Results 101 to 110 of about 17,013 (236)

In silico identification of benzamide-based aryl halides as EGFR inhibitors: multi-ligand ADMET, pharmacophore mapping, and target prediction

open access: yesIn Silico Research in Biomedicine
Cancer is one of the greatest global health challenges, with specific costs of US$25 trillion by 2050, including treatment and socioeconomic impacts. The epidermal growth factor receptor (EGFR), a central tyrosine kinase, is a key target for anticancer ...
Caroline do Nascimento Gonçalves   +2 more
doaj   +1 more source

Substituted Benzamides Containing Azaspiro Rings as Upregulators of Apolipoprotein A-I Transcription

open access: yesMolecules, 2012
Apolipoprotein A-I (Apo A-I) is the principal protein component of high density lipoprotein (HDL), which is generally considered as a potential therapeutic target against atherosclerosis.
Bin Hong   +7 more
doaj   +1 more source

Selective Photoinduced α‐Amino C(sp3)–H Alkylation Mediated by NHC–Borane

open access: yesAdvanced Synthesis &Catalysis, Volume 368, Issue 17, 1 September 2026.
Herein, we report a selective photoinduced functionalization of α‐amino C(sp3)─H bonds mediated by NHC–boranes. This reaction proceeds efficiently without the need for any external radical initiator or photoredox catalyst. Mechanistic studies reveal that the reaction proceeds via an efficient radical chain, featuring the formation of an aryl radical ...
Gabin Lalande   +2 more
wiley   +1 more source

Effect of methylated amides in the CEP profile of benzamides 48, 51 and 52.

open access: yes, 2018
Effect of methylated amides in the CEP profile of benzamides 48, 51 and 52.
Sonia Maria Gutiérrez Sanfeliciano (4961983)   +1 more
core   +1 more source

Design, anticonvulsive and neurotoxic properties of retrobenzamides - N-(nitrophenyl)benzamides and N-(aminophenyl)benzamides

open access: yes, 1999
Design, anticonvulsant properties in maximal electroshock-induced seizures [MES] and seizures induced by subcutaneous administration of pentetrazole (scPtz), and neurotoxicity of retrobenzamides (N-(nitrophenyl)benzamides and N-(aminophenyl) benzamides ...
Stables, JP.   +4 more
core  

Anticoccidial therapy small guide [PDF]

open access: yesMedicamentul Veterinar, 2007
Being a major challenge, because of ingenious parasite's survival strategies and treatment's transience, anticoccidal therapy it is a major priority. In this respect, therapeutic conduct must be adjusted as well is possible on the most efficient drug ...
Cristina, T. Romeo
doaj  

Synthesis of tertiary benzamides via Pd-catalyzed coupling of arylboronic esters and carbamoyl chlorides

open access: yes, 2005
Ortho-substituted arylboronic esters are efficiently coupled with carbamoyl chlorides under Pd-catalysis to give tertiary ...
Kristensen, Jesper Langgaard   +3 more
core   +1 more source

Antiglycation and Amyloid‐β Inhibitory Activities of Pandanus odorifer Extracts and Isolated Constituents: In Vitro and Molecular Docking Insights

open access: yesChemistry &Biodiversity, Volume 23, Issue 9, September 2026.
Pandanus odorifer methanolic extract exhibited strong antiglycation activity, moderate antioxidant capacity, and high flavonoid content. Three isolated compounds reduced Aβ‐associated ThT fluorescence, with blumenol C glucoside showing the greatest effect.
Patricia Marie P. Oliva   +4 more
wiley   +1 more source

Cobalt-Catalyzed Direct Carbonylation of Aminoquinoline Benzamides

open access: yes, 2015
A method for direct carbonylation of aminoquinoline benzamides has been developed. Reactions proceed at room temperature in trifluoroethanol solvent, use oxygen from air as an oxidant, and require Mn­(OAc)3 as a cocatalyst.
Liene Grigorjeva (1332981)   +1 more
core   +1 more source

Heterocyclic‐Based Fungicides: Emerging Strategies for Viable Plant Disease Control

open access: yesChemistry &Biodiversity, Volume 23, Issue 9, September 2026.
Heterocyclic compounds have attracted considerable attention because of their structural diversity, potent antifungal activity, and ability to interact with multiple fungal targets, offering broad‐spectrum protection against phytopathogens. Synthetic and semisynthetic/part‐natural scaffolds, particularly azole, quinoline, indole, cyclotryptamine, and ...
Sumit Tahlan   +4 more
wiley   +1 more source

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