Results 141 to 150 of about 38,481 (291)

High performance mixed bisimide resins and composites based thereon [PDF]

, 1986
Mixtures of bismaleimide/biscitraconirnide resins produces materials which have better handling, processing or mechanical and thermal properties, particularly in graphite composites, than materials made with the individual resins. The mechanical strength
ations., Parker, J. A.
core   +1 more source

Antiurolithiatic Potential of a Series of Phthalimide Derivatives on Calcium Oxalate Crystals

Chemistry &Biodiversity, Volume 23, Issue 1, January 2026.
ABSTRACT Urolithiasis, primarily caused by calcium oxalate crystals, represents a major health concern due to high recurrence rates and limitations of current treatments in dissolving existing stones. This study investigated the antiurolithiatic potential of 15 phthalimide derivatives against calcium oxalate monohydrate (COM) and dihydrate (COD ...
Daniele Regina Sonza, Laura Von Borell du Vernay França, Rita de Cássia Vilhena da Silva, Anelize Dada, Mariana Zanovello, Thaise Boeing, Priscila de Souza, Rogério Correa   +7 more
wiley   +1 more source

Connectivity Effects on the Kinetically Controlled Supramolecular Polymerization of Linear Scaffolds

ChemistryEurope, Volume 4, Issue 1, January 2026.
The kinetically controlled supramolecular homo‐ and heteropolymerization of BDTs (1a and 1b) and BODIPYs (2a and 2b), endowed with amido‐ester flexible ethylene linkers, that prompt the formation of seven‐membered, intramolecularly H‐bonded pseudocycles retarding the supramolecular polymerization, is investigated experimentally showing a complex ...
Cristina Naranjo, Rafael Gómez, Gustavo Fernández, Luis Sánchez   +3 more
wiley   +1 more source

Allosteric Inhibitors of SARS‐CoV‐2 RNA‐Dependent RNA Polymerase Based on N,N′‐Diphenylurea

ChemMedChem, Volume 21, Issue 1, January 2026.
Inhibitors of SARS‐CoV‐2 RdRp activity based on N,N′‐diphenylurea scaffold have been identified. Several compounds exhibit residual activity (RA) below 50% in an enzymatic assay (at 10 µM concentration) and improved aqueous solubility compared to the previously reported series of inhibitors.
Artem Chayka, Matěj Danda, Alžběta Dostálková, Vojtěch Spiwok, Lamija Zijadic, Anna Klimešová, Marina Kapisheva, Michala Zgarbová, Jan Weber, Tomáš Ruml, Michaela Rumlová, Zlatko Janeba   +11 more
wiley   +1 more source

Technetium-99m radiolabelling of anN-amino-alkyl-benzamide nitrido- and oxo-technetium bis(aminoethanethiol) derivative synthesis and biological results. Potential melanoma tracer agents [PDF]

, 1999
Philippe Auzeloux, Marie‐France Moreau, Janine Papon, Martine Bayle, Michèle Borel, Roberto Pasqualini, Jean-Claud Madelmont   +6 more
openalex   +1 more source

Transition Metal (II) Complexes of (E)-N-(4-methylbenzylidene)-2-((Z)-(4-methylbenzylidene)amino)benzamides: Synthesis, Characterization and their Biological Evaluation

