An Overview of Bioactive 1,3-Oxazole-Containing Alkaloids from Marine Organisms
Pharmaceuticals, 2021 1,3-Oxazole chemicals are a unique class of five-membered monocyclic heteroarenes, containing a nitrogen atom and an oxygen. These alkaloids have attracted extensive attention from medicinal chemists and pharmacologists owing to their diverse arrays of ...
Jinyun Chen +5 more
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Recent Advances in the Synthesis of Oxazole-Based Molecules via van Leusen Oxazole Synthesis
Molecules, 2020 Oxazole compounds, including one nitrogen atom and one oxygen atom in a five-membered heterocyclic ring, are present in various biological activities. Due to binding with a widespread spectrum of receptors and enzymes easily in biological systems through
Xunan Zheng, Wei Liu, Dawei Zhang
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A comprehensive review on biological activities of oxazole derivatives
BMC Chemistry, 2019 The utility of oxazole as intermediates for the synthesis of new chemical entities in medicinal chemistry have been increased in the past few years. Oxazole is an important heterocyclic nucleus having a wide spectrum of biological activities which drew ...
Saloni Kakkar +1 more
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Neue Bildungsweise der Oxazole [PDF]
Berichte der deutschen chemischen Gesellschaft, 1896 Bei dem Versuch, das Benzaldehydcyanhydrin mit Acetochlor-hydrose in atherischer Losung durch Salzsaure zu einem Glucosid zu vereinigen, wurde ein schon krystallisirtes chlorhaltiges Product gewonnen, an dessen Bildung die Acetochlorhydrose nicht betheiligt ist.
Emil Fischer
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Polarizability in Substituted Oxazoles: A PC-Model Data Analysis [PDF]
E-Journal of Chemistry, 2005 A systematic investigation of various Oxazole derivatives has been subjected to a Polarized Continuums Model (PCM) for evaluation of their physico-chemical parameters.
S. Harikrishna +3 more
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Crystal structure and Hirshfeld-surface analysis of the pesticide etoxazole [PDF]
Acta Crystallographica Section E: Crystallographic CommunicationsEtoxazole (C21H23F2NO2), systematic name 4-(4-tert-butyl-2-ethoxyphenyl)-2-(2,6-difluorophenyl)-4,5-dihydro-1,3-oxazole, is a fluorinated insecticide and acaricide that inhibits chitin biosynthesis, disrupting insect development by preventing proper ...
Chaluvarangaiah Sowbhagya +3 more
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Performance Analysis Of Regularized Linear Regression Models For Oxazolines And Oxazoles Derivitive Descriptor Dataset [PDF]
published International Journal of Computational Science and
Information Technology (IJCSITY) Vol.1, No.4, November 2013, 2013 Regularized regression techniques for linear regression have been created the last few ten years to reduce the flaws of ordinary least squares regression with regard to prediction accuracy. In this paper, new methods for using regularized regression in model choice are introduced, and we distinguish the conditions in which regularized regression ...
Chanabasayya .M
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Naturally Occurring Oxazole-Containing Peptides [PDF]
Marine Drugs, 2020 Oxazole-containing peptides are mostly of marine origin and they form an intriguing family with a broad range of biological activities. Here we classify these peptides on the basis of their chemical structure and discuss a number of representatives of each class that reflect the extraordinary potential of this family as a source of new drugs.
Jessica T. Mhlongo +4 more
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Design, Synthesis, In Vitro Biological Evaluation and In Silico Molecular Docking Study of Benzimidazole-Based Oxazole Analogues: A Promising Acetylcholinesterase and Butyrylcholinesterase Inhibitors [PDF]
Molecules, 2023 Alzheimer’s disease (AD) is a degenerative neurological condition that severely affects the elderly and is clinically recognised by a decrease in cognition and memory.
Rafaqat Hussain +7 more
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Synthesis of tricarbonylated propargylamine and conversion to 2,5-disubstituted oxazole-4-carboxylates [PDF]
Beilstein Journal of Organic ChemistryThe N,O-acetal derived from diethyl mesoxalate (DEMO) undergoes elimination of acetic acid upon treatment with a base, leading to the formation of N-acylimine in situ.
Kento Iwai +5 more
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