Results 161 to 170 of about 17,768 (339)
Flexibility of the pyrrolidine ring in proline peptides [PDF]
Vincent Madison
openalex +1 more source
Andrographolide (ADG) was conjugated with MOFs (MIL‐53(Al), ZIF‐8) carbon‐based quantum dots (CBQDs) and doped carbon‐based quantum dots (D‐CBQDs) using the green approach of high‐pressure (0.3 GPa) solid phase contact. This method enhances the drug solubility, as indicated by changes in hydrophobicity observed via 1H NMR. Abstract Andrographolide (ADG)
Wenndy Pantoja‐Romero+5 more
wiley +1 more source
Abstract Cryptocaryon irritans, one of the most devastating holotrichous ciliated protozoans, causes massive economic losses in the pompano, Trachinotus ovatus, mariculture industries. Considering the many advantages of phytochemicals, such as low cost, low residuals, and low pollution, they can be a good alternative for the prevention and control of C.
Wei‐Wei Mao+9 more
wiley +1 more source
Advances in Mechanochemical Methods for One‐Pot Multistep Organic Synthesis
Mechanochemical synthesis has emerged as a powerful and more sustainable alternative to conventional solution‐based methods, offering advantages such as no or only minimal solvent use, reduced reaction times, and simplified operational conditions.
Michael Schnürch, Nina Biedermann
wiley +1 more source
Piperidines from acid-catalysed cyclisations: Pitfalls, solutions and a new ring contraction to pyrrolidines [PDF]
Aldmairi, Abdu H.+4 more
core +2 more sources
Stereodivergent Synthesis of Multisubstituted Pyrrolidines via Metal-Catalyzed (3+2) Cycloaddition [PDF]
中央⼤学博士(工学)【学位授与の要件】中央大学学位規則第4条第1項 【論文審査委員主査】福澤 信一(中央大学理工学部教授) 【論文審査委員副査】石井 洋一(中央大学理工学部教授)、小松 晃之(中央大学理工学部教授)、山田 徹(慶應義塾大学理工学部教授)、工藤 一秋(東京大学生産技術研究所教授)doctoral ...
FURUYA,Shohei+2 more
core
Computational Analysis of the Stereoselective Synthesis of Substituted Pyrrolidines [PDF]
In this work we use computational methods to study the aza-Cope-Mannich tandem reaction of a substituted oxazolidine to form a formyl pyrrolidine. Pyrrolidine structural motifs are found in natural products, pharmaceutical compounds, and chiral catalysts.
Jones, Diamond T.
core +2 more sources
High‐throughput asymmetric reaction development of an organocatalytic Michael addition is achieved by using a readily available isatin molecule as amine protecting group, reagent for reactivity Umpolung, and as chiroptical yield and enantioselectivity reporter.
F Safia Kariapper+2 more
wiley +1 more source
The convergent synthesis of Lewis‐X‐containing betulinic acid and echinocystic acid saponins (1 and 2) is presented. The synthetic saponins were shown to inhibit, at the low micromolar range, the DC‐SIGN‐ and L‐SIGN‐mediated transfer of HIV‐1 infection to CD4‐positive cells, whereas free Lewis‐X, aglycones, and structurally similar triterpenoid ...
Oscar Javier Gamboa Marin+5 more
wiley +1 more source