A straightforward, gold‐catalyzed cycloisomerization of aromatic propargylamines is reported, enabling efficient access to quinoline and tetrahydroquinoline derivatives. Hexafluoroisopropanol acts as both solvent and activator, eliminating the need for silver salts or additives.
Efstathios Tonis +6 more
wiley +1 more source
Exploring insecticidal activity and SAR study of newly synthesized Benzo[h]quinoline-based heterocycles against Aphis craccivora Koch. and Culex pipiens L. Larvae. [PDF]
El-Helw EAE +3 more
europepmc +1 more source
New phosphino tricarbonylrhenium(I) complexes have efficient red emission in the aggregate and solid states. The good photostability and the vast possibilities of chemical modifications make these Re‐based complexes the starting point of a new generation of red emitters with aggregation‐induced phosphorescence emission (AIPE) characteristics.
Valentine Guilbaud +8 more
wiley +1 more source
Gallium/Indium-Promoted [4 + 2] Annulation of 2‑Aminobenzonitriles with Alkynes and Dimerization of 2‑Aminobenzonitriles: One-Pot Access to 4‑Aminoquinolines and 4‑Amino-2-Arylquinazolines. [PDF]
Sakai N +4 more
europepmc +1 more source
Single‐boron coordination converts the strong [1,2,5]thiadiazolo[3,4‐g]quinoxaline (TQ) acceptor into a superior electron‐deficient building block. Subsequent donor engineering and planarity modulation yield BLD3 NPs with intense NIR‐II absorption and high photothermal efficiency for effective photoacoustic imaging‐guided tumor therapy. ABSTRACT Strong
Qing‐Yun Ni +9 more
wiley +1 more source
Dual-Site Acetylcholinesterase Inhibition and Multiscale Stability of Fused Quinoline Sulfonamides: A Chemoinformatic GA-MLR and Molecular Dynamics Study. [PDF]
Nilewar SS +11 more
europepmc +1 more source
Evaluation of Novel Cloxyquin Analogs for K2P18.1 Channel Modulation
5‐Chloro‐/5‐bromoquinolines reveal how subtle changes at the 8‐position of the quinoline scaffold tune activity at hK2P18.1 channels. Among 14 synthesized derivatives, benzaldimine 3d emerged as a new lead for activator optimization potentiating hK2P18.1 activity by around 60% at 100 µM.
Jasmin Sörgel +6 more
wiley +1 more source
Synchronizing O<sub>2</sub> adsorption and proton-coupled electron transfer in carboxylated quinoline-linked covalent organic frameworks to boost photocatalytic H<sub>2</sub>O<sub>2</sub> production. [PDF]
Wang H +9 more
europepmc +1 more source
Novel extremophilic tryptophanases (TnaAs) are tested in the synthesis of L‐tryptophan analogues. This study compares a thermophilic and a halophilic TnaA with E. coli TnaA as benchmark, from both structural and catalytic perspectives, revealing enhanced stability, and a broader substrate scope for the new homologues.
Fatemeh Aziziyan +6 more
wiley +1 more source
Identification and Validation of 3-Cyano-Quinoline Ligands Targeting Integrin-Linked Kinase (ILK). [PDF]
Greco FA +11 more
europepmc +1 more source

