Results 191 to 200 of about 37,707 (289)

Synthetic Study on the Piperidine Alkaloids

, 1979
Mitsutaka Natsume, Masashi Ogawa
openalex   +1 more source

Aliphatische Flüssigkristalle, IV [1] Synthese einiger 1-(1,3-Dioxan-2- und -5-yl)piperidine / Aliphatic Liquid Crystals, IV [1] Synthesis of Some 1-(1.3-Dioxan-2- and -5-yl)Piperidines [PDF]

, 1985
Wolfgang Sucrow, Ronald Lüschen, Annette Risse   +2 more
openalex   +1 more source

Further SAR of GIRK1/2 activators: Synthesis and Biological Characterization of In Vitro Tool Compounds

ChemMedChem, Accepted Article.
The work presented herein outlines the ongoing structure‐activity relationship (SAR) studies centered around a potent, efficacious, and selective activators of the GIRK1/2 channel. Optimization studies centered around the pyrazole privileged scaffold, the N‐1‐position of the pyrazole and the right‐hand ether.
Sumaiya Nahid, Fahad Imtiaz Rahman, Yu Du, Brittany Spitznagel, Sandeep K Singh, Yashpal Chhonker, Daryl J Murry, David Weaver, Corey R Hopkins   +8 more
wiley   +1 more source

Base-Labile Safety-Catch Linker: Synthesis and Applications in Solid-Phase Peptide Synthesis. [PDF]

Int J Mol Sci
Noki S, Saneii H, de la Torre BG, Albericio F.   +3 more
europepmc   +1 more source

Aromatic Nucleophilic Substitution. XIII. Confirmation of the Anionic σ Complexes in the Reactions of 2,4-Dinitro- and 2,4,5-Trinitro-1-(1-piperidyl)naphthalenes with Piperidine in Dimethyl Sulfoxide [PDF]

, 1980
Shizen Sekiguchi, Reiko Hikage, Kenmi Obana, Kohji Matsui, Yumiko Ando, Noboru Tomoto   +5 more
openalex   +1 more source

Novel para‐phenylenediamine‐based derivatives as Receptor Tyrosine Kinase‐like Orphan Receptor 1 (ROR1) Inhibitors: An in vitro preliminary characterization

ChemMedChem, Accepted Article.
ROR1 kinase is an underexplored promising target for the development of novel anticancer drugs, being strongly expressed in several cancer cell lines, but poorly in non‐tumor cells. This property, together with the scarce number of molecules effective against ROR1, led us to design and develop a research program aimed to the discovery of new chemical ...
Gerardina Smaldone, Maria Rosaria Miranda, Francesca Di Matteo, Valeria Napolitano, Michela Aliberti, Simona Musella, Veronica Di Sarno, Gianluigi Lauro, Giuseppe Bifulco, Giacomo Pepe, Giovanna Aquino, Mario Felice Tecce, Isabel Maria Gomez-Monterrey, Pietro Campiglia, Carmine Ostacolo, Alessia Bertamino, Vincenzo Vestuto, Tania CIAGLIA   +17 more
wiley   +1 more source

Sustainable Ultrasound-Assisted Solid-Phase peptide synthesis (SUS-SPPS): Less Waste, more efficiency. [PDF]

Ultrason Sonochem
Mottola S, Bene AD, Mazzarella V, Cutolo R, Boccino I, Merlino F, Cosconati S, Maro SD, Messere A.   +8 more
europepmc   +1 more source

Lactams. XI. Construction of lactam carbonyl function in 1,3-disubstituted piperidines by mercuric acetate-EDTA oxidation: Effects of carbonyl and related groups at the 3-position.

, 1977
Tozo Fujii, Masashi Ohba, Shigeyuki Yoshifuji   +2 more
openalex   +2 more sources

Synthesis and Pharmacology of N-Substituted-4-(p-Metboxypbenyl) Piperidine-2,6-diones [PDF]

, 1980
S. D. SAMANT, K. D. DEODHAR
openalex   +1 more source

Wettability‐Controlled Electrocatalytic Carbon Dioxide Reduction

Chemistry–Methods, EarlyView.
Herein, the evolution of catalytic interface configurations in eCO2RR is introduced, outlines the major challenges associated with constructing stable and efficient TPIs, and summarize recent advancements, such as hydrophobic polymer/molecular modifications and hierarchical structure fabrication to improve hydrophobicity.
Lanze Li, Jiexin Wen, Tsz Woon Benedict Lo, Jun Yin, Qiong Lei   +4 more
wiley   +1 more source