Results 151 to 160 of about 24,259 (231)

5-(Thiophen-2-yl)isoxazoles as novel anti-breast cancer agents targeting ERα: synthesis, <i>in vitro</i> biological evaluation, <i>in silico</i> studies, and molecular dynamics simulation. [PDF]

RSC Med Chem
Pattanayak P, Nikhitha S, Halder D, Ghosh B, Chatterjee T.   +4 more
europepmc   +1 more source

Design, synthesis, and biological evaluation of phenylisoxazole-based histone deacetylase inhibitors. [PDF]

PLoS One
Qin X, Han M, Hu P, Que H, Shao Z, Yan D.   +5 more
europepmc   +1 more source

Regioselective Synthesis of 5-Substituted 3-(β-d-Glycopyranosyl)isoxazoles and -isoxazolines by 1,3-Dipolar Cycloaddition as Potential Anticancer Agents and Glycogen Phosphorylase Inhibitors. [PDF]

Int J Mol Sci
Kaszás T, Szakács B, Bertalan M, Blága T, Hameed F, Lengyel Á, Saifi S, Juhász-Tóth É, Varga LA, Docsa T, Sipos A, Bai P, Ábrahám A, Kiss-Szikszai A, Kun S, Kiss GA, József J, Juhász L, Tóth M.   +18 more
europepmc   +1 more source

Design, synthesis, characterization, and theoretical calculations, along with in silico and in vitro antimicrobial proprieties of new isoxazole-amide conjugates

Open Chemistry
Barghady Najoua, Assou Soumia Ait, Er-Rajy Mohammed, Boujdi Khalid, Arzine Aziz, Rhazi Yassine, Tüzün Burak, Nakkabi Asmae, Chalkha Mohammed, El Hassouni Mohammed, Kabra Atul, Alanazi Mohammed M., Baouid Abdesselam, El Yazidi Mohamed   +13 more
doaj   +1 more source

Novel and efficient synthesis of 5-chloro-6-methoxy-3-(2-((1-(aryl)-1<i>H</i>-1,2,3-triazol-4-yl)methoxy)ethyl)benzo[<i>d</i>]isoxazole derivatives as new <i>α</i>-glucosidase inhibitors. [PDF]

Biochem Biophys Rep
Mudireddy RR, Gundla R, Koraboina CP, Velavalapalli VM, Sarma Dhulipalla VV, Burle GS, Jonnalagadda SB, Katari NK.   +7 more
europepmc   +1 more source

Pharmacometabolomics Study of Sulfamethoxazole and Trimethoprim in Kidney Transplant Recipients: Real-World Metabolism and Urinary Excretion. [PDF]

Metabolites
Hof MAJ, de Haan H, Stepanovic S, Bakker SJL, Hak E, Hopfgartner G, Klont F, Investigators T.   +7 more
europepmc   +1 more source

Bioactivity of novel isoxazole-fused heterocycles: comprehensive antimicrobial, antioxidant activities, SwissADME predictions, molecular docking, and DFT analysis. [PDF]

Mol Divers
Reheim MAMA, Abdou MM, El-Gaby MSA, Al-Omari MH, Abu-Rayyan A, Al-Assy WH, Refat HM, Sarhan AAM, Hafiz ISA.   +8 more
europepmc   +1 more source

Neuronal Differentiation of GBM-Initiating Cells Combined with Elimination of Undifferentiated Cells Preserves Motor Function. [PDF]

Cells
Chen Z, Zou P, Kondo T.
europepmc   +1 more source

Development of a Late-Stage Functionalization Strategy to Access Diverse 3,5-Disubstituted 1,2,4-Thiadiazoles. [PDF]

J Org Chem
Dobria A, Petros ZA, Mickel P, Aldrich LN.   +3 more
europepmc   +1 more source

Regulating AMPA Receptors with Isoxazole-4-Carboxamide Derivatives: An Electrophysiological Study. [PDF]

J Xenobiot
Qneibi M, Hawash M, Bdir S, Bdair M, Idais T, Sarhan I, Touqan J.   +6 more
europepmc   +1 more source