Results 201 to 210 of about 199,077 (362)

BGATT-GR: accurate identification of glucocorticoid receptor antagonists based on data augmentation combined with BiGRU-attention. [PDF]

Sci Rep
Shoombuatong W, Mookdarsanit P, Schaduangrat N, Mookdarsanit L.   +3 more
europepmc   +1 more source

Tissue-specific regulation of glucocorticoid receptor mRNA by dexamethasone.

, 1987
Judith E. Kalinyak, Richard I. Dorin, Andrew R. Hoffman, A J Perlman   +3 more
openalex   +1 more source

Ethnomedicinal Uses, Phytochemistry, Pharmacological Activities, and Toxicology of the Subfamily Gomphrenoideae (Amaranthaceae): A Comprehensive Review

Chemistry &Biodiversity, EarlyView.
ABSTRACT The subfamily Gomphrenoideae is composed of about 480 accepted species, many of which have been historically used as medicinal plants, reason why they have been studied in terms of chemical profile, biological activity, and safety. This review consolidates the advances in research on this subfamily over the past 47 years, emphasizing its ...
Dayanna Isabel Araque Gelves, Giulia Cristina de Andreoli Souza, Alvaro Jose Hernandez Tasco, Marcos José Salvador   +3 more
wiley   +1 more source

Neutrophil elastase produces 52-kD and 30-kD glucocorticoid receptor fragments in the cytosol of human leukemia cells [PDF]

, 1987
CW Distelhorst, KE Janiga, KJ Howard, SE Strandjord, Campbell Ej   +4 more
openalex   +1 more source

Synthesis and Biological Evaluation of Bicyclic Pyrazolines with Promising Antimicrobial Activities

ChemMedChem, EarlyView.
Continuous flow technology is exploited for the generation of bicyclic pyrazolines via photo‐click reactions. These heterocyclic species contain a valuable 3D scaffold along with a polar succinimide moiety. Subsequent antimicrobial testing reveals that halogenated moieties such as chlorine atoms and trifluoromethoxy groups enhance the potency of these ...
Debora Caviglia, Anna Maria Schito, Susanna Penco, Chiara Brullo, Marcus Baumann   +4 more
wiley   +1 more source

Nuclear Localization of Unoccupied Receptors for Glucocorticoids, Estrogens, and Progesterone in GH³Cells*

, 1985
Wade V. Welshons, BARBARA M. KRUMMEL, Jack Gorski   +2 more
openalex   +1 more source

The endogenous heat-stable glucocorticoid receptor stabilizing factor and the H-2 locus [PDF]

, 1982
Karen L. Leach, Robert P. Erickson, William B. Pratt   +2 more
openalex   +1 more source

Pharmacokinetics, Safety, and Tolerability of Single‐Dose Dazukibart in Healthy Adults in China and Japan: Results From 2 Randomized, Double‐Blind, Phase 1 Studies

Clinical Pharmacology in Drug Development, EarlyView.
Abstract Dazukibart is a humanized monoclonal antibody selectively targeting interferon‐β. The pharmacokinetics (PK), safety, tolerability, and immunogenicity of dazukibart were evaluated in 2 double‐blind, randomized, placebo‐controlled, single‐dose, Phase 1 studies in healthy adults in China (Study 1: N = 18; dazukibart 900 mg = 15; placebo = 3) and ...
Naihan Chen, Yamato Sano, Xiaohong Wang, Shuiyi Hu, Junichi Tabira, Xin Luo, Hiroki Yoshimatsu, John Prybylski, Myron Chu, Haiyan Li, Kenji Takazawa   +10 more
wiley   +1 more source

Glucocorticoid receptors recognize DNA sequences in and around murine mammary tumour virus DNA.

, 1982
Sabine Geisse, Claus Scheidereit, H.M. Westphal, Nancy E. Hynes, Bernd Groner, Miguel Beato   +5 more
openalex   +1 more source

Stable Overproduction of Intact Glucocorticoid Receptors in Mammalian Cells Using a Selectable Glucocorticoid Responsive Dihydrofolate Reductase Gene [PDF]

, 1989
Deborah L. Bellingham, John A. Cidlowski
openalex   +1 more source