Results 111 to 120 of about 16,265 (239)

Palladium-Catalyzed Ortho-Arylation of Benzamides via Direct sp² C–H Bond Activation

, 2016
The palladium-catalyzed ortho-arylation of benzamides by aryl iodides has been demonstrated with the simplest amide CONH2 as a directing group for the first time.
Guan-Wu Wang (1456660), Ting-Ting Yuan (385353), Dan-Dan Li (137178)   +2 more
core   +1 more source

Synthesis of tertiary benzamides via Pd-catalyzed coupling of arylboronic esters and carbamoyl chlorides

, 2005
Ortho-substituted arylboronic esters are efficiently coupled with carbamoyl chlorides under Pd-catalysis to give tertiary ...
Kristensen, Jesper Langgaard, Lysén, M., Kelleher, Susan, Begtrup, M.   +3 more
core   +1 more source

Rhodium-Catalyzed Transarylation of Benzamides: C–C Bond vs C–N Bond Activation

, 2020
A rhodium-catalyzed transarylation of benzamides via selective C–C bond activation with arylboronic acids was described, which was distinct from the conventional metal-catalyzed C–N bond activation.
Yang Long (1521595), Zhishan Su (1395565), Shiyu He (8042639), Haifeng Xiang (742398), Xiangge Zhou (742399), Jing Zhong (230059), Yanling Zheng (603757)   +6 more
core   +1 more source

In silico identification of benzamide-based aryl halides as EGFR inhibitors: multi-ligand ADMET, pharmacophore mapping, and target prediction

In Silico Research in Biomedicine
Cancer is one of the greatest global health challenges, with specific costs of US$25 trillion by 2050, including treatment and socioeconomic impacts. The epidermal growth factor receptor (EGFR), a central tyrosine kinase, is a key target for anticancer ...
Caroline do Nascimento Gonçalves, Matheus Nunes da Rocha, Emmanuel Silva Marinho   +2 more
doaj   +1 more source

Electronic Smoking Devices Among University Students: Usage Patterns and Chemical Composition of Inhaled Substances

Analytical Science Advances, Volume 7, Issue 1, June 2026.
ABSTRACT This study investigated the prevalence of electronic smoking device (ESD) use and its associated behavioural and chemical risks among university students in Bahia, Brazil. A cross‐sectional survey was conducted with 355 students from public and private institutions through an online questionnaire between April and May 2023. Among participants,
Eduard F. Valenzuela, Raffael Silva Santos Almeida, Ivana Ferreira Simões, Aline Gonçalves Miranda, Magno Oliveira Ramos, Roberto Rodrigues Bandeira Tosta Maciel, Fernanda Warken Rosa, Aníbal de Freitas Santos Júnior   +7 more
wiley   +1 more source

Anticoccidial therapy small guide [PDF]

Medicamentul Veterinar, 2007
Being a major challenge, because of ingenious parasite's survival strategies and treatment's transience, anticoccidal therapy it is a major priority. In this respect, therapeutic conduct must be adjusted as well is possible on the most efficient drug ...
Cristina, T. Romeo
doaj  

Cholesterol and Cholesterol‐Derived Molecules Differentially Modulate Neuronal Kv7.2/7.3 Channels

Archiv der Pharmazie, Volume 359, Issue 6, June 2026.
Cholesterol, steroid hormones, and cholesterol‐based imidazolium salts (CHIMs) inhibit Kv7.2/Kv7.3 channels. Notably, NBD‐tagged CHIM‐L enhances currents. These findings demonstrate that both chemical modifications and linker length differentially modulate Kv7 activity, revealing variant‐specific sensitivities and potential pharmacological targets for ...
Elif Karabatak, Ronewa Nematswerani, Vivian Meiritz, Nicole Rychlik, Guiscard Seebohm, Frank Glorius, Thomas Budde   +6 more
wiley   +1 more source

Design, anticonvulsive and neurotoxic properties of retrobenzamides - N-(nitrophenyl)benzamides and N-(aminophenyl)benzamides

, 1999
Design, anticonvulsant properties in maximal electroshock-induced seizures [MES] and seizures induced by subcutaneous administration of pentetrazole (scPtz), and neurotoxicity of retrobenzamides (N-(nitrophenyl)benzamides and N-(aminophenyl) benzamides ...
Stables, JP., Vamecq, J., Vallee, L., Poupaert, Jacques, Bourhim, M   +4 more
core  

Mechanistic Insights into the Antimicrobial Effect of Benzodioxane-Benzamides Against Escherichia coli

Antibiotics
Background/Objectives: The bacterial cell division machinery is emerging as an attractive target for antimicrobial compounds. FtsZ, a highly conserved essential division protein, is the target for a number of small molecules such as benzamides.
Lorenzo Suigo, Alessia Lanzini, Valentina Straniero, William Margolin   +3 more
doaj   +1 more source

Gastrointestinal motility, prokinetic benzamides and serotonin : a study on the guinea-pig colon

, 1995
The prokinetic substituted benzamides stimulate gastrointestinal motility in animal models and in man. Studies done on the isolated guinea-pig ileum have led to the hypothesis that the benzamides act through facilitation of cholinergic transmission due ...
Briejer, M.R.
core