Results 101 to 110 of about 3,282 (218)
A highly efficient synthetic strategy for amidesviaoxidative amidation of benzaldehydes or benzylamines withN-substituted formamides has been developed using cobalt based heterogeneous catalyst.
Akhil V. Nakhate +4 more
core +1 more source
Reductive Amination with Zinc Borohydride. Efficient, Safe Route to Fluorinated Benzylamines
Fluorinated benzylamines are synthesized in high yields by reductive alkylation of secondary amines with appropriate fluoroaldehydes using a combination of zinc chloride and zinc borohydride.
Bhattacharyya, Sukanta +2 more
core +1 more source
Synthesis and Structure-Affinity Relationships of Receptor Ligands with 1,3-Dioxane Structure
Background/Objectives: Ligands blocking σ1 receptors or NMDA receptors show promising pharmacological properties, such as analgesia or neuroprotection.
Elisabeth Quick +2 more
doaj +1 more source
The rhodium(III)-catalyzed cross-coupling reaction between commercially available benzylamines and Morita-Baylis-Hillman (MBH) adducts is described. This protocol provides a facile access to various 2-benzazepine derivatives via the C(sp2)-H activation ...
Neeraj Kumar Mishra +9 more
core +1 more source
Qiong Huang,1– 3,* Rong Liu,1– 3,* Jing Liu,1– 3 Qi Huang,1– 3 Shao Liu,1– 3 Yueping Jiang1– 3 1Department of Pharmacy, Xiangya Hospital, Central South University, Changsha 410008, People’s Republic of China ...
Huang Q +5 more
doaj
Decomposition of Benzylamine Derivatives. III
Sunagawa, Genshun +2 more
openaire +4 more sources
Nickel-Catalyzed Benzylation of Aryl Alkenes with Benzylamines via C–N Bond Activation
We have developed the first example of nickel-catalyzed Heck-type benzylation of aryl olefins with various benzylamines as benzyl electrophiles, and the benzylic C–N bond cleavage was efficiently promoted by the amine–I2 charge transfer complex (CT ...
Hui Yu (27723) +2 more
core +1 more source
Rh(III)‐Catalyzed Synthesis of Multisubstituted Isoquinolines from Benzylamines and Diazo Compounds
International audienceMultisubstituted isoquinolines have been prepared by Rh(III)-catalyzed cyclization of benzylamines with diazo compounds via aryl C-H bond activation using molecular oxygen from air as an oxidant.
Xiuling Cui +11 more
core +1 more source
Base and solvent dependency of an oxidative retro-alkylation of secondary and tertiary benzylamines
An iodine and caesium carbonate amine oxidation protocol is described. Non-branched secondary benzylamines were cleanly oxidised to aldimines that could be isolated without the need for chromatography.
Feula, A., Fossey, J.S.
core +1 more source
Novel syntheses by directed lithiations of N-Boc benzylamines and cyclopropylamines
The lithiation-substitution of N-Boc benzylamines and cyclopropylamines have been investigated to explore the synthetic potential of these substrates. We have achieved the syntheses of highly enantioenriched benzylic $\alpha$-substituted N-Boc secondary ...
Park, Yong Sun
core

