Results 91 to 100 of about 4,568 (194)
Supplemental Figure 4 from Combination Drug Scheduling Defines a “Window of Opportunity” for Chemopotentiation of Gemcitabine by an Orally Bioavailable, Selective ChK1 Inhibitor, GNE-900
, 2023 Elizabeth Blackwood, Jennifer Epler, Ivana Yen, Michael Flagella, Tom O’Brien, Marie Evangelista, Stephen Schmidt, Yang Xiao, Jonathan Choi, Kaska Kowanetz, Judi Ramiscal, Kenton Wong, Diana Jakubiak, Sharon Yee, Gary Cain, Lewis Gazzard, Karen Williams, Jason Halladay, Peter K. Jackson, Shiva Malek +19 moreopenalex +1 more sourceBRD4 PROTAC Degradation Agent GNE-987 Inhibits Acute Myeloid Leukemia by Targeting Super Enhancers [PDF]
, 2021 Xu Sang, Yongping Zhang, Fang Fang, Li Gao, Yanfang Tao, Xiaolu Li, Zimu Zhang, Jianwei Wang, Yuanyuan Tian, Zhiheng Li, Di Yao, Yumeng Wu, Xinran Chu, Kunlong Zhang, Li Ma, Lihui Lu, Yanling Chen, Juanjuan Yu, Ran Zhuo, Shuiyan Wu, Zhen Zhang, Jian Pan, Shaoyan Hu +22 moreopenalex +1 more sourceDiscovery of GNE-502 as an orally bioavailable and potent degrader for estrogen receptor positive breast cancer
, 2021 Jennifer E. Klomp, Jun Liang, Jun Li, Robert A. Blake, Jae H. Chang, Lori S. Friedman, Simon Goodacre, Steven J. Hartman, Ellen Ingalla, James R. Kiefer, Tracy Kleinheinz, Sharada S. Labadie, Tommy Lai, Jiangpeng Liao, Nev McLean, Ciara Metcalfe, Vidhi Mody, Michelle Nannini, Daniel F. Ortwine, Yingqing Ran, Nick Ray, Fabien Roussel, Amy Sambrone, Deepak Sampath, Maia Vinogradova, John Wai, Tao Wang, Kuen Yeap, Birong Zhang, Xiaoping Zheng, Yu Zhong, Xiaojing Wang +31 moreopenalex +1 more sourceGNE-886: A Potent and Selective Inhibitor of the Cat Eye Syndrome Chromosome Region Candidate 2 Bromodomain (CECR2)
, 2017 Terry D. Crawford, James E. Audia, S.F. Bellon, Daniel J. Burdick, Archana Bommi‐Reddy, Alexandre Côté, Richard Cummings, Martin Duplessis, E. Megan Flynn, Michael C. Hewitt, Hon-Ren Huang, Hariharan Jayaram, Ying Jiang, Shivangi Joshi, James R. Kiefer, Jeremy Murray, Christopher G. Nasveschuk, Arianne Neiss, Eneida Pardo, F. Anthony Romero, Péter Sandy, Robert J. Sims, Yong Tang, Alexander M. Taylor, Vickie Tsui, Jian Wang, Shumei Wang, Yongyun Wang, Zhaowu Xu, Laura E. Zawadzke, Xiaoqin Zhu, Brian K. Albrecht, Steven Magnuson, Andrea G. Cochran +33 moreopenalex +2 more sourcesNovel Pathogenic Variants in a French Cohort Widen the Mutational Spectrum of GNE Myopathy
, 2015 Mathieu Cérino, Svetlana Gorokhova, Anthony Béhin, Jon Andoni Urtizberea, Virginie Kergourlay, Eric Salvo, Rafaëlle Bernard, Nicolas Lévy, Marc Bartoli, Martin Krahn +9 moreopenalex +2 more sources