Results 41 to 50 of about 17,013 (236)

Antiallergic Activity of Substituted Benzamides: Characterization, Estimation and Prediction [PDF]

, 2007
Antiallergic activity of twenty-three substituted N 4-methoxyphenyl benzamides was model by the use of an original methodology. After sketching out the compounds structure and creating the file with the observed activities, strictly based on compounds ...
BOLBOACA, Dr. Sorana D., JÄNTSCHI, Dr. Lorentz   +1 more
core  

Cobalt-Promoted Dimerization of Aminoquinoline Benzamides

, 2016
A method for aminoquinoline-directed, cobalt-promoted dimerization of benzamides has been developed. Reactions proceed in ethanol solvent in the presence of Mn­(OAc)2 cocatalyst and Na2CO3 base and use oxygen as a terminal oxidant.
Liene Grigorjeva (1332981), Olafs Daugulis (1322985)   +1 more
core   +1 more source

Benzamide Trimethoprim Derivatives as Human Dihydrofolate Reductase Inhibitors—Molecular Modeling and In Vitro Activity Study

Biomedicines
Human dihydrofolate reductase (hDHFR) is an essential cellular enzyme, and inhibiting its activity is a promising strategy for cancer therapy. We have chosen the trimethoprim molecule (TMP) as a model compound in our search for a new class of hDHFR ...
Danuta Drozdowska, Agnieszka Wróbel-Tałałaj, Cezary Parzych, Artur Ratkiewicz   +3 more
doaj   +1 more source

Microwave assisted green synthesis of aryl methoxylated benzamides and 2-oxazolines from biomass

Green Processing and Synthesis, 2013
This paper presents a simple, rapid and efficient green synthesis of aryl methoxylated benzamides and 2-oxazolines from renewable Eucalyptus biomass – tar derivatives.
Okuma Adriana Akemi, Antônio Daphne Chiara, Carazza Fernando, Duarte Lucienir Pains   +3 more
doaj   +1 more source

An Electrochemical Way to Generate Amphiphiles from Hydrazones for the Synthesis of 1,2,4‐Triazole Scaffold Cyclic Compounds

ChemistryOpen, 2022
An electro‐oxidative cyclization pathway in which hydrazones are selected as starting materials to generate amphiphiles by reacting with benzylamines and benzamides was reported.
Wangyu Li, Mingteng Xiong, Xiao Liang, Dungai Wang, Heping Zhu, Prof. Dr. Yuanjiang Pan   +5 more
doaj   +1 more source

Nickel‐Catalyzed Three‐Component Difluoroalkylation‐Amination for the Direct Access to Anti‐Inflammatory β‐Difluoroalkyl Amines

Advanced Science, EarlyView.
A nickel‐catalyzed three‐component reductive fluoroalkylation‐amination strategy of N‐vinylamides for the direct access to the α‐amidyl‐β‐difluoroalkyl amines was reported here. The synthetic method features with broad substrate scope, mild conditions, high functional group tolerance, and convenience to handle.
Chang Xu, Fangting Ma, Fan Ding, Luyan Wang, Yunxi Li, Yunzhi He, Xingang Zhang, Siyu He, Dandan Liu   +8 more
wiley   +1 more source

Synthesis of Phthalimides: A New Entry via TBAI-Catalyzed Intramolecular Cyclization of 2-(Hydroxymethyl)benzamides

SynOpen, 2018
Herein we report an unprecedented metal-free TBAI/TBHP mediated C–N bond formation via intramolecular cyclization of 2-(hydroxymethyl)benzamides to furnish N-substituted phthalimides in excellent yields.
Kare Nagaraju, Nomula Rajesh, Palakodety Radha Krishna   +2 more
doaj   +1 more source

Effectiveness of anti-psychotics and related drugs in the Huntington French-speaking group cohort. [PDF]

PLoS ONE, 2014
PURPOSE: Huntington's disease is a rare condition. Patients are commonly treated with antipsychotics and tetrabenazine. The evidence of their effect on disease progression is limited and no comparative study between these drugs has been conducted.
Gaëlle Désaméricq, Guillaume Dolbeau, Christophe Verny, Perrine Charles, Alexandra Durr, Katia Youssov, Clémence Simonin, Jean-Philippe Azulay, Christine Tranchant, Cyril Goizet, Philippe Damier, Emmanuel Broussolle, Jean-François Demonet, Graca Morgado, Laurent Cleret de Langavant, Isabelle Macquin-Mavier, Anne-Catherine Bachoud-Lévi, Patrick Maison   +17 more
doaj   +1 more source

NiH‐Catalyzed Enantio‐ and Regioselective Hydroselenylation of Unactivated Alkenes

Advanced Science, EarlyView.
Nickel‐hydride‐catalyzed enantio‐ and regioselective hydroselenylation of unactivated alkenes provides access to chiral organoselenium compounds. Enantiodetermining Ni–H insertion followed by single‐electron diselenide activation generates selenyl radical.
Hyung‐Joon Kang, Jaehun Kim, Sungwoo Hong   +2 more
wiley   +1 more source

Stereospecific photochemical ring expansion of lithiated benzamides

, 2003
Treatment of N-benzyl benzamides with a strong base (LDA or t-BuLi) followed by irradiation with a 500 W tungsten lamp provides, according to the substitution pattern of the starting amides, either norcaradienes or cycloheptadienones by overall insertion
Jonathan Clayden, Clayden, Jonathan, Knowles, Faye E., Menet, Christel J., Christel J. Menet, Faye E. Knowles   +5 more
core   +1 more source