Results 81 to 90 of about 645,171 (161)

Administration of a recombinant secretory leukocyte protease inhibitor prevents aortic aneurysm growth in mice. [PDF]

Mol Cell Biochem
Yamawaki-Ogata A, Mutsuga M, Narita Y.
europepmc   +1 more source

Preclinical characterization of EGT710, an oral non-peptidomimetic reversible covalent SARS-CoV-2 main protease inhibitor. [PDF]

NPJ Drug Discov
Moquin SA, Lakshminarayana SB, Balavenkatraman KK, Schiller H, Claas A, Bhhatarai B, Loisios-Konstantinidis I, Vulic K, Kurhade C, Kalveram BK, Chen JY, Zou J, Xie X, Tandeske L, Dovala D, Ornelas E, Knapp MS, Fuller D, Nguyen Z, Barkan DT, Bebrevska L, Wright SK, Busby SA, Blais J, Shi PY, Gaudet S, Bergeron R, Yu H, Zack J, Sarko C, Gu F, Bradner JE, Tallarico JA, Diagana TT, Papillon JPN.   +34 more
europepmc   +1 more source

Production of human cathepsins using Expi293™ mammalian cell expression system for off-target activity of cysteine protease inhibitor screening. [PDF]

Protein Sci
Turner Z, Arutyunova E, Bui DT, Han L, Kandadai AS, Bai B, Young HS, Mahal LK, Klassen JS, Lemieux MJ.   +9 more
europepmc   +1 more source

Expression and purification of a broad-spectrum human protease inhibitor in <i>Pichia pastoris</i>. [PDF]

Biochem Biophys Rep
Bhakta V, Tehrani NC, Ask A, Sheffield WP.   +3 more
europepmc   +1 more source

Immunoregulation mediated by the enzyme inhibitory activity of helminth-derived serine protease inhibitor affects the protective efficiency of vaccines. [PDF]

Virulence
Shi W, Liu Y, Bai X, Liang Y, Zhang S, Sun L, Lin W, Liu X, Xu N.   +8 more
europepmc   +1 more source

Serine protease inhibitor dipetalogastin-like from Galleria mellonella is involved in insect immunity. [PDF]

Sci Rep
Kordaczuk J, Sułek M, Mak P, Pawlikowska-Pawlęga B, Wojda I.   +4 more
europepmc   +1 more source

Ligand Versatility and Resistance Mechanism of Monotherapy-Grade HIV-1 Protease Inhibitor GRL-142 Binding the Multidrug Resistant Variant p51: Insights from 1 μs MD Simulations. [PDF]

J Chem Inf Model
Arias A, Cappelli C, Restrepo A, Alí-Torres J, Gómez S.   +4 more
europepmc   +1 more source

Anti-Melanoma Activity and Potential Mechanism of Purified Potato Protease Inhibitor. [PDF]

Foods
Li Q, Jiang L, Chen N, Wang X, Yao J, Su Z, Zhao S.   +6 more
europepmc   +1 more source

Drug Repurposing: Conversion of the Peripherally Restricted HIV Protease Inhibitor Amprenavir to Potent, Selective, and CNS-Penetrant Agonists for the Cannabinoid Receptor 2. [PDF]

J Med Chem
Haymer DH, Duncan RA, Rodriguez AL, Han A, Lindsay RJ, Wijesiri NK, Thompson Gray A, Krishnan S, Qi A, Brown BP, Boutaud O, Engers DW, Jones CK, Niswender CM, Lindsley CW, Bender AM.   +15 more
europepmc   +1 more source

Species-Dependent Metabolism of a Covalent nsP2 Protease Inhibitor with In Vivo Antialphaviral Activity. [PDF]

J Med Chem
Hossain MA, Mayo AK, Ghoshal A, Taft-Benz S, Anderson E, Morales NL, Pressey KD, Vargason A, Brouwer KLR, Moorman NJ, Heise MT, Willson TM.   +11 more
europepmc   +1 more source