Results 21 to 30 of about 15,060 (197)

Bifunctional organocatalysts for the asymmetric synthesis of axially chiral benzamides

Beilstein Journal of Organic Chemistry, 2017
Bifunctional organocatalysts bearing amino and urea functional groups in a chiral molecular skeleton were applied to the enantioselective synthesis of axially chiral benzamides via aromatic electrophilic bromination.
Ryota Miyaji, Yuuki Wada, Akira Matsumoto, Keisuke Asano, Seijiro Matsubara   +4 more
doaj   +1 more source

Bioevaluation of Novel Anti-Biofilm Coatings Based on PVP/Fe3O4 Nanostructures and 2-((4-Ethylphenoxy)methyl)-N- (arylcarbamothioyl)benzamides

Molecules, 2014
Novel derivatives were prepared by reaction of aromatic amines with 2-(4-ethylphenoxymethyl)benzoyl isothiocyanate, affording the N-[2-(4-ethylphenoxymethyl) benzoyl]-Nꞌ-(substituted phenyl)thiourea.
Carmen Limban, Alexandru Vasile Missir, Alexandru Mihai Grumezescu, Alexandra Elena Oprea, Valentina Grumezescu, Bogdan Ștefan Vasile, Gabriel Socol, Roxana Trușcă, Miron Teodor Caproiu, Mariana Carmen Chifiriuc, Bianca Gălățeanu, Marieta Costache, Laurențiu Morușciag, Grațiela Pîrcălăbioru, Diana Camelia Nuță   +14 more
doaj   +1 more source

5-(4H)-Oxazolones and Their Benzamides as Potential Bioactive Small Molecules

Molecules, 2020
The five membered heterocyclic oxazole group plays an important role in drug discovery. Oxazolones present a wide range of biological activities. In this article the synthesis of 4-substituted-2-phenyloxazol-5(4H)-ones from the appropriate substituted ...
Evangelos Mavridis, Eleftherios Bermperoglou, Eleni Pontiki, Dimitra Hadjipavlou-Litina   +3 more
doaj   +1 more source

Experimental pharmacological research regarding some newly synthesized benzamides on central nervous system functions

Journal of Mind and Medical Sciences, 2017
Three newly synthesized benzamides by the Department of Pharmaceutical Chemistry of the Faculty of pharmacy from the University of Medicine and Pharmacy „Carol Davila” Bucharest were tested in order to determine whether these new molecules have similar ...
Cornel Chiriță, Emil Ștefănescu, Cristina D. Marineci, Simona Negreș, Diana C. Nuță   +4 more
doaj   +1 more source

N-(9,10-Dioxo-9,10-dihydroanthracen-1-yl)-2-methylbenzamide

Molbank, 2020
In the present Short Note, we report a synthesis for the title compound, N-(9,10-dioxo-9,10-dihydroanthracen-1-yl)-2-methylbenzamide by reacting 2-methylbenzoyl chloride (or 2-methylbenzoic acid) with 1-aminoanthraquinone. The synthesized target compound
Hamad H. Al Mamari, Ahmed Al Sheidi
doaj   +1 more source

N-(Cyanomethyl)benzamide [PDF]

Acta Crystallographica Section E Structure Reports Online, 2010
In the structure of the title compound, C(9)H(8)N(2)O, the amide group is twisted by a dihedral angle of 21.86 (7)° with respect to the benzene ring, while the planes of the benzene ring and cyano-methyl group form a dihedral angle of 53.13 (11)°. In the crystal structure, mol-ecules are linked via N-H⋯O hydrogen bonds, forming a chain running parallel
Abdelrhani Elachqar, Abdelilah El Hallaoui, Anouar Alami, Younas Aouine, Hafid Zouihri   +4 more
openaire   +3 more sources

Investigating Spectrum of Biological Activity of 4- and 5-Chloro-2-hydroxy-N-[2-(arylamino)-1-alkyl-2-oxoethyl]benzamides

Molecules, 2011
In this study, a series of twenty-two 5-chloro-2-hydroxy-N-[2-(arylamino)-1-alkyl-2-oxoethyl]benzamides and ten 4-chloro-2-hydroxy-N-[2-(arylamino)-1-alkyl-2-oxoethyl]benzamides is described.
Jirina Stolarikova, Jarmila Vinsova, Marcela Vejsova, Katarina Kralova, Ales Imramovsky, Matus Pesko, Josef Jampilek   +6 more
doaj   +1 more source

4-Iodo-N-(phenylsulfonyl)benzamide hemihydrate

IUCrData, 2017
In the title hemihydrate, 2C13H10INO3S·H2O, there are two organic molecules (A and B) and one water molecule in the asymmetric unit. The benzene rings are inclined to one another by 77.98 (1)° in A and 79.81 (9)° in B. The A and B molecules are connected
P. A. Suchetan, A. G. Sudha, E. Suresha, N. K. Lokanath, S. Naveen, Ismail Warad   +5 more
doaj   +1 more source

Electrochemically Driven Regioselective Radical Functionalization of Allenes: Scope and Mechanistic Insights

Advanced Science, EarlyView.
Allenes emerge as powerful platforms for electrochemical functionalization through radical pathways. Selective radical addition at the central carbon triggers anodic oxidation and intramolecular cyclization, enabling efficient synthesis of oxazolines and oxazolidine‐2‐imines without external oxidants.
Pranjal Pyne, Prateek Saini, Rohel Hoque, Shivam Pandey, Srinivasan Ramakrishnan, Chandra M. R. Volla   +5 more
wiley   +1 more source

Discovery of (phenylureido)piperidinyl benzamides as prospective inhibitors of bacterial autolysin E from Staphylococcus aureus

Journal of Enzyme Inhibition and Medicinal Chemistry, 2018
Autolysin E (AtlE) is a cell wall degrading enzyme that catalyzes the hydrolysis of the β-1,4-glycosidic bond between the N-acetylglucosamine and N-acetylmuramic acid units of the bacterial peptidoglycan.
Jure Borišek, Sara Pintar, Mitja Ogrizek, Simona Golič Grdadolnik, Vesna Hodnik, Dušan Turk, Andrej Perdih, Marjana Novič   +7 more
doaj   +1 more source