Results 181 to 190 of about 36,678 (260)

Chemical tools for BAZ2A/B biology: discovery of dual and BAZ2B-selective PROTAC degraders. [PDF]

RSC Med Chem
Cheng-Sánchez I, Gosselé KA, Palaferri L, Krummhaar M, Laul E, Ciulli A, Nevado C.   +6 more
europepmc   +1 more source

Rational design, synthesis, and antimicrobial evaluation of novel 1,2,3-triazole hybrids: structure-activity relationships, molecular docking, and DFT studies. [PDF]

Sci Rep
Sallam MN, Hassan AMA, Alzahrani AYA, El-Masry HM, El-Naggar AM, Abbass EM.   +5 more
europepmc   +1 more source

Electricity-Controlled Divergent Synthesis of CF₃‑Tethered Pyrazolines and Pyrazoles via Tandem Radical Trifluoromethylation and Annulation. [PDF]

JACS Au
Pattanayak P, Girase YK, Chatterjee T.
europepmc   +1 more source

Synthesis, molecular docking and biological evaluation of 2,4-diaminopyrimidines and pyrazoles as aurora kinase inhibitors. [PDF]

EXCLI J
Sankhe K, Jadhav M, Prabhu A, Khan T.
europepmc   +1 more source

Multicomponent Selective and Efficient Synthesis of Spiro[furo[2,3-<i>d</i>]pyrimidine-6,4'-pyrazole] Scaffold Under a Column Chromatography-Free Protocol at Room Temperature. [PDF]

Molecules
Elinson MN, Ryzhkova YE, Kalashnikova VM, Egorov MP.   +3 more
europepmc   +1 more source

Investigating the Inhibitory Properties of Diazo and Pyrazole-Carboxamide-Linked Benzenesulfonamides Against Carbonic Anhydrase Isoforms I, II, IX, and XII. [PDF]

ChemMedChem
Akocak S, Lolak N, Ammara A, Gürbüz G, Bozgeyik I, Taşdemir D, Hashem H, Bräse S, Supuran CT.   +8 more
europepmc   +1 more source

Electrochemical oxidative amidation of alcohols towards <i>N</i>-acyl azoles as precursors for amides, esters and thioesters.

Org Biomol Chem
Bartels IMA, Witte MD, Minnaard AJ.
europepmc   +1 more source

Design, synthesis, biological assessment, and integrated computational analysis of new pyrazole-based antimicrobial candidates. [PDF]

Sci Rep
El-Helw EAE, Hamed S, El-Ziaty AK, Alzahrani AYA, Ramadan SK.   +4 more
europepmc   +1 more source

Rational design of pyrazole-oxime hybrids as dual-targeting agents for glioma and breast cancer brain metastasis. [PDF]

Naunyn Schmiedebergs Arch Pharmacol
Gul M, Alagoz MA, Hepokur C, Algul O.
europepmc   +1 more source

Quinazolinone-diarylpyrazole hybrids as dual EGFR/COX-2 inhibitors: antiproliferative, mechanistic, and <i>in silico</i> studies. [PDF]

RSC Adv
Alkhammash A, Saleem BAA, Oudah KH, Ahmed M, Abass KS, Farhan SM, Zaki MEA, Gomha SM.   +7 more
europepmc   +1 more source