Results 141 to 150 of about 17,613 (213)

Synthesis of isoxazoles and their hydrazinolysis to 5-aminopyrazoles: an approach to fluorescent derivatives. [PDF]

RSC Adv
Ríos MC, Ladino-Bejarano A, Miscione GP, Portilla J.   +3 more
europepmc   +1 more source

PyMolGen: Database-Driven Molecular Generation of Drug-Like Compounds. [PDF]

J Chem Inf Model
Falcone BN, Hutcheon MJ, Zaidi JM, Stocks MJ, Hamill KE, Jamieson C, Williams HJ, Palmer DS, Baxter A, Pickett SD, Hirst JD.   +10 more
europepmc   +1 more source

Synthesis and bioactivity evaluation of isoxazoline scaffolds using heterogeneous photocatalytic (3+2) cycloaddition. [PDF]

J Adv Res
Li S, Liu B, Chen X, Wang G, Zhang C, Ma S, Li Y.   +6 more
europepmc   +1 more source

A Review on Farnesoid X Receptor (FXR) Modulators Focusing on Benzimidazole Scaffold. [PDF]

Molecules
Teno N, Gohda K, Fujimori K.
europepmc   +1 more source

Structure-Guided Optimization and Biological Validation of 1,3,4-Thiadiazole-Based SIRT2 Inhibitors Reinforcing Channel Entrance Interactions. [PDF]

Drug Dev Res
Aksel AB, Ozgencil F, Bakar-Ates F, Gunindi HB, Massarotti A, Ozkan E, Kaya SG, Gozelle M, Ozkan Y, Eren G.   +9 more
europepmc   +1 more source

Biocatalytic Synthesis of Isoxazolines Enabled by Cryptic Nitrile Oxide Formation by a Vanadium-Dependent Chloroperoxidase. [PDF]

Angew Chem Int Ed Engl
Sharma M, Biegasiewicz KF.
europepmc   +1 more source

Synthesis of Isoxazole- and Oxazole-4-carboxylic Acids Derivatives by Controlled Isoxazole-Azirine-Isoxazole/Oxazole Isomerization

The Journal of Organic Chemistry, 2019
The first synthesis of isoxazole-4-carboxylic acid derivatives by domino isoxazole-isoxazole isomerization is reported. Fe(II)-catalyzed isomerization of 4-acyl-5-methoxy-/5-aminoisoxazoles (dioxane, 105 °C) leads to the formation of isoxazole-4-carboxylic esters and amides in good yields. 4-Formyl-5-methoxyisoxazoles give methyl oxazole-4-carboxylates
Anna V. Serebryannikova, Ekaterina E. Galenko, Mikhail S. Novikov, Alexander F. Khlebnikov   +3 more
core   +4 more sources

Isoxazole Hydrate

Canadian Journal of Chemistry, 1974
X-Ray, n.m.r., and dielectric studies show that the hydrate of isoxazole is a typical type II clathrate hydrate in structure, in reorientation rates of host and guest molecules, and in composition.
Gough, S.R., Garg, S.K., Ripmeester, J.A., Davidson, D.W.   +3 more
openaire   +3 more sources

Design and Synthesis of Novel Isoxazole-Based HDAC Inhibitors

European Journal of Medicinal Chemistry, 2010
A series of isoxazole-based histone deacetylase (HDAC) inhibitors structurally related to SAHA were designed and synthesized. The isoxazole moiety was inserted in the vicinity of the Zn2+-binding group in order to check its participation in the ...
Ciro Mercurio, Roberta Ettari, Andrea Pinto   +2 more
exaly   +2 more sources

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Isoxazole anthelmintics

Journal of Medicinal Chemistry, 1977
A series of 3-halo-5-phenyl- and 3-phenyl-5-haloisoxazoles has demonstrated anthelmintic activity at doses ranging from 16 to 500 mg/kg orally against the rat roundworm, Nippostrongylus braziliensis. In the 5-phenyl series a halogen at the 3 position of the isoxazole ring was required for activity.
J B, Carr, H G, Durham, D K, Hass
openaire   +2 more sources