Results 31 to 40 of about 43,444 (345)

On-Demand Detachment of Maleimide Derivatives on Cysteine to Facilitate (Semi)Synthesis of Challenging Proteins [PDF]

, 2020
The maleimide group is a widely used reagent for bio-conjugation of peptides, proteins and oligonucleotides employing Michael addition and Diels-Alder cycloaddition reactions.
Guy, Mann, Ganga B., Vamisetti, Michael H., Glickman, ashraf, brik, satish, gandhesiri, Prasad, Sulkshane   +5 more
core   +2 more sources

Natural Product-Based Pesticide Discovery: Design, Synthesis and Bioactivity Studies of N-Amino-Maleimide Derivatives

Molecules, 2018
Natural products are an important source of pesticide discovery. A series of N-amino-maleimide derivatives containing hydrazone group were designed and synthesized based on the structure of linderone and methyllinderone which were isolated from Lindera ...
Xiangmin Song, Chunjuan Liu, Peiqi Chen, Hao Zhang, Ranfeng Sun   +4 more
doaj   +1 more source

Maleimide-functionalized poly(2-ethyl-2-oxazoline): Synthesis and reactivity [PDF]

, 2016
Poly(2-ethyl-2-oxazoline)s (PEtOx23 - Mn = 2300 g mol-1, D = 1.07; PEtOx46 - Mn = 4400 g mol-1, D = 1.06) end-functionalized with a maleimide moiety were prepared from azide-terminated PEtOxx-N3via copper-catalyzed azide-alkyne cycloaddition (CuAAC) with
Wendler, Felix, Barner-Kowollik, C., Görls, H., Schacher, F. H., Jasinski, Nils, Wendler, F., Jasinski, N., Schacher, Felix H., Trouillet, V., Trouillet, Vanessa, Rudolph, T., Görls, Helmar, Barner-Kowollik, Christopher, Rudolph, Tobias   +13 more
core   +1 more source

Stereoselective synthesis of fused tetrahydroquinazolines through one-pot double [3 + 2] dipolar cycloadditions followed by [5 + 1] annulation

Beilstein Journal of Organic Chemistry, 2016
The one-pot [3 + 2] cycloaddition of an azomethine ylide with a maleimide followed by another [3 + 2] cycloaddition of an azide with the second maleimide gives a 1,5-diamino intermediate which is used for a sequential aminomethylation reaction with ...
Xiaofeng Zhang, Kenny Pham, Shuai Liu, Marc Legris, Alex Muthengi, Jerry P. Jasinski, Wei Zhang   +6 more
doaj   +1 more source

Fluorinated maleimide-substituted porphyrins and chlorins: synthesis and characterization

Beilstein Journal of Organic Chemistry, 2019
Maleimide-containing fluorinated porphyrins and chlorins were prepared based on the reaction of Zn(II) or Ni(II) complexes of 5,10,15,20-tetrakis(4-amino-2,3,5,6-tetrafluorophenyl)porphyrin and chlorin with maleic anhydride.
Valentina A. Ol’shevskaya, Elena G. Kononova, Andrei V. Zaitsev   +2 more
doaj   +1 more source

Maleimido-Functionalized NOTA Derivatives as Bifunctional Chelators for Site-Specific Radiolabeling

Molecules, 2011
Two basic and simple synthetic routes for mono- and bis-maleimide bearing 1,4,7-triazacyclononane-N,N’,N’’-triacetic acid (NOTA) chelators as new bifunctional chelators are described. The syntheses are characterized by their simplicity and short reaction
Jörg Steinbach, Christian Förster, Maik Schubert, Hans-Jürgen Pietzsch   +3 more
doaj   +1 more source

Maleimide-modification reaction parameters^a.

, 2016
Maleimide-modification reaction parametersa.
Christopher G. Rowe (3181443), Beth Chen (3181440), Yimin Wu (130710), David L. Narum (130745), David S. Jones (633681), Karine Reiter (320322), Kelly M. Rausch (320326), Patrick E. Duffy (155813)   +7 more
core   +1 more source

Evaluation of Antifibrotic Mechanisms of 3′5-Dimaleamylbenzoic Acid on Idiopathic Pulmonary Fibrosis: A Network Pharmacology and Molecular Docking Analysis

Drugs and Drug Candidates
Background: Idiopathic pulmonary fibrosis (IPF) is a chronic, disabling disorder of unknown etiology, poor prognosis, and limited therapeutic options. Previously, 3′5-dimaleamylbenzoic acid (3′5-DMBA) was shown to exert resolving effects in IPF, offering
Karina González-García, Jovito Cesar Santos-Álvarez, Juan Manuel Velázquez-Enríquez, Cecilia Zertuche-Martínez, Edilburga Reyes-Jiménez, Rafael Baltiérrez-Hoyos, Verónica Rocío Vásquez-Garzón   +6 more
doaj   +1 more source

N-(4-Chlorophenyl)maleimide [PDF]

Acta Crystallographica Section E Structure Reports Online, 2008
في مركب العنوان، C(10)H(6) ClNO (2)، تبلغ الزاوية الثنائية السطوح بين حلقات البنزين والماليميد 47.54 (9) درجة. تشكل جزيئات المول دايمرات متماثلة مركزيًا من خلال روابط هيدروجينية C-H O، مما يؤدي إلى حلقات من عزر مجموعة الرسم البياني R(2) (2) (8) وسلاسل في اتجاه [100]. ترتبط جزيئات المول أيضًا بروابط هيدروجينية C-H- Cl على طول [001]. في هذا الاتجاه نفسه،
Rodolfo Moreno‐Fuquen, Zulay Pardo-Botero, Javier Ellena   +2 more
openaire   +3 more sources

A pyrene maleimide with a flexible linker for sampling of longer inter-thiol distances by excimer formation. [PDF]

PLoS ONE, 2011
Pyrene-containing compounds are commonly used in a number of fluorescence-based applications because they can form excited-state dimers (excimers) by stacking interaction between excited-state and ground-state monomers.
Satomi Niwayama, Abdullatif S Kassar, Tian Zhao, Roger B Sutton, Guillermo A Altenberg   +4 more
doaj   +1 more source