Enantiocontrolled Azetidine Library Synthesis via Strain-Release Functionalization of 1-Azabicyclobutanes. [PDF]
Bielecki M +9 more
europepmc +1 more source
Novel Sulfonium Reagents for the Modular Synthesis of Spiro[2.3]Hexanes and Heteroatom-Containing Analogues: Synthesis, Application, and Evaluation as Bioisosteres. [PDF]
Natho P +10 more
europepmc +1 more source
Potent, Selective, and Brain Penetrant Ether-Linked 2-Aminopyridine Inhibitors of Human Neuronal Nitric Oxide Synthase with Excellent Oral Bioavailability. [PDF]
Ansari A +6 more
europepmc +1 more source
Acid Versus Amide-Facts and Fallacies: A Case Study in Glycomimetic Ligand Design. [PDF]
Smieško M +5 more
europepmc +1 more source
TLR9-activating cholesterol azetidine derivative-assisted therapeutic vaccines for cancer immunotherapy. [PDF]
Chen J +6 more
europepmc +1 more source
Structural Characterization, Toxicity Assessment and Molecular Modeling of Forced Degradation Products of Siponimod. [PDF]
Liang Y, Zhang T, Zhang D, Jin B, Ma C.
europepmc +1 more source
Fused-Linked and Spiro-Linked N-Containing Heterocycles. [PDF]
Moskalik MY, Shainyan BA.
europepmc +1 more source
Accessing Azetidines through Magnesium-Mediated Nitrogen Group Transfer from Iminoiodinane to Donor-Acceptor Cyclopropanes. [PDF]
Bansode AH +5 more
europepmc +1 more source
Site-Selective Carbonylation of Azetidines via Copper-Catalyzed Difluorocarbene Insertion. [PDF]
Zhou F, Tan TD, Koh MJ.
europepmc +1 more source

