Results 111 to 120 of about 1,283,132 (206)

Phospholipid flippases ATP8A1 and ATP8A2 regulate GABA_A receptor trafficking through distinct mechanisms in hippocampal neurons. [PDF]

iScience
Kawase M, Tokunaga S, Umemura Y, Shawki HH, Omi J, Hoshiai A, Ohshima T, Nakajima T, Kohno T, Sakurai T, Aoki J, Oishi H, Hattori M.   +12 more
europepmc   +1 more source

AMPA and GABAA receptor nanodomains assemble in the absence of synaptic neurotransmitter release. [PDF]

Front Mol Neurosci, 2023
Ramsay HJ, Gookin SE, Ramsey AM, Kareemo DJ, Crosby KC, Stich DG, Olah SS, Actor-Engel HS, Smith KR, Kennedy MJ.   +9 more
europepmc   +1 more source

Gallic Acid-Mediated Enhancement of Diazepam-Induced Sedation via GABA_A Receptor Modulation: In Vivo and In Silico Evaluation. [PDF]

Food Sci Nutr
Yana NT, Chakrabarty A, Saha CK, Siddiqi NJ, Alnazhan N, Al Hasan MS, Nun FK, Rakib IH, Shipon MNH, Mia E, Jony MA, Hasan AMW, Hasan AMW, Islam MT, Khan AA.   +14 more
europepmc   +1 more source

Activation of endothelial GABA_A receptor α1 subunit protects against barrier dysfunction in acute lung injury. [PDF]

BMC Pulm Med
Zhou S, He X, Ni X, Wang A, Xu X.
europepmc   +1 more source

Global emergence and γ-aminobutyric acid type A (GABA_A) receptor activity of the new designer benzodiazepine ethylbromazolam. [PDF]

Arch Toxicol
Norman C, Acreman D, Bissram M, Curtis B, Hamer S, Westphal F, Putz M, Stefan C, Delaney SR, Lines R, McLeod MD, McDonald K, Green H.   +12 more
europepmc   +1 more source

A frameshift variant in FAM129C contributes to achalasia through B cell responses against the GABA_A receptor. [PDF]

Nat Commun
Li XQ, Li XY, Chen WF, Xu ZY, Liu ZQ, Wang Y, Zhang JY, Gu YY, Yao L, Tan YF, Chen XJ, Deng B, Wang KH, Xu JQ, He MJ, Geng ZH, Fan KY, Zhang ZC, Wang L, Xiang AY, Pan HT, Hu ZB, Xie YL, Wang C, Zhou PH, Li QL.   +25 more
europepmc   +1 more source

Synthesis, Spectroscopic Characterization, Molecular Docking Studies Toward the GABA_A Receptor, ADMET Prediction, GABA Aminotransferase Inhibition, and Anxiolytic Evaluation of Novel Thiazine Derivatives. [PDF]

Pharmaceuticals (Basel)
Sonu, Thajudeen KY, Alshehri SA, Ahmed MM, Porwal M, Verma S.   +5 more
europepmc   +1 more source

Editorial: The GABAA receptor: a target of pharmacologically active molecules. [PDF]

Front Pharmacol
Ernst M, Lu W, Mattei C.
europepmc   +1 more source

Activation of the human β3 GABA_A receptor by combinations of receptor protonation with chemical agonists and gain-of-function mutations. [PDF]

Biochem Pharmacol
Germann AL, Pierce SR, Steinbach JH, Akk G.   +3 more
europepmc   +1 more source

Improving Proteostasis of Trafficking-Deficient GABA_A Receptor Variants by Activating IRE1. [PDF]

ACS Chem Neurosci
Fu X, Wang YJ, Lee K, Ahn LY, Chen X, Harvey BT, Wang M, Seibert H, Zhang PP, Guerrero A, Schaffer AE, Richards CI, Wiseman RL, Kelly JW, Mu TW.   +14 more
europepmc   +1 more source