Optimization of Pyrazolo[3,4‑<i>b</i>]pyridine Analogues: Synthesis, In Vitro Anticancer Evaluation and In Vivo Pharmacokinetics. [PDF]
Georgiou M +8 more
europepmc +1 more source
Thiazole-driven heterocyclic hybrids as EGFR inhibitors: progress in synthesis and anticancer applications. [PDF]
Dsouza A, Subrahmanyam VM, Shetty NS.
europepmc +1 more source
Innovative Amino-Functionalization of Pyrido[2,3-<i>d</i>]pyrimidine Scaffolds for Broad Therapeutic Applications Supported by Computational Analyses. [PDF]
El-Hema HS +9 more
europepmc +1 more source
Pyrazole-Imidazoline Derivative Prevents Cardiac Damage and Mortality in Acute <i>Trypanosoma cruzi</i> Infection. [PDF]
Orlando LMR +9 more
europepmc +1 more source
Accessing trifluoromethylated SuFEx-able pyrazole <i>via</i> distortion-accelerated 1,3-dipolar cycloadditions. [PDF]
Khanal B, Feliciano MAM, Gold B.
europepmc +1 more source
Biocatalyzed aza-michael addition <i>via</i> continuous flow technology: a game-changer for the facile synthesis of <i>N-</i>alkylated pyrazole derivatives. [PDF]
Du LH, Yan BL, Xue MM, Wang L, Luo XP.
europepmc +1 more source
Triazole and Pyrazole Hybrids of Electrophilic Natural Products as Promising Anticancer Agents. [PDF]
Fermo AD +4 more
europepmc +1 more source
Synthesis, antiproliferative screening, and molecular docking of some heterocycles derived from N-(1-(5-chloro-3-methyl-1-phenyl-1H-pyrazol-4-yl)-3-hydrazineyl-3-oxoprop-1-en-2-yl)benzamide. [PDF]
El-Helw EAE +6 more
europepmc +1 more source
Discovery of Pyrazoline Benzenesulfonamide Derivatives as Anticancer Agents: A Review. [PDF]
Hasyim DM +5 more
europepmc +1 more source

