Results 131 to 140 of about 27,094 (219)

Editorial Expression of Concern: The bromodomain and extra-terminal inhibitor CPI203 enhances the antiproliferative effects of rapamycin on human neuroendocrine tumors. [PDF]

Cell Death Dis
Wong C, Laddha SV, Tang L, Vosburgh E, Levine AJ, Normant E, Sandy P, Harris CR, Chan CS, Xu EY.   +9 more
europepmc   +1 more source

Development of a Lysine-Reactive Targeted Covalent Inhibitor for the P300/CBP-Associated Factor Bromodomain Through Structure-Based Design. [PDF]

ChemMedChem
Ede RR, Peterson KE, Begyinah RK, Tom IP, Ochoada JM, Sneddon MS, Tiu AKY, Fischer M, Shelat AA, Pomerantz WCK.   +9 more
europepmc   +1 more source

Structural insights into the recognition of mono- and di-acetyllysine by the ATAD2B bromodomain

, 2017
Click on the Resource Link to find this item in the ACPHS Library catalog.The ATPase family, AAA+ domain-containing protein 2B (ATAD2B) is a nuclear protein that may play a role in the development of neuronal tissues and tumorigenesis. The ATAD2B protein
Lloyd, Jonathan '17
core  

BRD4 binds the nucleosome via both histone and DNA interactions. [PDF]

Mol Cell
Zhu J, Leith EM, O'Donnell EN, Manzano BP, Wu SY, Chiang CM, Armache JP, Tan S.   +7 more
europepmc   +1 more source

Unusual backfolded binding poses of BAZ2A bromodomain binders. [PDF]

Acta Crystallogr D Struct Biol
Dalle Vedove A, Cazzanelli G, D'Agostino VG, Vargas Rosales PA, Caflisch A, Lolli G.   +5 more
europepmc   +1 more source

Bridging BET bromodomain and immune checkpoint inhibitors through generative bioorganic frameworks for next-generation cancer immunotherapy. [PDF]

RSC Med Chem
Diab MK, Yassen ASA, Fahmy SA, Ashour HF, Nafie MS.   +4 more
europepmc   +1 more source

Parasite-specific essential bromodomain protein TgBDP4 is a key epigenetic reader and a potential drug target for the parasite Toxoplasma gondii. [PDF]

J Biol Chem
Gurupwar R, Khandavalli CR, Deshmukh AS.
europepmc   +1 more source

Advances in Mechanism of Action and Efficacy of CBP/p300 Inhibitors in Different Subtypes of Breast Cancer. [PDF]

Molecules
Yang Y, Yang T, Lin Y, Gan L.
europepmc   +1 more source

PAX3-FOXO1 Contacts BRD4 through Its Acetylated Intrinsically Disordered Region. [PDF]

Biochemistry
Fraser OA, Schleicher MN, Pagano ML, Showalter SA.   +3 more
europepmc   +1 more source

Chromatin dynamics and cellular energy homeostasis. [PDF]

J Biochem
Suganuma T, Workman JL.
europepmc   +1 more source