Indole-ynones as Privileged Substrates for Radical Dearomatizing Spirocyclization Cascades [PDF]
, 2022 Indole-ynones have been established as general substrates for radical dearomatizing spirocyclization cascade reactions. Five distinct and varied synthetic protocols have been developedcyanomethylation, sulfonylation, trifluoromethylation, stannylation ...
Jason M. Lynam +17 more
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Synthesis of Indole-Fused Six, Seven or Eight-Membered N,O-Heterocycles via Rhodium-Catalyzed NH-Indole-Directed CH Acetoxylation/Hydrolysis/Annulation [PDF]
, 2021 We report herein the facile synthesis of indole-fused six-, seven-, or eight-membered N,O-heterocycles through rhodium-catalyzed C–H acetoxylation/hydrolysis/annulation. The notable features of this method include C–H acetoxylation using NH-indole as the
Leipeng Lu +7 more
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Indole-Fused Benzoxepine Synthesis via Visible-Light-Driven Aerobic Dehydrogenative [5 + 2] Annulation [PDF]
, 2023 A photocatalyzed oxidative dehydrogenative annulation between 2-(1H-indol-2-yl)phenols and alkenylphenols is presented. Various indole-fused benzoxepines can be obtained at room temperature using atom-efficient strategies. This method not only avoids the
Kui Dong (8747232) +3 more
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Electronic substitution effect on the ground and excited state properties of indole chromophore: A computational study [PDF]
, 2022 Indole, being the main chromophore of amino acid tryptophan and several other biologically relevant molecules like serotonin, melatonin, has prompted considerable theoretical and experimental interest.
Padmabati, Mondal, Soumyadip, Ray
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Organocatalytic Enantioselective Nucleophilic Addition of Indole Imine 5-Methides [PDF]
, 2023 Despite the enormous developments in the asymmetric transformations of indole imine methides (IIMs), the remote asymmetric induction involving IIMs remains challenging due to the spatial interaction requirement between the substrate and catalyst.
Jianwei, Sun +5 more
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Indole-2-carboxamide Inhibitors of Human Liver Glycogen Phosphorylase† [PDF]
, 2016 Indole-2-carboxamide Inhibitors of Human Liver Glycogen Phosphorylase†
Dennis J. Hoover (1878532) +9 more
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Crystals, 2020 The designed target compound of N-acetyl indole linked to a fused triazolo/thiadiazole scaffold was synthesized via the reaction of 4-amino-5-(1H-indol-2-yl)-1,2,4-triazol-3(2H)-thione as the starting material with acetic anhydride under reflux ...
Ahmed T. A. Boraei +4 more
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Indole-3-carbinol ameliorated the isoproterenol-induced myocardial infarction via multimodal mechanisms in Wistar rats [PDF]
, 2022 The present study investigated the cardioprotection of Indole-3-carbinol on isoproterenol (ISO)-induced myocardial infarction in Wistar rats. I3C treatment significantly reduced the prolongation of the QRS complex, QT interval, and ST-segment elevation ...
Sairam Krishnamurthy (5874050) +1 more
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Plants, 2019 Selenium (Se) is an essential micronutrient for human health, entering the diet mainly through the consumption of plant material. Members of the Brassicaceae are Se-accumulators that can accumulate up to 1g Se kg−1 dry weight (DW) from the ...
Marian McKenzie +6 more
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Increasing sustainability in pork production by using high inclusion levels of co-products distillers dried grains with solubles, wheat middling and canola meal doesn’t affect pig growth performance and meat quality but reduces boar taint [PDF]
Animal Bioscience, 2023 Objective The present study is to examine the effect of high inclusion of co-products in pig diets (referred to as an alternative diet) during the finishing stage on pig growth performance, meat quality and boar taint compounds. Methods Growing pigs were
Thanh T. Nguyen +5 more
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