney, R. Mook, G. Dorsey, R. Hiner, K. Batchelor, H. N. Bramson, J. Stuart, S. Schweiker   +9 more
semanticscholar   +1 more source

Synthesis Of 11-azasteroids from aromatic amines, formaldehyde and cyclopentadiene

, 1991
P. J. Gregoire, J. M. Mellor, Glynn D. Merriman   +2 more
semanticscholar   +1 more source

Total synthesis of 3-azasteroids via the transannular Diels–Alder strategy

Tetrahedron, 2001
Daniel Fortin, Eric Marsault, Pierre Deslongchamps   +2 more
exaly  

19-Nor-10-azasteroids. 5.(1) A Synthetic Strategy for the Preparation of (+)-17-(3-Pyridyl)-(5beta)-10-azaestra-1,16- dien-3-one, a Novel Potential Inhibitor for Human Cytochrome P450(17)(alpha) (17alpha-Hydroxylase/C(17,20)-lyase).

Journal of Organic Chemistry, 1999
A. Guarna, E. Occhiato, F. Machetti, V. Giacomelli   +3 more
semanticscholar   +1 more source

Preparation of (5α,13α)-d-azasteroids as key precursors of a new family of potential GABAA receptor modulators

Steroids, 2003
Yuefei Hu, Shaozhong Wang, Hongwen Hu
exaly  

3D-QSAR studies on unsaturated 4-azasteroids as human 5α-reductase inhibitors: A self organizing molecular field analysis approach

European Journal of Medicinal Chemistry, 2010
Suresh Thareja
exaly