Results 171 to 180 of about 7,109 (211)
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Thiazolyl-pyrazole derivatives as potential antimycobacterial agents
Bioorganic & Medicinal Chemistry Letters, 2019Mycobacterium tuberculosis (Mtb) is an obligate aerobe that is capable of long-term persistence under conditions of low oxygen tension. A series of thiazolyl-pyrazole derivatives (6a-f, 7a-f, 8c, 8e) were screened for antimycobacterial activity against dormant M. tuberculosis H37Ra (D-MTB) and M. bovis BCG (D-BCG).
Sushma J. Takate +6 more
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Novel pyrazole-5-carboxamide and pyrazole–pyrimidine derivatives: Synthesis and anticancer activity
European Journal of Medicinal Chemistry, 2015A series of novel pyrazole-5-carboxamide and pyrazole-pyrimidine derivatives were designed and synthesized. All compounds have been screened for their antiproliferative activity against MGC-803, SGC-7901 and Bcap-37 cell lines in vitro. The results revealed that compounds 8a, 8c and 8e exhibited strong inhibitory activity against MGC-803 cell line. The
Jing Bo, Shi +4 more
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PYRAZOLE DERIVATIVES AS PSYCHOPHARMACEUTICALS
2003The invention relates to pyrazole derivatives of Formula (I), in which ...
MERCK PATENT GMBH +4 more
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Synthesis and Antimalarial Activity of Substituted Pyrazole Derivatives
Arzneimittelforschung, 2002AbstractFor Abstract see ChemInform Abstract in Full Text.
José N, Domínguez +3 more
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2001
The present invention relates to certain pyrazole derivatives of Formula (I) that are p-38 MAP kinase inhibitors, pharmaceutical compositions containing them, methods for their use, and methods for preparing these compounds.
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The present invention relates to certain pyrazole derivatives of Formula (I) that are p-38 MAP kinase inhibitors, pharmaceutical compositions containing them, methods for their use, and methods for preparing these compounds.
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PESTICIDAL 5- (ACYLAMINO) PYRAZOLE DERIVATIVES
2004Substituted-acylaminopyrazole derivatives of formula (I) or salts thereof wherein the various symbols are as defined in the description, processes for their preparation, compositions thereof, and their use for the control of pests, such as anthropods, (e.g. insects and arachnids) and helminths.
BAYER CROPSCIENCE SA +8 more
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Integrative oncology: Addressing the global challenges of cancer prevention and treatment
Ca-A Cancer Journal for Clinicians, 2022Jun J Mao,, Msce +2 more
exaly