Results 61 to 70 of about 18,814 (259)

Copper(I)-Catalyzed Synthesis of Substituted 2-Mercapto Benzimidazoles

open access: yes, 2016
An efficient method for the preparation of various substituted 2-mercapto benzimidazoles from their corresponding thioureas has been developed. S-Alkylation of thioureas followed by Cu-catalyzed intramolecular N-arylation furnished substituted 2-mercapto
Bhisma K. Patel (1479115)   +3 more
core   +1 more source

First Report of Anthelmintic Resistance in Gastrointestinal Nematodes in Goats in Romania

open access: yesAnimals, 2021
Currently, there are three classes of anthelmintics most commonly used in small ruminants: the benzimidazoles (BZs), macrocyclic lactones (MLs) and cholinergic agonists (especially levamisole; LEV).
Adrian Valentin Potârniche   +10 more
doaj   +1 more source

Accelerating Discovery of Organic Molecular Crystals via Materials Informatics and Autonomous Experiments

open access: yesAdvanced Intelligent Discovery, EarlyView.
Materials informatics and autonomous experimentation are transforming the discovery of organic molecular crystals. This review presents an integrated molecule–crystal–function–optimization workflow combining machine learning, crystal structure prediction, and Bayesian optimization with robotic platforms.
Takuya Taniguchi   +2 more
wiley   +1 more source

Preparation of Newer Fused Benzimidazoles

open access: yes, 1995
Nadkamy-Sacasa Research Laboratory, St Xavier's College, Bombay-400 001 Manuscript received 3 August 1993, revised 27 January 1994, accepted 8 February 1994 Preparation of Newer Fused ...
H. E. MASTER, J. R. KAMATH
core   +1 more source

Interactions médicamenteuses en médecine vétérinaire : exemple de benzimidazoles [PDF]

open access: yes, 2005
Les benzimidazoles sont des médicaments utilisés à la fois en médecine humaine et vétérinaire. Deux molécules appartenant à cette famille ont récemment été retirées du marché chez l'homme pour de sérieuses interactions médicamenteuses impliquant les ...
Labadie, Mathieu
core   +3 more sources

Importance of Fluorine in Benzazole Compounds

open access: yesMolecules, 2020
Fluorine-containing heterocycles continue to receive considerable attention due to their unique properties. In medicinal chemistry, the incorporation of fluorine in small molecules imparts a significant enhancement their biological activities compared to
Thuraya Al-Harthy   +2 more
doaj   +1 more source

The Link between Protein Kinase CK2 and Atypical Kinase Rio1

open access: yesPharmaceuticals, 2017
The atypical kinase Rio1 is widespread in many organisms, ranging from Archaebacteria to humans, and is an essential factor in ribosome biogenesis. Little is known about the protein substrates of the enzyme and small-molecule inhibitors of the kinase ...
Konrad Kubiński, Maciej Masłyk
doaj   +1 more source

Benzimidazoles Pharmacodynamics in Equine Strongyles

open access: yes, 2016
Our research aimed to assess the effectiveness of four benzimidazoles: albendazole, fenbendazole, mebendazole and thiabendazole against equine strongyles. The tests were performed between March 2015 and May 2016, on samples collected from 20 horses and 8
Csongor Olah   +3 more
core   +1 more source

Designer benzimidazoles: Synthesis, characterization, and applications [PDF]

open access: yes, 2008
The research presented in this thesis is centered on the design and synthesis of molecules which are derived from benzimidazoles and their applications. The first chapter provides an introduction to benzimidazoles and N-heterocyclic carbenes, a unique
Chao, Steven Tai-hsiang
core   +1 more source

Design, Synthesis and Evaluation of Antiproliferative Activity of New Benzimidazolehydrazones

open access: yesMolecules, 2016
The synthesis and antiproliferative activity of new benzimidazole derivatives bearing an hydrazone mojety at the 2-position is described. The new N′-(4-arylidene)-1H-benzo[d]imidazole-2-carbohydrazides were evaluated for their cytostatic activity toward ...
Valentina Onnis   +8 more
doaj   +1 more source

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