Results 131 to 140 of about 1,018 (177)

Discovery of benzyl carbamate inhibitors of coronavirus M^pro enzymes from a legacy collection of cysteine protease inhibitors. [PDF]

J Enzyme Inhib Med Chem
Sá Magalhães Serafim M, Kronenberger T, Francisco KR, de Sousa Reis EV, Gonçalves de Oliveira E, Marcelino E Oliveira FK, Serraglio Fortes I, Maciel Fernandes TH, Barbosa da Silva E, Fajtova P, Skinner DE, Syed RO, Lage de Siqueira-Neto J, Poso A, Fernandes Mota BE, Alves Coelho-Dos-Reis JG, Santos Abrahão J, Gonçalves Maltarollo V, O'Donoghue AJ, Caffrey CR.   +19 more
europepmc   +1 more source

Discovery of a Potent Triazole-Based Reversible Targeted Covalent Inhibitor of Cruzipain. [PDF]

ACS Med Chem Lett
Cerutti JP, Diniz LA, Corrêa Santos V, Vilchez Larrea SC, Alonso GD, Ferreira RS, Quevedo MA, Dehaen W.   +7 more
europepmc   +1 more source

Structure Elucidation, Biosynthetic Gene Cluster Distribution, and Biological Activities of Ketomemicin Analogs in <i>Salinispora</i>. [PDF]

Mar Drugs
Castro-Falcón G, Guillén-Matus DG, Silva EBD, Guo W, Ross A, Sá Magalhães Serafim M, Fernandes THM, Tantillo DJ, O'Donoghue AJ, Jensen PR.   +9 more
europepmc   +1 more source

The pH-Dependent Specificity of Cathepsin S and Its Implications for Inflammatory Communications and Disease. [PDF]

Biochemistry
DeHority R, Gil Pineda LI, Cochran K, Chen B, Bratek D, Helm RF, Lemkul JA, Zhang C.   +7 more
europepmc   +1 more source

Synthesis and Biological Evaluation of New Chalcogen Semicarbazone (<i>S</i>, <i>Se</i>) and Their Azole Derivatives against Chagas Disease. [PDF]

J Med Chem
Rubio-Hernández M, Alcolea V, Barbosa da Silva E, Giardini MA, M Fernandes TH, Martínez-Sáez N, O'Donoghue AJ, Siqueira-Neto JL, Pérez-Silanes S.   +8 more
europepmc   +1 more source

Chalcogen Derivatives for the Treatment of African Trypanosomiasis: Biological Evaluation of Thio- and Seleno-Semicarbazones and Their Azole Derivatives. [PDF]

ACS Omega
Rubio-Hernández M, Teixeira TR, Nguyen TP, Shingyoji M, da Silva EB, O'Donoghue AJ, Caffrey CR, Pérez-Silanes S, Martínez-Sáez N.   +8 more
europepmc   +1 more source

Marine Pharmacology in 2022-2023: Marine Compounds with Antibacterial, Antidiabetic, Antifungal, Anti-Inflammatory, Antiprotozoal, Antituberculosis and Antiviral Activities, Affecting the Immune and Nervous Systems, and Other Miscellaneous Mechanisms of Action. [PDF]

Mar Drugs
Mayer AMS, Mayer VA, Swanson-Mungerson M, Pierce ML, Roberts CM, Rodríguez AD, Nakamura F, Taglialatela-Scafati O.   +7 more
europepmc   +1 more source

Marine Cyanobacteria: A Rich Source of Structurally Unique Anti-Infectives for Drug Development. [PDF]

Molecules
Tan LT, Salleh NF.
europepmc   +1 more source

Host-Directed Therapies Based on Protease Inhibitors to Control <i>Mycobacterium tuberculosis</i> and HIV Coinfection. [PDF]

Microorganisms
Mandal M, Pires D, Azevedo-Pereira JM, Anes E.   +3 more
europepmc   +1 more source