Results 61 to 70 of about 20,263 (222)
2-Hydroxy-N-phenylbenzamides and Their Esters Inhibit Acetylcholinesterase and Butyrylcholinesterase
The development of novel inhibitors of acetylcholinesterase (AChE) and butyrylcholinesterase (BuChE) represents a viable approach to alleviate Alzheimer’s disease.
Martin Krátký +5 more
doaj +1 more source
N,N'-1,2-Phenylenebis[4-(chloromethyl)benzamide] [PDF]
4 páginas, 1 esquema.-- This article is an open access article distributed under the terms and conditions of the Creative Commons Attribution license.N,N'-1,2-Phenylenebis[4-(chloromethyl)benzamide] (3) was obtained in 61% yield by nucleophilic acyl ...
Bachl, Jürgen, Díaz Díaz, David
core +2 more sources
Serotonin 5-HT4 Agonist Activity of a Series of Meso-Azanoradamantane Benzamides [PDF]
A series of meso-amino(methyl)azanoradamantane benzamides has been prepared and evaluated for 5-HT4agonism activity in the rat tunica muscularis mucosae (TMM) assay.
Becker, Daniel +3 more
core +1 more source
Ab-initio crystal structure analysis and refinement approaches of oligo p-benzamides based on electron diffraction data [PDF]
Ab-initio crystal structure analysis of organic materials from electron diffraction data is presented. The data were collected using the automated electron diffraction tomography (ADT) technique.
Brunklaus, Gunther +4 more
core +1 more source
N-(Pyrrolidin-1-ylcarbothioyl)benzamide [PDF]
In the title compound, C(12)H(14)N(2)OS, the pyrrolidine ring adopts an envelope conformation with the C atom at the 3-position as the flap and makes a dihedral angle of 65.80 (9)° with the benzene ring. In the crystal, N-H⋯O hydrogen bonds join c-glide related mol-ecules into chains extended along [001] that are further connected into (100) layers via
Al-Abbasi, Aisha A. +2 more
openaire +3 more sources
4-Iodo-N-(phenylsulfonyl)benzamide hemihydrate
In the title hemihydrate, 2C13H10INO3S·H2O, there are two organic molecules (A and B) and one water molecule in the asymmetric unit. The benzene rings are inclined to one another by 77.98 (1)° in A and 79.81 (9)° in B. The A and B molecules are connected
P. A. Suchetan +5 more
doaj +1 more source
A regioselective method for the synthesis of 1-(hydroxymethyl)-2,3-dihydropyrrolo[1,2-a]quinazolin-5(1H)-ones – close structural analogs of naturally occurring vasicinone alkaloids – is described.
Alla I. Vaskevych +5 more
doaj +1 more source
Azaadamantane Benzamide 5-HT4 Agonists: Gastrointestinal Prokinetic SC-54750 [PDF]
Azaadamantanone 1 was converted to a series of aminoazaadamantane benzamides 9a–d, which were profiled for serotonin receptor activity. Aminomethylazaadamantane SC-54750 is a potent 5-HT4 agonist and 5-HT3 antagonist with in vivo efficacy in ...
Becker, Daniel +3 more
core +1 more source
The title compound, C(15)H(12)N(2)O, is a derivative of 4-(amino-meth-yl)benzonitrile, an important pestcide inter-mediate. In the crystal structure, mol-ecules are linked via inter-molecular N-H⋯O hydrogen bonds, forming infinite chains.
Hong-Jun Zhu +4 more
openaire +3 more sources
Antiviral Mechanisms of N-Phenyl Benzamides on Coxsackie Virus A9
Enteroviruses are one of the most abundant groups of viruses infecting humans, and yet there are no approved antivirals against them. To find effective antiviral compounds against enterovirus B group viruses, an in-house chemical library was screened ...
Mira Laajala +7 more
doaj +1 more source

