Results 121 to 130 of about 36,400 (237)
An approach to prepare pyrido[2,1‐a]isoindoles via the cycloaddition of pyridine‐based 1,3‐dipoles and benzyne is described, offering modular access to a range of substituted products by systematic tuning of the dipole. A modular strategy for the synthesis of fused indolizine/isoindole hybrids, pyrido[2,1‐α]isoindoles, via cycloaddition of pyridine ...
Samira Taghizadeh Nodehi +2 more
wiley +1 more source
2-[(2,5-Di-methyl-phen-yl)amino]-quinoline-3-carb-oxy-lic acid. [PDF]
Ji X, Long S.
europepmc +1 more source
Conformational restriction strategies to increase the activity and selectivity of the STAT5b inhibitor Stafib‐2 are presented. The best conformationally restricted inhibitor Stafib‐2‐CR has threefold higher activity against STAT5b than Stafib‐2. A cell‐permeable prodrug of Stafib‐2‐CR inhibits phosphorylation of STAT5b in cultured human leukemia cells ...
Theresa Münzel +5 more
wiley +1 more source
Reprogramming RiPP scaffolds through skeletal editing unlocks chemical space. [PDF]
Ogawa H +8 more
europepmc +1 more source
2-[(2-Methyl-phen-yl)amino]-quinoline-3-carb-oxy-lic acid. [PDF]
Guo S, Long S.
europepmc +1 more source
A new series of structurally rich polyaromatic isonitriles is presented as photoredox catalysts. Their photophysical properties are investigated by UV–Vis absorption and fluorescence measurements, combined with experimental and theoretical studies to evaluate both ground‐ and excited‐state redox properties.
Cristina Martini +9 more
wiley +1 more source
Evaluation of Antiplasmodial Activity of Quinoline Derivatives Incorporating Arylnitro and Aminochalcone Moieties. [PDF]
Ariefta NR +3 more
europepmc +1 more source
In this article, we present a new modular approach for the synthesis of bulky monophosphine ligands by nucleophilic addition of Grignard reagents to peri‐phosphine isoindolium salts as stable building blocks. Outcompeting the established catalytic systems (PPh3)AuCl and (XPhos)AuCl, the phosphine gold complexes show high catalytic activity at low ...
Karl Georg Leistikow +9 more
wiley +1 more source
Structural Basis for Potent Inhibition of Human DHODH by Quinoline-4-carboxylic Acid Derivatives. [PDF]
de Oliveira Viana J +10 more
europepmc +1 more source

