Results 71 to 80 of about 524 (174)

NanoLuc Luciferase as a Fluorogen-Activating Protein for GFP Chromophore Based Fluorogens. [PDF]

open access: yesInt J Mol Sci, 2023
Bogdanova YA   +11 more
europepmc   +1 more source

Synthesis and pharmacological evaluation of new imidazolones planned as inhibitors of cysteine proteases for the treatment of leukemia

open access: yes, 2013
A palavra câncer é utilizada para designar um conjunto de mais de 100 doenças diferentes que têm, em comum, o crescimento desordenado de células anormais que invadem tecidos e órgãos, e é considerada pela Organização Mundial da Saúde um dos maiores ...
Azevedo, Luciana Luiz de
core  

Palladation and functionalization of pyrimidinones and imidazolones

open access: yes, 2018
Depuis ces dix dernières années, notre laboratoire a développé une expertise dans le domaine de la fonctionnalisation de liaisons carbone-hydrogène (dite fonctionnalisation C-H) d’hétérocycles par catalyse aux métaux de transition.
Collado Ruiz, Sandra
core  

Synthèse et fonctionnalisation directe catalytique de la liaison C-H d'imidazolones : nouvel accès aux fluorophores analogues de la GFP

open access: yes, 2017
Imidazolones have been studied for a long time, either as bioactive molecules or for their fluorescence properties, the best known example being the Green Fluorescent Protein or GFP.
Muselli, Mickaël
core  

General Installation of (4H)‑Imidazolone cis-Amide Bioisosteres Along the Peptide Backbone

open access: yes
Imidazolones represent an important class of heterocycles present in a wide range of pharmaceuticals, metabolites, and bioactive natural products and serve as the active chromophore in green fluorescent protein.
Krishna K. Sharma (2403073)   +4 more
core   +1 more source

Discovery of novel quinoline-based analogues of combretastatin A-4 as tubulin polymerisation inhibitors with apoptosis inducing activity and potent anticancer effect. [PDF]

open access: yesJ Enzyme Inhib Med Chem, 2021
Ibrahim TS   +8 more
europepmc   +1 more source

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