Results 41 to 50 of about 15,060 (197)
BiomedicinesHuman dihydrofolate reductase (hDHFR) is an essential cellular enzyme, and inhibiting its activity is a promising strategy for cancer therapy. We have chosen the trimethoprim molecule (TMP) as a model compound in our search for a new class of hDHFR ...
Danuta Drozdowska +3 more
doaj +1 more source
Microwave assisted green synthesis of aryl methoxylated benzamides and 2-oxazolines from biomass
Green Processing and Synthesis, 2013 This paper presents a simple, rapid and efficient green synthesis of aryl methoxylated benzamides and 2-oxazolines from renewable Eucalyptus biomass – tar derivatives.
Okuma Adriana Akemi +3 more
doaj +1 more source
Exploring the Synthesis of Metalloporphyrin Equipped Pd12L24 Supramolecular Spheres
Chemistry – A European Journal, EarlyView.We expand the scope of Pd12L24 nanospheres equipped with porphyrins. Focusing on the porphyrin metallation state, synthetic strategies for porphyrin building block (BB)compounds are developed. The compounds are evaluated against nanosphere self‐assembly conditions.
Tom Keijer +8 more
wiley +1 more source
Catalytic Cleavage of Lignin C–C Bonds and Subsequent Amination: A Valorization Roadmap
EcoEnergy, EarlyView.By systematically integrating the reaction pathway and mechanisms underlying lignin C–C bond cleavage and the subsequent product amination, this review aims to provide guidance for the rational design of multifunctional catalytic systems capable of coupling bond cleavage and amination reactions.
Jingxuan Zhang +6 more
wiley +1 more source
Molecules, 2022 To develop new compounds with high activity, broad spectrum and low-toxicity, 17 benzamides substituted with quinoline-linked 1,2,4-oxadiazole were designed using the splicing principle of active substructures and were synthesized.
Bin-Long Sun +7 more
doaj +1 more source
The Mechanism of Visible-Light Photochemical Rearrangements of Conjugated Amide Enolates. [PDF]
ChemistryVisible light irradiation of extended enolates of N‐benzylamides leads to homolytic C─N Bond cleavage, generating a biradical. Computational and mechanistic studies suggest rapid radical recombination within a solvent cage to give either ring‐expanded or rearranged products. ABSTRACT Deprotonation of conjugated amides forms colored solutions of lithium
Mortimer J +3 more
europepmc +2 more sources
Mass Spectrometry Reviews, EarlyView.ABSTRACT The use of MALDI mass spectrometry for the analysis of carbohydrates and glycoconjugates is a well‐established technique and this comprehensive review is the twelfth update of the original article published in 1999 and brings coverage of the literature to the end of 2024.
David J. Harvey
wiley +1 more source
Synthesis and Antifungal Activity of N-(3-(4-(1,3-dioxolan-2-yl) phenyl)-1,2,4-thiadiazol-5-yl) Benzamide Derivatives: An in-vitro Study [PDF]
Journal of Clinical and Diagnostic ResearchIntroduction: Fungal infections are associated with morbidity and mortality globally and immense economic burden. With the emergence of multidrug resistant fungal strains, it is essential to develop new antifungal drugs.
K Dayana +3 more
doaj +1 more source
2-(Methylsulfinyl)benzamide [PDF]
Acta Crystallographica Section E Structure Reports Online, 2010 In the crystal of the title compound, C(8)H(9)NO(2)S, synthesized by the oxidation of 2-(methyl-sulfan-yl)benzamide using NaOCl with 2,2,6,6-tetra-methyl-piperidyl-1-oxy (TEMPO) as the catalyst, mol-ecules are linked via inter-molecular N-H⋯O(amide) hydrogen bonds, forming centrosymmetric amide-amide dimers which are extended into a two-dimensional ...
openaire +3 more sources
Pest Management Science, EarlyView.Using cellular phenotyping and resistance profiling, we show that herbicides across the Herbicide Resistance Action Committee (HRAC) Groups 3 and 23 induce indistinguishable, dose‐dependent microtubule defects. Resistance patterns, rather than cellular phenotypes, reveal distinct sites of action and support reclassifying Group 3 as α‐tubulin binders ...
Katharina Kaprocki +6 more
wiley +1 more source