Results 141 to 150 of about 611 (196)
O,S,Se-containing Biginelli products based on cyclic β-ketosulfone and their postfunctionalization. [PDF]
Beilstein J Org ChemDil KV, Palchykov VA.
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Synthesis and anticancer activity of new dihydropyrimidinone derivatives
European Journal of Medicinal Chemistry, 2018A series of dihydropyrimidinone derivatives bearing various N-heterocyclic moieties was designed and synthesized. Twelve new compounds were screened for their cytotoxic activity using 60 cancer cell lines according to NCI (USA) protocol. Compound 19 showed a significant activity against NCI-H460, SK-MEL-5, and HL-60 (TB) cell lines with growth ...
Amany S Mostafa, Khalid B Selim
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The Biginelli Dihydropyrimidinone Synthesis [PDF]
ChemInform, 2004 AbstractFor Abstract see ChemInform Abstract in Full Text.
C. Oliver Kappe, Alexander Stadler
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SAR studies on dihydropyrimidinone antibiotics [PDF]
Bioorganic & Medicinal Chemistry Letters, 2011 There is an urgent need for the development of novel antimicrobial agents that offer effective treatment against MRSA. Using a new class of dipeptide antibiotic TAN-1057A/B as lead, we designed, synthesized and evaluated analogs of TAN-1057A/B. Several novel dihydropyrimidinone antibiotics demonstrating comparable antibiotic efficacy while possessing ...
Lianhong, Xu +14 more
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Synthesis and carbonic anhydrase inhibitory properties of tetrazole- and oxadiazole substituted 1,4-dihydropyrimidinone compounds [PDF]
Artificial Cells, Nanomedicine and Biotechnology, 2014 A new series of tetrazole-, oxadiazole-and cyanosubstituted 1,4-dihydropyrimidinone compounds were synthesized, and their inhibitory effects on the activity of purified human carbonic anhydrase (hCA) I were evaluated.
Mustafa Arslan +2 more
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New Journal of Chemistry, 2023
A series of chromene-dihydropyrimidinone and xanthene-dihydropyrimidinone hybrid compounds were easily synthesized through a multicomponent reaction followed by the copper-catalyzed alkyne–azide cycloaddition reaction.
Samuel J. Santos +7 more
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A series of chromene-dihydropyrimidinone and xanthene-dihydropyrimidinone hybrid compounds were easily synthesized through a multicomponent reaction followed by the copper-catalyzed alkyne–azide cycloaddition reaction.
Samuel J. Santos +7 more
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Synthesis and in vitro study of antiproliferative benzyloxy dihydropyrimidinones
Archiv der Pharmazie, 2021AbstractIn this study, we report on antiproliferative benzyloxy dihydropyrimidinones (DHPMs) produced by the Biginelli reaction of benzyloxy benzaldehyde, urea, and diverse 1,3‐diones. The reaction was catalyzed by lanthanum triflate and completed within 1–1.5 h, with 74–97% yield.
Ruturajsinh M. Vala +7 more
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Recent Advance in the Pharmacology of Dihydropyrimidinone
Mini-Reviews in Medicinal Chemistry, 2012Dihydropyrimidinones (DHPMs) are a series of highly valuable small molecules possessing versatile pharmaceutical properties. Although the first one-pot synthesis of DHPMs had been reported more than 100 years ago, the fascinating achievement in DHPMs-based pharmacology during the past century promoted durative interests to the pharmacological and ...
J-P, Wan, Y, Pan
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A Versatile Synthesis of DihydropyrimidinoneC‐Nucleosides
Nucleosides, Nucleotides and Nucleic Acids, 2004AbstractFor Abstract see ChemInform Abstract in Full Text.
Ram Chandra, Mishra +3 more
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Stereoselective synthesis of new dihydropyrimidinone glycoconjugates #
Journal of Heterocyclic Chemistry, 2005AbstractChemInform is a weekly Abstracting Service, delivering concise information at a glance that was extracted from about 200 leading journals. To access a ChemInform Abstract, please click on HTML or PDF.
G. V. M. Sharma +3 more
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