Results 91 to 100 of about 17,013 (236)
, 2016 A Rh(III)-catalyzed one-pot reaction of benzamides, ketones, and hydrazines for facile access to isoindolinones is reported. In this method, various ketones are transformed into donor–donor diazo compounds, which sequentially engage in insertion with ...
Yan Zhang (8098) +2 more
core +1 more source
Cytogenotoxic Effects of Fluopyram in Allium cepa Root Cells Involving Microtubule Disruption
Environmental Toxicology, EarlyView.ABSTRACT Fluopyram is a next‐generation fungicide widely used in agriculture; however, its persistence in soils and mobility toward aquatic systems have raised concerns regarding potential ecotoxicological risks. This study evaluated the cytogenotoxic effects of a commercial fluopyram‐based pesticide formulation on Allium cepa root meristem cells ...
Carlos Filipe Camilo‐Cotrim +10 more
wiley +1 more source
British Journal of Pharmacology, EarlyView.Abstract Venetoclax combined with hypomethylating agents has improved treatment for older or unfit patients with acute myeloid leukaemia (AML), but resistance and relapse remain common. This review analyses the rationale for combining venetoclax with inhibitors of histone deacetylase (HDAC).
Jaebok Lee, Marc Diederich
wiley +1 more source
Rhodium-Catalyzed Transarylation of Benzamides: C–C Bond vs C–N Bond Activation
, 2020 A rhodium-catalyzed transarylation of benzamides via selective C–C bond activation with arylboronic acids was described, which was distinct from the conventional metal-catalyzed C–N bond activation.
Yang Long (1521595) +6 more
core +1 more source
Benzamide-4-Sulfonamides Are Effective Human Carbonic Anhydrase I, II, VII, and IX Inhibitors
Metabolites, 2018 A series of benzamides incorporating 4-sulfamoyl moieties were obtained by reacting 4-sulfamoyl benzoic acid with primary and secondary amines and amino acids. These sulfonamides were investigated as inhibitors of the metalloenzyme carbonic anhydrase (CA,
Morteza Abdoli +3 more
doaj +1 more source
, 1999 Two series of N-[4-(alkyl)cyclohexyl]-substituted benzamides, i.e. a series of N-[4-(tert-butyl)cyclohexyl]-substituted benzamides and a series of N-[4-(ethyl)cyclohexyl]-substituted benzamides, were synthesised and evaluated for their anti-inflammatory ...
Pau, Amedeo +8 more
core
Ruthenium-catalyzed ortho-C–H halogenations of benzamides
, 2014 [Ru-3(CO)(12)] and AgO2C(1-Ad) enabled the first ruthenium-catalyzed intermolecular halogenations of arenes via C-H activation. Thereby, brominations and iodinations of electron-rich and electron-deficient benzamides were achieved in a highly selective ...
Ackermann, Lutz, Wang, Lianhui
core +1 more source
Ars PharmaceuticaA series of 4-(2-(4-substituted phenyl)-4-oxoquinazolin-3(4H)-yl)-N-(2-(4-fluorophenyl)-4-oxo-5-(arylidene)thiazolidin-3-yl) benzamides (VIa-n) have been synthesized by condensation of N-(2-(4-fluorophenyl)-4-oxothiazolidin-3-yl)-4-(4-oxo-2-(4 ...
Sukanya Nara, Achaiah Garlapati
doaj +1 more source
Substituted [(4-Phenylpiperazinyl)- methyl]benzamides: Selective Dopamine D4 Agonists
, 2016 Substituted [(4-Phenylpiperazinyl)- methyl]benzamides: Selective Dopamine D4 ...
Lawrence D. Wise (2537467) +7 more
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Palladium-Catalyzed Ortho-Arylation of Benzamides via Direct sp2 C–H Bond Activation
, 2016 The palladium-catalyzed ortho-arylation of benzamides by aryl iodides has been demonstrated with the simplest amide CONH2 as a directing group for the first time.
Guan-Wu Wang (1456660) +2 more
core +1 more source