Results 1 to 10 of about 16,265 (239)

Rh(III)-Catalyzed Annulation of Boc-Protected Benzamides with Diazo Compounds: Approach to Isocoumarins

Molecules, 2019
A mild rhodium-catalyzed annulation of Boc-protected benzamides with diazo compounds via C−C/C−O bond formation has been explored. In the presence of [Cp*RhCl2]2, AgSbF6 and Cs2CO3, Boc-protected benzamides can be effectively annulated to ...
Chunpu Li
exaly   +4 more sources

Synthesis and Single Crystal Structures of N-Substituted Benzamides and Their Chemoselective Selenation/Reduction Derivatives [PDF]

Molecules, 2021
A series of N-aryl-N-(2-oxo-2-arylethyl) benzamides and cinnamides has been prepared. The reaction of the benzamides with Woollins’ reagent, a highly efficient chemoselective selenation/reduction reagent, gave the corresponding N-aryl-N-(arylenethyl ...
Guoxiong Hua, Cameron L. Carpenter-Warren, David B. Cordes, Alexandra M. Z. Slawin, J. Derek Woollins   +4 more
doaj   +2 more sources

Photoredox-catalyzed arylation of isonitriles by diaryliodonium salts towards benzamides [PDF]

Beilstein Journal of Organic Chemistry
The arylation of isonitriles by diaryliodonium salts under photoredox conditions has been proposed for the first time. The suggested procedure allows preparing a broad range of benzamides using both symmetric and unsymmetric diaryliodonium salts under ...
Nadezhda M. Metalnikova, Nikita S. Antonkin, Tuan K. Nguyen, Natalia S. Soldatova, Alexander V. Nyuchev, Mikhail A. Kinzhalov, Pavel S. Postnikov   +6 more
doaj   +2 more sources

Management of Clozapine Induced Hypersalivation on Slow Stream Rehabilitation Ward [PDF]

BJPsych Open
Aims: Sialorrhoea (hypersalivation), a common side effect of clozapine can impact the quality of life of patients. At present, no drugs are licensed to manage clozapine-induced hypersalivation, but there are various practical and pharmacological ...
Neeti Sud, Yousra Ghandour
doaj   +2 more sources

QSAR study of benzylidene hydrazine benzamides derivatives with in vitro anticancer activity against human lung cancer cell line A459 [PDF]

Journal of Pharmacy & Pharmacognosy Research, 2023
Context: In the last decade, resistance to epidermal growth factor receptor-tyrosine kinase inhibitors (EGFR-TKIs) in lung cancer cases has been widespread. The discovery and development of new drugs need to be done to overcome the case.
Galih Satrio Putra, Melanny Ika Sulistyowaty, Tegar Achsendo Yuniarta, Yahmin Yahmin, Sumari Sumari, Charinrat Saechan, Takayasu Yamauchi   +6 more
doaj   +1 more source

Base-Promoted One-Pot Synthesis of Pyridine Derivatives via Aromatic Alkyne Annulation Using Benzamides as Nitrogen Source

Molecules, 2021
In the presence of Cs2CO3, the first simple, efficient, and one-pot procedure for the synthesis of 3,5-diaryl pyridines via a variety of aromatic terminal alkynes with benzamides as the nitrogen source in sulfolane is described. The formation of pyridine
Hina Mehmood, Muhammad Asif Iqbal, Muhammad Naeem Ashiq, Ruimao Hua   +3 more
doaj   +1 more source

Structure-Based Bioisosterism Design, Synthesis, Biological Evaluation and In Silico Studies of Benzamide Analogs as Potential Anthelmintics

Molecules, 2022
A recent screen of 67,012 compounds identified a new family of compounds with excellent nematicidal activity: the ortho-substituted benzamide families Wact-11 and Wact-12.
Franco Vairoletti, Margot Paulino, Graciela Mahler, Gustavo Salinas, Cecilia Saiz   +4 more
doaj   +1 more source

Determination and structural correlation of pKBH+ for meta- and para- substituted benzamides in sulfuric acid solutions [PDF]

Journal of the Serbian Chemical Society, 2006
The protonation of some meta and para substituted benzamides in sulfuric acid solutions was studied by UV spectroscopy in the 190–350 nm region. Principal component analysis was applied to separate the effect of protonation from the medium effect.
EMIL POPOVSKI, GORAN STOJKOVIC
doaj   +3 more sources

Synthesis and In Silico Evaluation of Potential Insecticide Activity of Benzamides

Chemistry Proceedings, 2021
In order to find alternative pesticides, a series of benzamide derivatives was synthesized. An in silico inverted virtual screening protocol considering the 13 common insecticide protein targets was used to evaluate the potential insecticide activity of ...
Miguel A. F. Ribeiro, Tatiana F. Vieira, Maria José G. Fernandes, Renato B. Pereira, David M. Pereira, Elisabete M. S. Castanheira, A. Gil Fortes, Sérgio F. Sousa, M. Sameiro T. Gonçalves   +8 more
doaj   +1 more source

4’-Methyl-2’-(quinolin-8-ylcarbamoyl)-biphenyl-4-carboxylic Acid Ethyl Ester

Molbank, 2020
In this short note communication, we report the synthesis of a novel amide 4’-methyl-2’-(quinolin-8-ylcarbamoyl)-biphenyl-4-carboxylic acid ethyl ester by the Ru-catalyzed C(sp2)-H bond arylation reaction.
Hamad H. Al Mamari, Anfal Al Hasani
doaj   +1 more source