, 2021
Venkatesh K. Bhovi, Sulochana P. Melinmath, Vrushabendra Basavanna, Srikantamurthy Ningaiah, Y Matsumoto, J Sawamura, Y Murata, T Nishikata, R Yazaki, T Ohshima, M Maclachlan, M Park, L Thompson, A Hamil, K Khalifa, A Almutaleb, M Nouradean, Synthesis, H Schiff, M Shamsipur, A Ghiasvand, H Sharghi, Naeimi, F Mahmoudi, S Farhadi, M Dusek, M Poupon, Synthesis, Y Xia, J Wang, A Hamed, I Abdelhamid, G Saad, N Elkady, M Elsabee, T Magalhaes, C Da Silva, L Dos Santos, D Santos, L Silva, B Fuchs, E Mylonakis, C Martins, M De Resende-Stoianoff, A De Fatima, A Hassan, A Osman Said, B Heakal, A Younis, M Abdelmoaz, M Abdrabou, S Zhu, S Xu, X Yi, J Wang, Z Zhao, J Jiang, N Beyazit, H akran, A Cabir, Y Akiscan, C Demetgul, E Yuksel, A Bilici, I Gecibesler, Kaya, F Tokali, P Taslimi, H Usanmaz, M Karaman, K Sendil, Synthesis, R Joshi, A Kumari, K Singh, H Mishra, S Pokharia, A Frei, A King, G Lowe, A Cain, F Short, H Dinh, A Elliott, J Zuegg, J Wilson, M Blaskovich, K Singh, M Barwa, P Tyagi, H Barbosa, M Attjioui, A Ferreira, B Moerschbacher, E Cavalheiro, K Buldurun, N Turan, E Bursal, A Mantarci, F Turkan   +99 more
openalex   +1 more source

Optimization of 4‐Amino‐2‐Pyridone Inhibitors of Proprotein Convertase Subtilisin/Kexin Type 9: Integrating Structure–Activity and Structure–Metabolism Relationships

ChemMedChem, Volume 21, Issue 1, January 2026.
Green chemistry‐based late‐stage functionalization (LSF) of the anti‐proprotein convertase subtilisin/kexin type 9 (PCSK9) early lead compound 5c led to optimized analogs with improved metabolic stability/PCSK9 IC50 ratio. Proprotein convertase subtilisin/kexin type 9 (PCSK9) is a key drug target for the treatment of different hypercholesterolemia ...
Lisa Giannessi, Maria Giovanna Lupo, Martina Ugolotti, Bianca Papotti, Beatrice Mattina, Maria Grazia Martina, Anna Demurtas, Cristina Padula, Sara Nicoli, Marco Crescenzio, Nicola Ferri, Francesca Zimetti, Marco Radi   +12 more
wiley   +1 more source

Conformational analysis, part 43. A theoretical and LIS/NMR investigation of the conformations of substituted benzamides [PDF]

, 2015
Raymond J. Abraham, Nuria Aboitiz, Marco Filippi, Eva Genesio, Paola Piaggio, Fernando Sancassan   +5 more
openalex   +1 more source

Glyoxalase‐1 Inhibition Leads to Ferroptosis Induction in Lung Cancer Cells: A Dual Mechanism of Action of Hydroxamic Acids Derived from Cysteine

ChemMedChem, Volume 21, Issue 1, January 2026.
A set of three cysteine‐derived hydroxamic acids were synthesized and evaluated for human gloxalase‐1 inhibition and ferroptosis induction activities. Among them, compound 2 exhibited a potent inhibitory effect against human glyoxalase‐1 and induced ferroptosis in non‐small cell lung cancer cell lines, increasing reactive oxygen species production and ...
Josué Martínez‐Miranda, Dolores Aguilar‐Cázares, Angélica Flores–Flores, Miguel Ángel Santos‐Contreras, José S. López‐González, Rodrigo Aguayo‐Ortiz, Rogélio Hernández‐Pando, Francisco Hernández‐Luis   +7 more
wiley   +1 more source

Liquid Chromatography‐Tandem Mass Spectrometry Methods for Rapid Measurement of the Molar Activity (Am) of Cyclotron‐Produced [18F]Fluoride and Derived Radiotracers

Chemistry–Methods, Volume 6, Issue 1, January 2026.
Accurate and simple liquid chromatography‐tandem mass spectrometry methods for measuring Am for [18F]fluoride on two rapidly derived surrogates, [18F]FAY and [18F]PCBSF, can serve as forensic tools for investigating the sources of carrier, Am determinations during routine tracer productions and be applied to radiotracers lacking a strong ultraviolet ...
Nicholas R. Ellin, Sean W. Costner, Cheryl L. Morse, Fatemak Ahmadi, Sanjay Telu, Fabrice G. Siméon, Shuiyu Lu, H. Umesha Shetty, Victor W. Pike   +8 more
wiley   +1 more source