Results 231 to 240 of about 83,038 (344)
Sulfenate anion catalyzed enantio- and diastereoselective aziridination. [PDF]
Pu Y, Smaldone AM, Adrio J, Walsh PJ.
europepmc +1 more source
Iturin A is an antifungal lipopeptide with broad applications. Here, we present a novel synthesis and semisynthesis of trifluoromethylated iturin A analogues. Their antifungal activity was evaluated against Fusarium graminearum and Candida albicans.
Periklis Karamanis +5 more
wiley +1 more source
Catalytic enantioselective total synthesis of antitubercular agents (-)-bedaquiline and (-)-sudapyridine enabled by dynamic kinetic resolution-asymmetric transfer hydrogenation. [PDF]
Han J, Zhang D, Tao Y, Tang P, Chen FE.
europepmc +1 more source
Isomerization of α‐Pinene Oxide to Trans‐Pinocarveol
An operationally simple protocol for the selective isomerization of α‐pinene oxide (APO) to trans‐pinocarveol (TPC) is disclosed, which leverages inexpensive pyridinium‐halide organocatalysts to mitigate competing 1,2‐alkyl shifts. The scalability of this methodology is demonstrated on a decagram scale and catalyst‐recycling is validated through the ...
Emanuel Studer +2 more
wiley +1 more source
Stereoselective Pudovik reaction of aldehydes, aldimines, and nitroalkenes with CAMDOL-derived H-phosphonate. [PDF]
Li N +6 more
europepmc +1 more source
Piperazine Derivatives: A Privileged Scaffold in Modern Synthesis and Medicinal Chemistry
Piperazine‐based bioactive molecules represent a versatile class of compounds with broad therapeutic potential. Structural modification of the piperazine scaffold governs key structure–activity relationships, enabling antibacterial, antifungal, antitumor, neuroactive, and anti‐inflammatory activities.
Assel Ten +5 more
wiley +1 more source
Unified Enantioselective Synthesis of 5-Phenylmorphans and <i>cis</i>-Octahydroisoquinolines. [PDF]
Mahgoub AA +3 more
europepmc +1 more source

