Results 1 to 10 of about 3,554 (196)

Molecular Conformations and Biological Activity of N-Hetaryl(aryl)alkyl-4-methyl-2,2-dioxo-1H-2λ⁶,1-benzothiazine-3-carboxamides

Scientia Pharmaceutica, 2018
The analysis of our previous studies on the search for synthetic analgesics among N-R-amides of bicyclic hetaryl-3-carboxylic acids has been performed; on its basis N-hetaryl(aryl)-alkyl-4-methyl-2,2-dioxo-1H-2λ6,1-benzothiazine-3-carboxamides have ...
Igor V. Ukrainets, Ganna M. Hamza, Anna A. Burian, Natali I. Voloshchuk, Oxana V. Malchenko, Svitlana V. Shishkina, Lina A. Grinevich, Vasyl V. Grynenko, Galina Sim   +8 more
doaj   +1 more source

Synthesis and characterization of N-substitutedphenyl -2-(4, 6-dimethoxypyrimidin-2-ylthio) benzylamines(N-取代苯基-2-（4，6-二甲氧基-2-嘧啶硫基）苄胺的合成和表征)

Zhejiang Daxue xuebao. Lixue ban, 2011
以2-巯基苯甲酸、取代苯胺和2-甲砜基-4，6-二甲氧基嘧啶为原料，经酰氯化、酰胺化、还原、亲核取代反应合成了一系列N-取代苯基-2-（4，6-二甲氧基-2-嘧啶硫基）苄胺类化合物，经氢核磁共振光谱、红外光谱、质谱和元素分析确证了它们的结构.
CHENYi-fei(陈一飞), ZHANGPei-zhi(张培志), SUNYan-ping(孙燕萍), WUJun(吴军)   +3 more
doaj   +1 more source

Synthesis and Structure-Affinity Relationships of Receptor Ligands with 1,3-Dioxane Structure

Pharmaceuticals
Background/Objectives: Ligands blocking σ1 receptors or NMDA receptors show promising pharmacological properties, such as analgesia or neuroprotection.
Elisabeth Quick, Dirk Schepmann, Bernhard Wünsch   +2 more
doaj   +1 more source

Integrated Network Pharmacology Analysis and Experimental Validation to Reveal the Mechanism of Anti-Insulin Resistance Effects of Moringa oleifera Seeds

Drug Design, Development and Therapy, 2020
Qiong Huang,1– 3,* Rong Liu,1– 3,* Jing Liu,1– 3 Qi Huang,1– 3 Shao Liu,1– 3 Yueping Jiang1– 3 1Department of Pharmacy, Xiangya Hospital, Central South University, Changsha 410008, People’s Republic of China ...
Huang Q, Liu R, Liu J, Huang Q, Liu S, Jiang Y   +5 more
doaj  

Programmable remodelling of carbon-nitrogen connectivity in amines. [PDF]

Nature
Robinson JD, Richard F, Ratkovich KA, Phelps JM, Gaunt MJ.   +4 more
europepmc   +1 more source

α-C-H Functionalization of Benzylamines: A Crucial Yet Challenging Transformation. [PDF]

Chemistry
Dinesh M S, Varghese IM, Mohanraj S, Das A.   +3 more
europepmc   +1 more source

Enantioselective Lithiation of <i>N</i>-Benzyl Ureas with a Chiral Lithium Amide: Dicyclopropylmethyl (Dcpm) as an Organolithium-Resistant Nitrogen Protecting Group. [PDF]

Org Lett
Schwarz M, Clayden J.
europepmc   +1 more source

Deaminative C(<i>sp</i>³)─C(<i>sp</i>³) Cross-Coupling of Benzylamines with Alcohols and Carboxylic Acids via Radical Sorting. [PDF]

J Am Chem Soc
Zhao WY, Takanashi N, Cabré A, Martinelli JR, MacMillan DWC.   +4 more
europepmc   +1 more source

Metal-free sustainable synthesis of oximes and hydrazones from benzyl alcohol and benzylamine. [PDF]

RSC Adv
Devgunde RB, Rupanawar BD, Rupnavar PB, Waghmode SB.   +3 more
europepmc   +1 more source

Excellent Catalytic Performances of a Au/C–CuO Binary System in the Selective Oxidation of Benzylamines to Imines under Atmospheric Oxygen

ACS Omega, 2021
Yuki Yamamoto, Miyuto Ota, Shintaro Kodama, Michio Ueshima, Akihiro Nomoto, Akiya Ogawa, Mitsunori Furuya, Kiminori Kawakami   +7 more
doaj   +1 more source