Results 71 to 80 of about 3,171 (179)

Lewis Acid Catalyzed Dual Strain-Release Platform for Transforming Azabicyclo[1.1.0]butanes into Functionalized Azetidines with Donor-Acceptor(D-A) Cyclopropanes and Bicyclo[1.1.0]butanes. [PDF]

Org Lett
Hazra S, Patel M, Mondal S, Ahmed R, Sasmal P, De S, Saha J.   +6 more
europepmc   +1 more source

Triplet Energy Transfer-Driven Intermolecular [2+2] Photocycloaddition of Acyclic Imines and Indoles: Facile Access to Azetidine-Fused Indolines. [PDF]

Adv Sci (Weinh)
Yang G, Han Z, Zhang H, Cui X.
europepmc   +1 more source

4″-Methyl-<i>S</i>-Adenosyl-l-Methionines Are Substrates for 4-Methylazetidinecarboxylic Acid Synthases. [PDF]

ACS Chem Biol
Nagano N, Kiuchi K, Minato A, Sato S, Moriwaki Y, Müller R, Eguchi T, Kudo F.   +7 more
europepmc   +1 more source

A Convenient Synthesis of CHF₂O-Containing Pyrrolidines and Related Compounds — Prospective Building Blocks for Drug Discovery

SynOpen
Kostiantyn Levchenko, Ivan Virstiuk, Daria Menshykova, Nazariy Pokhodylo   +3 more
doaj   +1 more source

Structural and mechanistic insights into azetidine-associated αKG-NHFe enzyme OkaE with multifunctional catalysis. [PDF]

Nat Commun
Wang X, Yu J, Liu T, Zhang X, Ju M, Xie Z, Naowarojna N, Ping L, Dong Y, Gong B, Xie Y, Nie Y, Hsiang T, Wu R, Zhang L, Liu P, Zhu G, Yan W, Liu X.   +18 more
europepmc   +1 more source

Discovery and Development of a Small-Molecule Inhibitor Targeting the GAS41 YEATS Domain in Nonsmall Cell Lung Cancer. [PDF]

J Med Chem
Listunov D, Winkler A, Ray J, Linhares BM, Clegg B, Weaver S, Kim E, Zari S, Park SR, Zolov SN, Chuikov S, Zhao L, Shah YM, Keshamouni VG, Grembecka J, Cierpicki T.   +15 more
europepmc   +1 more source

Editorial: Recent advances in synthesizing and utilizing nitrogen-containing heterocycles

Frontiers in Chemistry
Takashi Ohshima, Hsyueh-Liang Wu, Hyun-Joon Ha   +2 more
doaj   +1 more source

Optimization Leading to a Potent and Selective Cbl‑b Inactive-State Inhibitor That Demonstrated <i>In Vivo</i> Efficacy. [PDF]

ACS Med Chem Lett
Liang J, Lambrecht MJ, Huestis MP, Zhu B, Barton LM, Castanedo GM, Ung PM, Larouche-Gauthier R, Jakalian A, Leclerc JP, Yadav A, Haghshenas P, Aubert-Nicol S, Ismaili H, Zhao L, Leblanc M, de Almeida H, Wang Q, Garner T, Tan S, Prangley MS, Pang J, Murray JM, Yu C, Hsu PL, Rutz S, Ishizuka I, Huang H, Gao C, Chen M, Mutter-Rottmayer L, Kakiuchi-Kiyota S, Leung DH, Kou P, Bao L, Wang X.   +35 more
europepmc   +1 more source

Discovery and Mechanism of a Diiron Enzyme in Ethylidene Azetidine Formation. [PDF]

J Am Chem Soc
Shen Y, Zheng YC, Palacios PM, Wang K, Maggiolo AO, Guo Y, Chang WC.   +6 more
europepmc   +1 more source

Design, synthesis, and biological evaluation of novel 3-oxo-2,3-dihydropyridazine derivatives as interleukin-2-inducible T-cell kinase (ITK) inhibitors. [PDF]

RSC Adv
Tangallapalli S, Gundla R, Paidikondala K, Gurská S, Rampeesa NK, Anugu SR, Džubák P, Hajdúch M, Das V, Katari NK.   +9 more
europepmc   +1 more source