Results 101 to 110 of about 24,787 (257)

4-Bromo-N-(diethylcarbamothioyl)benzamide [PDF]

Acta Crystallographica Section E Structure Reports Online, 2009
The synthesis of the title compound, C(12)H(15)BrN(2)OS, involves the reaction of 4-bromo-benzoyl chloride with potassium thio-cyanate in dry acetone, followed by condensation of 4-bromo-benzoyl isothio-cyanate with diethyl-amine. The carbonyl and thio-carbonyl bond lengths indicate that these correspond to double bonds.
Binzet, Gün, Flörke, Ulrich, Külcü, Nevzat, Arslan, Hakan   +3 more
openaire   +4 more sources

Steroid Hormones Are Potent and Putatively Endogenous Activators of Human Bitter Taste Receptors

Annals of the New York Academy of Sciences, EarlyView.
Human bitter taste receptors are not only involved in sensing tastants within the oral cavity but also play crucial roles in internal tissues of the body. The current report identifies numerous structurally and functionally diverse steroid hormones as activators of the two human bitter taste receptors, TAS2R14 and TAS2R46.
Tatjana Lang, Francesco Ferri, Florian Ziegler, Antonella Di Pizio, Maik Behrens   +4 more
wiley   +1 more source

Assessment of labelled products with different radioanalytical methods: study on 18F-fluorination reaction of 4-[18F]fluoro-N-[2-[1-(2-methoxyphenyl)-1-piperazinyl]ethyl-N-2-pyridinyl-benzamide (p-[18F]MPPF) [PDF]

, 2010
Peer ...
Bergström, Kim, Koivula, Teija, Kämäräinen, Eeva-Liisa, Laine, Jaana, Lipponen, Tiina, Perhola, Outi, Solin, Olof   +6 more
core   +1 more source

N-(Naphthalen-1-yl)benzamide [PDF]

Acta Crystallographica Section E Structure Reports Online, 2011
In the title compound, C(17)H(13)NO, the N-H and C=O bonds are anti with respect to each other. The dihedral angle between the naphthalene ring system and the phenyl ring is 86.63 (5)°. In the crystal, N-H⋯O hydrogen bonds link mol-ecules into chains along [010].
Ruitao Zhu, Yuehong Ren, Wenjuan Li
openaire   +3 more sources

Harnessing benzamides as plant stress inhibitors, growth promoters and in management of crop resilience—A review

Plant Biology, EarlyView.
Benzamides boost crop resilience by inhibiting poly(ADP‐ribose) polymerase (PARP) to enhance stress tolerance and, through their antimicrobial, herbicidal, and insecticidal derivatives, they offer broad protection for sustainable crop improvement. Abstract Benzamides have emerged as potent stress inhibitors and growth promoters in plant biotechnology ...
M. J. Koetle, T. E. Motaung, S. O. Amoo
wiley   +1 more source

Synthesis of carbon-11-labeled CK1 inhibitors as new potential PET radiotracers for imaging of Alzheimer’s disease [PDF]

, 2018
The reference standards methyl 3-((2,2-difluoro-5H-[1,3]dioxolo[4′,5′:4,5]benzo[1,2-d]imidazol-6-yl)carbamoyl)benzoate (5a) and N-(2,2-difluoro-5H-[1,3]dioxolo[4′,5′:4,5]benzo[1,2-d]imidazol-6-yl)-3-methoxybenzamide (5c), and their corresponding ...
Gao, Mingzhang, Wang, Min, Zheng, Qi-Huang   +2 more
core   +2 more sources

Crystal Structures and Intermolecular Interactions in α$\alpha$‐ and β$\beta$‐phosgene

Angewandte Chemie, Volume 138, Issue 2, 9 January 2026.
Despite its notorious reputation as a war gas, phosgene (COCl2${\rm COCl}_2$) is one of the most important intermediate chemicals in industry. In this study, we present the crystal structures of two phosgene polymorphs as deduced from powder neutron diffraction and show which intermolecular interactions stabilise the different modifications.
Sven Ringelband, Jonathan Pfeiffer, A. Dominic Fortes, Christopher M. Howard, Stewart F. Parker, Antti J. Karttunen, Frank Tambornino   +6 more
wiley   +2 more sources

Species-specific pharmacology of Trichloro(sulfanyl)ethyl benzamides as transient receptor potential ankyrin 1 (TRPA1) antagonists

Molecular Pain, 2007
Agonists of TRPA1 such as mustard oil and its key component AITC cause pain and neurogenic inflammation in humans and pain behavior in rodents. TRPA1 is activated by numerous reactive compounds making it a sensor for reactive compounds in the body ...
Immke David C, Wang Weiya, Gao BaoXi, Tamir Rami, Klionsky Lana, Nishimura Nobuko, Gavva Narender R   +6 more
doaj   +1 more source

Making Blank Faces Expressive: Chemical Approaches to the Modification of Chemically Inert Peptides

Journal of Peptide Science, Volume 32, Issue 3, March 2026.
As an alternative to the conventional approach, which combines amino acid monomers in a one‐by‐one fashion to peptide derivatives, the chemical modification of existing peptides has attracted significant attention in recent years. However, such approaches generally target the reactive functional groups in cysteine and lysine residues, particularly in ...
Yoshitaka Moriyama, Hikari Sada, Takeshi Nanjo   +2 more
wiley   +1 more source

The search for the 'next' euphoric non-fentanil novel synthetic opioids on the illicit drugs market: current status and horizon scanning [PDF]

, 2019
Purpose: A detailed review on the chemistry and pharmacology of non-fentanil novel synthetic opioid receptor agonists, particularly N-substituted benzamides and acetamides (known colloquially as U-drugs) and 4-aminocyclohexanols, developed at the Upjohn ...
A Helander, A Regina La, A Schneir, AG Hayes, AG Hayes, AJ Krotulski, AJ Krotulski, ALA Mohr, C McKenzie, C Soussan, Craig McKenzie, D Fabregat-Safont, D Lednicer, D Lednicer, D Lednicer, D Lednicer, D Lednicer, D Papsun, E Gerace, GW Peng, I Metushi, IM McIntyre, J Seither, J Szmuszkovicz, J Szmuszkovicz, JB Zawilska, JK O’Donnell, K Domanski, K Koch, KA Rambaran, Kirti Kumari Sharma, KN Ellefsen, KT Vo, L Ventura, M Dziadosz, M Katselou, MC Hout Van, MH Baumann, MJ Jones, MP Prekupec, Niamh NicDaeid, NJ Harper, P Armenian, P Armenian, P Nikolaou, PF Voigtlander Von, PF Voigtlander Von, PF Voigtlander Von, RA Fujimoto, RA Lahti, RT Brittain, SA Harding, SC Ifeagwu, SP Elliott, Tim G. Hales, TP Rohrig, USAN Council, V Coopman, Vaidya Jayathirtha Rao, W Fleming, X Ruan, Z Davey, Z Li, ZH Liu   +63 more
core   +2 more sources